Molecular basis for inhibiting human glucose transporters by exofacial inhibitors
Wang, Nan, Zhang, Shuo, Yuan, Yafei, Xu, Hanwen, Defossa, Elisabeth, Matter, Hans, Besenius, Melissa, Derdau, Volker, Dreyer, Matthias, Halland, Nis, He, Kaihui Hu, Petry, Stefan, Podeschwa, Michael, Tennagels, Norbert, Jiang, Xin, Yan, Nieng
Published in Nature communications (12.05.2022)
Published in Nature communications (12.05.2022)
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Journal Article
Computational Investigation of Drug Phototoxicity: Photosafety Assessment, Photo-Toxophore Identification, and Machine Learning
Schmidt, Friedemann, Wenzel, Jan, Halland, Nis, Güssregen, Stefan, Delafoy, Laure, Czich, Andreas
Published in Chemical research in toxicology (18.11.2019)
Published in Chemical research in toxicology (18.11.2019)
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Journal Article
SGK1 Inhibition Induces Fetal Hemoglobin in Erythroid Cells
Hara, Yannis, Stottlemyer, Mark, Alving, Kim, Halland, Nis, Hicks, Alexandra, Light, David R.
Published in Blood (23.11.2021)
Published in Blood (23.11.2021)
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Journal Article
A General and Mild Palladium‐Catalyzed Domino Reaction for the Synthesis of 2H‐Indazoles
Halland, Nis, Nazaré, Marc, R'kyek, Omar, Alonso, Jorge, Urmann, Matthias, Lindenschmidt, Andreas
Published in Angewandte Chemie (01.09.2009)
Published in Angewandte Chemie (01.09.2009)
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Journal Article
A Palladium-Catalyzed Domino Reaction To Access 3-Amino-2 H -indazoles from Hydrazines and 2-Halobenzonitriles
Alsalim, Rana, Lindemann, Peter, López-Alberca, María Pascual, Miksche, Sandra, Czechtizky, Werngard, Halland, Nis, Nazaré, Marc
Published in Organic letters (18.09.2020)
Published in Organic letters (18.09.2020)
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Journal Article
Rational Design of Highly Potent, Selective, and Bioavailable SGK1 Protein Kinase Inhibitors for the Treatment of Osteoarthritis
Halland, Nis, Schmidt, Friedemann, Weiss, Tilo, Li, Ziyu, Czech, Jorg, Saas, Joachim, Ding-Pfennigdorff, Danping, Dreyer, Matthias K., Strubing, Carsten, Nazare, Marc
Published in Journal of medicinal chemistry (27.01.2022)
Published in Journal of medicinal chemistry (27.01.2022)
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Journal Article
A Palladium-Catalyzed Domino Reaction To Access 3‑Amino‑2H‑indazoles from Hydrazines and 2‑Halobenzonitriles
Alsalim, Rana, Lindemann, Peter, López-Alberca, María Pascual, Miksche, Sandra, Czechtizky, Werngard, Halland, Nis, Nazaré, Marc
Published in Organic letters (18.09.2020)
Published in Organic letters (18.09.2020)
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Journal Article
Organocatalytic Asymmetric Michael Reaction of Cyclic 1,3-Dicarbonyl Compounds and α,β-Unsaturated Ketones-A Highly Atom-Economic Catalytic One-Step Formation of Optically Active Warfarin Anticoagulant
Halland, Nis, Hansen, Tore, Jørgensen, Karl Anker
Published in Angewandte Chemie (International ed.) (20.10.2003)
Published in Angewandte Chemie (International ed.) (20.10.2003)
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Journal Article
A general and mild domino approach to substituted 1-aminoindoles
Halland, Nis, Nazare, Marc, Alonso, Jorge, R'kyek, Omar, Lindenschmidt, Andreas
Published in Chemical communications (Cambridge, England) (01.01.2011)
Published in Chemical communications (Cambridge, England) (01.01.2011)
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Journal Article
Direct Organocatalytic Asymmetric α-Chlorination of Aldehydes
Halland, Nis, Braunton, Alan, Bachmann, Stephan, Marigo, Mauro, Jørgensen, Karl Anker
Published in Journal of the American Chemical Society (21.04.2004)
Published in Journal of the American Chemical Society (21.04.2004)
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Journal Article
Novel Small Molecule Inhibitors of Activated Thrombin Activatable Fibrinolysis Inhibitor (TAFIa) from Natural Product Anabaenopeptin
Halland, Nis, Brönstrup, Mark, Czech, Jörg, Czechtizky, Werngard, Evers, Andreas, Follmann, Markus, Kohlmann, Markus, Schiell, Matthias, Kurz, Michael, Schreuder, Herman A, Kallus, Christopher
Published in Journal of medicinal chemistry (11.06.2015)
Published in Journal of medicinal chemistry (11.06.2015)
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Journal Article
Sulfamide as Zinc Binding Motif in Small Molecule Inhibitors of Activated Thrombin Activatable Fibrinolysis Inhibitor (TAFIa)
Halland, Nis, Czech, Jörg, Czechtizky, Werngard, Evers, Andreas, Follmann, Markus, Kohlmann, Markus, Schreuder, Herman A, Kallus, Christopher
Published in Journal of medicinal chemistry (27.10.2016)
Published in Journal of medicinal chemistry (27.10.2016)
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Journal Article