Pd-Catalyzed Cross-Coupling Reactions Promoted by Biaryl Phosphorinane Ligands
Laffoon, Summer D, Chan, Vincent S, Fickes, Michael G, Kotecki, Brian, Ickes, Andrew R, Henle, Jeremy, Napolitano, José G, Franczyk, Thaddeus S, Dunn, Travis B, Barnes, David M, Haight, Anthony R, Henry, Rodger F, Shekhar, Shashank
Published in ACS catalysis (06.12.2019)
Published in ACS catalysis (06.12.2019)
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Discovery and Development of Metal-Catalyzed Coupling Reactions in the Synthesis of Dasabuvir, an HCV-Polymerase Inhibitor
Barnes, David M, Shekhar, Shashank, Dunn, Travis B, Barkalow, Jufang H, Chan, Vincent S, Franczyk, Thaddeus S, Haight, Anthony R, Hengeveld, John E, Kolaczkowski, Lawrence, Kotecki, Brian J, Liang, Guangxin, Marek, James C, McLaughlin, Maureen A, Montavon, Donna K, Napier, James J
Published in Journal of organic chemistry (19.04.2019)
Published in Journal of organic chemistry (19.04.2019)
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A General Method for the Synthesis of Unsymmetrically Substituted Ureas via Palladium-Catalyzed Amidation
Kotecki, Brian J, Fernando, Dilinie P, Haight, Anthony R, Lukin, Kirill A
Published in Organic letters (19.02.2009)
Published in Organic letters (19.02.2009)
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Journal Article
BCL-X L -targeting antibody-drug conjugates are active in preclinical models and mitigate on-mechanism toxicity of small-molecule inhibitors
Judd, Andrew S, Bawa, Bhupinder, Buck, Wayne R, Tao, Zhi-Fu, Li, Yingchun, Mitten, Michael J, Bruncko, Milan, Catron, Nathaniel, Doherty, George, Durbin, Kenneth R, Enright, Brian, Frey, Robin, Haasch, Deanna, Haman, Sandra, Haight, Anthony R, Henriques, Tracy A, Holms, James, Izeradjene, Kamel, Judge, Russell A, Jenkins, Gary J, Kunzer, Aaron, Leverson, Joel D, Martin, Ruth L, Mitra, Diya, Mittelstadt, Scott, Nelson, Lorne, Nimmer, Paul, Palma, Joann, Peterson, Richard, Phillips, Darren C, Ralston, Sherry L, Rosenberg, Saul H, Shen, Xiaoqiang, Song, Xiaohong, Vaidya, Kedar R, Wang, Xilu, Wang, Jin, Xiao, Yu, Zhang, Haichao, Zhang, Xinxin, Blomme, Eric A, Boghaert, Erwin R, Kalvass, John C, Phillips, Andrew, Souers, Andrew J
Published in Science advances (04.10.2024)
Published in Science advances (04.10.2024)
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Journal Article
BCL-XL-targeting antibody-drug conjugates are active in preclinical models and mitigate on-mechanism toxicity of small-molecule inhibitors
Judd, Andrew S, Bawa, Bhupinder, Buck, Wayne R, Tao, Zhi-Fu, Li, Yingchun, Mitten, Michael J, Bruncko, Milan, Catron, Nathaniel, Doherty, George, Durbin, Kenneth R, Enright, Brian, Frey, Robin, Haasch, Deanna, Haman, Sandra, Haight, Anthony R, Henriques, Tracy A, Holms, James, Izeradjene, Kamel, Judge, Russell A, Jenkins, Gary J, Kunzer, Aaron, Leverson, Joel D, Martin, Ruth L, Mitra, Diya, Mittelstadt, Scott, Nelson, Lorne, Nimmer, Paul, Palma, Joann, Peterson, Richard, Phillips, Darren C, Ralston, Sherry L, Rosenberg, Saul H, Shen, Xiaoqiang, Song, Xiaohong, Vaidya, Kedar R, Wang, Xilu, Wang, Jin, Xiao, Yu, Zhang, Haichao, Zhang, Xinxin, Blomme, Eric A, Boghaert, Erwin R, Kalvass, John C, Phillips, Andrew, Souers, Andrew J
Published in Science advances (04.10.2024)
Published in Science advances (04.10.2024)
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Journal Article
General Method for the Palladium-Catalyzed Allylation of Aliphatic Alcohols
Haight, Anthony R, Stoner, Eric J, Peterson, Matthew J, Grover, Vandana K
Published in Journal of organic chemistry (17.10.2003)
Published in Journal of organic chemistry (17.10.2003)
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Journal Article
The Discovery and Development of a Safe, Practical Synthesis of ABT-869
Kruger, Albert W, Rozema, Michael J, Chu-Kung, Alexander, Gandarilla, Jorge, Haight, Anthony R, Kotecki, Brian J, Richter, Steven M, Schwartz, Albert M, Wang, Zhe
Published in Organic process research & development (20.11.2009)
Published in Organic process research & development (20.11.2009)
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Journal Article
Process Development for ABT-472, a Benzimidazole PARP Inhibitor
Barkalow, Jufang H, Breting, Jeffrey, Gaede, Bruce J, Haight, Anthony R, Henry, Rodger, Kotecki, Brian, Mei, Jianzhang, Pearl, Kurt B, Tedrow, Jason S, Viswanath, Shekhar K
Published in Organic process research & development (01.07.2007)
Published in Organic process research & development (01.07.2007)
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Journal Article
Selective Reduction of Cysteine Mutant Antibodies for Site-Specific Antibody–Drug Conjugates
Liao, Xiaoli, Haight, Anthony, Welch, Dennie, Han, Linjie
