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MILLER, Alita A, BUNDY, Gordon L, SWEENEY, Michael T, BAMMERT, Gary F, HAMEL, Judith C, FORD, Charles W, ZHONG, Wei-Zhu, GRABER, David R, MARTIN, Gary E, HAN, Fusen, DOLAK, Lester A, SEEST, Eric P, MOTT, John E, RUBLE, J. Craig, KAMILAR, Gregg M, PALMER, John R, BANITT, Lee S, HURD, Alexander R, BARBACHYN, Michael R, SKEPNER, Jill E, BOYLE, Timothy P, HARRIS, Douglas W, HROMOCKYJ, Alexander E, MAROTTI, Keith R, ZURENKO, Gary E, MUNZNER, Jennifer B
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Published in Antimicrobial Agents and Chemotherapy (01.08.2008)
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Novel 3-fluoro-6-methoxyquinoline derivatives as inhibitors of bacterial DNA gyrase and topoisomerase IV
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Published in Bioorganic & medicinal chemistry letters (01.08.2017)
Published in Bioorganic & medicinal chemistry letters (01.08.2017)
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Novel quinoline derivatives as inhibitors of bacterial DNA gyrase and topoisomerase IV
Mitton-Fry, Mark J., Brickner, Steven J., Hamel, Judith C., Brennan, Lori, Casavant, Jeffrey M., Chen, Michael, Chen, Tao, Ding, Xiaoyuan, Driscoll, James, Hardink, Joel, Hoang, Thuy, Hua, Erbing, Huband, Michael D., Maloney, Meghan, Marfat, Anthony, McCurdy, Sandra P., McLeod, Dale, Plotkin, Michael, Reilly, Usa, Robinson, Shaughn, Schafer, John, Shepard, Richard M., Smith, James F., Stone, Gregory G., Subramanyam, Chakrapani, Yoon, Kwansik, Yuan, Wei, Zaniewski, Richard P., Zook, Christopher
Published in Bioorganic & medicinal chemistry letters (15.05.2013)
Published in Bioorganic & medicinal chemistry letters (15.05.2013)
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Identification of Phenylisoxazolines as Novel and Viable Antibacterial Agents Active against Gram-Positive Pathogens
Barbachyn, Michael R, Cleek, Gary J, Dolak, Lester A, Garmon, Stuart A, Morris, Joel, Seest, Eric P, Thomas, Richard C, Toops, Dana S, Watt, William, Wishka, Donn G, Ford, Charles W, Zurenko, Gary E, Hamel, Judith C, Schaadt, Ronda D, Stapert, Douglas, Yagi, Betty H, Adams, Wade J, Friis, Janice M, Slatter, J. Gregory, Sams, James P, Oien, Nancee L, Zaya, Matthew J, Wienkers, Larry C, Wynalda, Michael A
Published in Journal of medicinal chemistry (16.01.2003)
Published in Journal of medicinal chemistry (16.01.2003)
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The synthesis and antibacterial activity of 1,3,4-Thiadiazole phenyl oxazolidinone analogues
Thomasco, Lisa M, Gadwood, Robert C, Weaver, Elizabeth A, Ochoada, Jason M, Ford, Charles W, Zurenko, Gary E, Hamel, Judith C, Stapert, Douglas, Moerman, Judy K, Schaadt, Ronda D, Yagi, Betty H
Published in Bioorganic & medicinal chemistry letters (01.12.2003)
Published in Bioorganic & medicinal chemistry letters (01.12.2003)
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Synthesis and biological evaluation of benzazepine oxazolidinone antibacterials
Johnson, Paul D., Aristoff, Paul A., Zurenko, Gary E., Schaadt, Ronda D., Yagi, Betty H., Ford, Charles W., Hamel, Judith C., Stapert, Douglas, Moerman, Judy K.
Published in Bioorganic & medicinal chemistry letters (01.12.2003)
Published in Bioorganic & medicinal chemistry letters (01.12.2003)
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Carbon–carbon-linked (pyrazolylphenyl)oxazolidinones with antibacterial activity against multiple drug resistant gram-positive and fastidious gram-negative bacteria
Lee, Chi Sing, Allwine, Debra A, Barbachyn, Michael R, Grega, Kevin C, Dolak, Lester A, Ford, Charles W, Jensen, Randy M, Seest, Eric P, Hamel, Judith C, Schaadt, Ronda D, Stapert, Douglas, Yagi, Betty H, Zurenko, Gary E, Genin, Michael J
Published in Bioorganic & medicinal chemistry (01.12.2001)
Published in Bioorganic & medicinal chemistry (01.12.2001)
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Nitrogen−Carbon-Linked (Azolylphenyl)oxazolidinones with Potent Antibacterial Activity Against the Fastidious Gram-Negative Organisms Haemophilus influenzae and Moraxella catarrhalis
Genin, Michael J, Hutchinson, Douglas K, Allwine, Debra A, Hester, Jackson B, Emmert, D. Edward, Garmon, Stuart A, Ford, Charles W, Zurenko, Gary E, Hamel, Judith C, Schaadt, Ronda D, Stapert, Douglas, Yagi, Betty H, Friis, Janice M, Shobe, Eric M, Adams, Wade J
Published in Journal of medicinal chemistry (17.12.1998)
Published in Journal of medicinal chemistry (17.12.1998)
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Substituent Effects on the Antibacterial Activity of Nitrogen−Carbon-Linked (Azolylphenyl)oxazolidinones with Expanded Activity Against the Fastidious Gram-Negative Organisms Haemophilus i nfluenzae and Moraxella c atarrhalis
Genin, Michael J, Allwine, Debra A, Anderson, David J, Barbachyn, Michael R, Emmert, D. Edward, Garmon, Stuart A, Graber, David R, Grega, Kevin C, Hester, Jackson B, Hutchinson, Douglas K, Morris, Joel, Reischer, Robert J, Ford, Charles W, Zurenko, Gary E, Hamel, Judith C, Schaadt, Ronda D, Stapert, Douglas, Yagi, Betty H
Published in Journal of medicinal chemistry (09.03.2000)
Published in Journal of medicinal chemistry (09.03.2000)
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Synthesis and antibacterial activity of new tropone-substituted phenyloxazolidinone antibacterial agents 2. Modification of the phenyl ring — the potentiating effect of fluorine substitution on in vivo activity
Barbachyn, Michael R., Toops, Dana S., Grega, Kevin C., Hendges, Susan K., Ford, Charles W., Zurenko, Gary E., Hamel, Judith C., Schaadt, Jonda D., Stapert, Douglas, Yagi, Betty H., Buysse, Jerry M., Demyan, William F., Kilburn, James O., Glickman, Suzanne E.
