Identification of 4-Substituted 1,2,3-Triazoles as Novel Oxazolidinone Antibacterial Agents with Reduced Activity against Monoamine Oxidase A
Reck, Folkert, Zhou, Fei, Girardot, Marc, Kern, Gunther, Eyermann, Charles J, Hales, Neil J, Ramsay, Rona R, Gravestock, Michael B
Published in Journal of medicinal chemistry (27.01.2005)
Published in Journal of medicinal chemistry (27.01.2005)
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Kinetic and Structural Characteristics of the Inhibition of Enoyl (Acyl Carrier Protein) Reductase by Triclosan
Ward, Walter H. J, Holdgate, Geoffrey A, Rowsell, Siân, McLean, Estelle G, Pauptit, Richard A, Clayton, Edward, Nichols, Wright W, Colls, Jeremy G, Minshull, Claire A, Jude, David A, Mistry, Anil, Timms, David, Camble, Roger, Hales, Neil J, Britton, Carolyn J, Taylor, Ian W. F
Published in Biochemistry (Easton) (21.09.1999)
Published in Biochemistry (Easton) (21.09.1999)
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Polymer-supported cobalt carbonyl complexes as novel solid-phase catalysts of the Pauson-Khand reaction
Comely, AC, Gibson, SE, Hales, NJ
Published in Chemical communications (Cambridge, England) (01.01.2000)
Published in Chemical communications (Cambridge, England) (01.01.2000)
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The Azomethine Ylid Strategy in β-Lactam Synthesis. Application to Selenapenams
Brown, Giles A., Anderson, Kirsty M., Murray, Martin, Gallagher, Timothy, Hales, Neil J.
Published in Tetrahedron (28.07.2000)
Published in Tetrahedron (28.07.2000)
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Chromium carbonyl complexes as novel traceless linkers
Gibson (née Thomas), Susan E., Hales, Neil J., Peplow, Mark A.
Published in Tetrahedron letters (12.02.1999)
Published in Tetrahedron letters (12.02.1999)
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Polymer supported cobalt carbonyl complexes as novel traceless alkyne linkers for solid-phase synthesis
Comely, AC, Gibson, SE, Hales, NJ
Published in Chemical communications (Cambridge, England) (21.10.1999)
Published in Chemical communications (Cambridge, England) (21.10.1999)
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A Direct and Convergent Approach to Penams and Penems
Planchenault, Denis, Wisedale, Richard, Gallagher, Timothy, Hales, Neil J
Published in Journal of organic chemistry (30.05.1997)
Published in Journal of organic chemistry (30.05.1997)
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β-Lactam-Based Azomethine Ylide Reactivity. Expedient Synthesis of Carbapenams and Carbapenems
Martel, Sarah R, Wisedale, Richard, Gallagher, Timothy, Hall, Lee D, Mahon, Mary F, Bradbury, Robert H, Hales, Neil J
Published in Journal of the American Chemical Society (05.03.1997)
Published in Journal of the American Chemical Society (05.03.1997)
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Aldehydes and ketones as dipolarophiles: application to the synthesis of oxapenams
Andrews, MD, Brown, GA, Charmant, JPH, Peakman, TM, Rebello, A, Walsh, KE, Gallagher, T, Hales, NJ
Published in Chemical communications (Cambridge, England) (07.02.1999)
Published in Chemical communications (Cambridge, England) (07.02.1999)
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The azomethine ylide strategy for beta-lactam synthesis. Azapenams and 1-azacephams
Brown, D, Brown, GA, Andrews, M, Large, JM, Urban, D, Butts, CP, Hales, NJ, Gallagher, T
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2002)
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2002)
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Trapping highly reactive dipolarophiles. Exploiting the mechanism associated with the azomethine ylide strategy for beta-lactam synthesis
Brown, GA, Anderson, KM, Large, JM, Planchenault, D, Urban, D, Hales, NJ, Gallagher, T
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (2001)
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (2001)
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The azomethine ylide strategy for beta-lactam synthesis. An evaluation of alternative pathways for azomethine ylide generation
Brown, GA, Martel, Wisedale, R, Charmant, JPH, Hales, NJ, Fishwick, CWG, Gallagher, T
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2001)
Published in Perkin 1 : an international journal of organic and bio-organic chemistry (01.01.2001)
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