Published in Bioconjugate chemistry (20.12.2023)
Published in Bioconjugate chemistry (20.12.2023)
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Journal Article
Impact of Entropic Effects in the Classical Resolution of a 2-Arylpyrrolidine
Barnes, David M, Barkalow, Jufang, Chen, Yong, Gupta, Ashok, Haight, Anthony R, Hengeveld, John E, Kerdesky, Francis A. J, Kotecki, Brian J, Macri, Bryan, Pal, Agnes
Published in Organic process research & development (20.03.2009)
Published in Organic process research & development (20.03.2009)
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A Scaleable Synthesis of Fiduxosin
Haight, Anthony R, Bailey, Anne E, Baker, William S, Cain, Michael H, Copp, Richard R, DeMattei, John A, Ford, Kelley L, Henry, Rodger F, Hsu, Margaret C, Keyes, Robert F, King, Steven A, McLaughlin, Maureen A, Melcher, Laura M, Nadler, William R, Oliver, Patricia A, Parekh, Shyamal I, Patel, Hemant H, Seif, Louis S, Staeger, Mike A, Wayne, Gregory S, Wittenberger, Steven J, Zhang, Weijiang
Published in Organic process research & development (01.11.2004)
Published in Organic process research & development (01.11.2004)
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Journal Article
Chlorination at the 8-Position of a Functionalized Quinolone and the Synthesis of Quinolone Antibiotic ABT-492
Barnes, David M, Christesen, Alan C, Engstrom, Kenneth M, Haight, Anthony R, Hsu, Margaret C, Lee, Elaine C, Peterson, Matthew J, Plata, Daniel J, Raje, Prasad S, Stoner, Eric J, Tedrow, Jason S, Wagaw, Seble
Published in Organic process research & development (21.07.2006)
Published in Organic process research & development (21.07.2006)
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Journal Article
Synthesis of the Quinolone ABT-492: Crystallizations for Optimal Processing
Haight, Anthony R, Ariman, Sema Z, Barnes, David M, Benz, Nancy J, Gueffier, Francoix X, Henry, Rodger F, Hsu, Margaret C, Lee, Elaine C, Morin, Larry, Pearl, Kurt B, Peterson, Matthew J, Plata, Daniel J, Willcox, David R
Published in Organic process research & development (21.07.2006)
Published in Organic process research & development (21.07.2006)
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Journal Article
Synthesis of Erythromycin Derivatives via the Olefin Cross-Metathesis Reaction
Hsu, Margaret C, Junia, Adam J, Haight, Anthony R, Zhang, Weijiang
Published in Journal of organic chemistry (28.05.2004)
Published in Journal of organic chemistry (28.05.2004)
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Journal Article
Internal coordination at tin promotes selective alkyl transfer in the Stille coupling reaction
Vedejs, Edwin, Haight, Anthony R, Moss, William O
Published in Journal of the American Chemical Society (01.07.1992)
Published in Journal of the American Chemical Society (01.07.1992)
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Journal Article
Preclinical Characterization of Catabolic Pathways and Metabolism of ABBV-011, a Novel Calicheamicin-Based SEZ6-Targeting Antibody-Drug Conjugate
Ladror, Daniel, Gu, Christine, Tong, Vince, Schammel, Alexander, Gavrilyuk, Julia, Haight, Anthony, Sarvaiya, Hetal
Published in Drug metabolism and disposition (01.02.2024)
Published in Drug metabolism and disposition (01.02.2024)
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Journal Article
Allylation of Erythromycin Derivatives: Introduction of Allyl Substituents into Highly Hindered Alcohols
Stoner, Eric J, Peterson, Matthew J, Allen, Michael S, DeMattei, John A, Haight, Anthony R, Leanna, M. Robert, Patel, Subhash R, Plata, Daniel J, Premchandran, Ramiya H, Rasmussen, Michael
Published in Journal of organic chemistry (14.11.2003)
Published in Journal of organic chemistry (14.11.2003)
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Synthesis of (R)‑Boc-2-methylproline via a Memory of Chirality Cyclization. Application to the Synthesis of Veliparib, a Poly(ADP-ribose) Polymerase Inhibitor
Kolaczkowski, Lawrence, Barkalow, Jufang, Barnes, David M, Haight, Anthony, Pritts, Wayne, Schellinger, Adam
Published in Journal of organic chemistry (19.04.2019)
Published in Journal of organic chemistry (19.04.2019)
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Journal Article
Reduction of an Enaminone: Synthesis of the Diamino Alcohol Core of Ritonavir
Haight, Anthony R, Stuk, Timothy L, Allen, Michael S, Bhagavatula, Lakshmi, Fitzgerald, Michael, Hannick, Steven M, Kerdesky, Francis A. J, Menzia, Jerome A, Parekh, Shyamal I, Robbins, Timothy A, Scarpetti, David, Tien, Jien-Heh J
Published in Organic process research & development (01.03.1999)
Published in Organic process research & development (01.03.1999)
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