Published in Bioorganic & medicinal chemistry letters (07.05.1996)
Published in Bioorganic & medicinal chemistry letters (07.05.1996)
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Substituent Effects on the Antibacterial Activity of Nitrogen−Carbon-Linked (Azolylphenyl)oxazolidinones with Expanded Activity Against the Fastidious Gram-Negative Organisms Haemophilus influenzae and Moraxella catarrhalis
GENIN, Michael J., ALLWINE, Debra A., ANDERSON, David J., BARBACHYN, Michael R., EMMERT, D. Edward, GARMON, Stuart A., GRABER, David R., GREGA, Kevin C., HESTER, Jackson B., HUTCHINSON, Douglas K., MORRIS, Joel, REISCHER, Robert J., FORD, Charles W., ZURENKO, Gary E., HAMEL, Judith C., SCHAADT, Ronda D., STAPERT, Douglas, YAGI, Betty H.
Published in Journal of medicinal chemistry (09.03.2000)
Published in Journal of medicinal chemistry (09.03.2000)
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In vivo activities of U-100592 and U-100766, novel oxazolidinone antimicrobial agents, against experimental bacterial infections
FORD, C. W, HAMEL, J. C, WILSON, D. M, MOERMAN, J. K, STAPERT, D, YANCEY, R. J, HUTCHINSON, D. K, BARBACHYN, M. R, BRICKNER, S. J
Published in Antimicrobial Agents and Chemotherapy (01.06.1996)
Published in Antimicrobial Agents and Chemotherapy (01.06.1996)
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Oxazolidinones: New antibacterial agents
Ford, Charles W., Hamel, Judith C., Stapert, Douglas, Moerman, Judy K., Hutchinson, Douglas K., Barbachyn, Michael R., Zurenko, Gary E.
Published in Trends in microbiology (Regular ed.) (01.05.1997)
Published in Trends in microbiology (Regular ed.) (01.05.1997)
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Synthesis and biological evaluation of benzazepine oxazolidinone antibacterials: Antibacterial agents: solutions for the evolving problems of resistance
JOHNSON, Paul D, ARISTOFF, Paul A, ZURENKO, Gary E, SCHAADT, Ronda D, YAGI, Betty H, FORD, Charles W, HAMEL, Judith C, STAPERT, Douglas, MOERMAN, Judy K
Published in Bioorganic & medicinal chemistry letters (2003)
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Published in Bioorganic & medicinal chemistry letters (2003)
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The synthesis and antibacterial activity of 1,3,4-thiadiazole phenyl oxazolidinone analogues: Antibacterial agents: solutions for the evolving problems of resistance
THOMASCO, Lisa M, GADWOOD, Robert C, YAGI, Betty H, WEAVER, Elizabeth A, OCHOADA, Jason M, FORD, Charles W, ZURENKO, Gary E, HAMEL, Judith C, STAPERT, Douglas, MOERMAN, Judy K, SCHAADT, Ronda D
Published in Bioorganic & medicinal chemistry letters (2003)
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Published in Bioorganic & medicinal chemistry letters (2003)
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Synthesis and antibacterial activity of new tropone-substituted phenyloxazolidinone antibacterial agents 1. Identification of leads and importance of the tropone substitution pattern
Barbachyn, Michael R., Toops, Dana S., Ulanowicz, Debra A., Grega, Kevin C., Brickner, Steven J., Ford, Charles W., Zurenko, Gary E., Hamel, Judith C., Schaadt, Ronda D., Stapert, Douglas, Yagi, Betty H., Buysse, Jerry M., Demyan, William F., Kilburn, James O., Glickman, Suzanne E.
Published in Bioorganic & medicinal chemistry letters (07.05.1996)
Published in Bioorganic & medicinal chemistry letters (07.05.1996)
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Journal Article
Synthesis and Biological Evaluation of Benzazepine Oxazolidinone Antibacterials
Johnson, Paul D., Aristoff, Paul A., Zurenko, Gary E., Schaadt, Ronda D., Yagi, Betty H., Ford, Charles W., Hamel, Judith C., Stapert, Douglas, Moerman, Judy K.
Published in ChemInform (30.03.2004)
Published in ChemInform (30.03.2004)
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