Efficacious intermittent dosing of a novel JAK2 inhibitor in mouse models of polycythemia vera
Kraus, Manfred, Wang, Yuxun, Aleksandrowicz, Dan, Bachman, Eric, Szewczak, Alexander A, Walker, Deborah, Xu, Lin, Bouthillette, Melaney, Childers, Kaleen M, Dolinski, Brian, Haidle, Andrew M, Kopinja, Johnny, Lee, Linda, Lim, Jongwon, Little, Kevin D, Ma, Yanhong, Mathur, Anjili, Mo, Jan-Rung, O'Hare, Erin, Otte, Ryan D, Taoka, Brandon M, Wang, Wenxian, Yin, Hong, Zabierek, Anna A, Zhang, Weisheng, Zhao, Shuxia, Zhu, Joe, Young, Jonathan R, Marshall, C Gary
Published in PloS one (18.05.2012)
Published in PloS one (18.05.2012)
Get full text
Journal Article
Building a Culture of Medicinal Chemistry Knowledge Sharing
Beshore, Douglas C, Haidle, Andrew M, Arasappan, Ashok, Lim, Yeon-Hee, Raheem, Izzat, Roecker, Anthony J, Shockley, Samantha E, Simov, Vladimir
Published in Journal of medicinal chemistry (10.03.2022)
Published in Journal of medicinal chemistry (10.03.2022)
Get full text
Journal Article
Discovery of MK-1454: A Potent Cyclic Dinucleotide Stimulator of Interferon Genes Agonist for the Treatment of Cancer
Chang, Wonsuk, Altman, Michael D, Lesburg, Charles A, Perera, Samanthi A, Piesvaux, Jennifer A, Schroeder, Gottfried K, Wyss, Daniel F, Cemerski, Saso, Chen, Yiping, DiNunzio, Edward, Haidle, Andrew M, Ho, Thu, Kariv, Ilona, Knemeyer, Ian, Kopinja, Johnny E, Lacey, Brian M, Laskey, Jason, Lim, Jongwon, Long, Brian J, Ma, Yanhong, Maddess, Matthew L, Pan, Bo-Sheng, Presland, Jeremy P, Spooner, Edward, Steinhuebel, Dietrich, Truong, Quang, Zhang, Zhibo, Fu, Jianmin, Addona, George H, Northrup, Alan B, Parmee, Emma, Tata, James R, Bennett, David Jonathan, Cumming, Jared N, Siu, Tony, Trotter, B. Wesley
Published in Journal of medicinal chemistry (14.04.2022)
Published in Journal of medicinal chemistry (14.04.2022)
Get full text
Journal Article
Augmenting Hit Identification by Virtual Screening Techniques in Small Molecule Drug Discovery
Yan, Xin Cindy, Sanders, John M, Gao, Ying-Duo, Tudor, Matthew, Haidle, Andrew M, Klein, Daniel J, Converso, Antonella, Lesburg, Charles A, Zang, Yi, Wood, Harold B
Published in Journal of chemical information and modeling (28.09.2020)
Published in Journal of chemical information and modeling (28.09.2020)
Get full text
Journal Article
Informing the Selection of Screening Hit Series with in Silico Absorption, Distribution, Metabolism, Excretion, and Toxicity Profiles
Sanders, John M, Beshore, Douglas C, Culberson, J Christopher, Fells, James I, Imbriglio, Jason E, Gunaydin, Hakan, Haidle, Andrew M, Labroli, Marc, Mattioni, Brian E, Sciammetta, Nunzio, Shipe, William D, Sheridan, Robert P, Suen, Linda M, Verras, Andreas, Walji, Abbas, Joshi, Elizabeth M, Bueters, Tjerk
Published in Journal of medicinal chemistry (24.08.2017)
Published in Journal of medicinal chemistry (24.08.2017)
Get full text
Journal Article
Informing the Selection of Screening Hit Series with in Silico Absorption, Distribution, Metabolism, Excretion, and Toxicity Profiles: Miniperspective
Sanders, John M, Beshore, Douglas C, Culberson, J. Christopher, Fells, James I, Imbriglio, Jason E, Gunaydin, Hakan, Haidle, Andrew M, Labroli, Marc, Mattioni, Brian E, Sciammetta, Nunzio, Shipe, William D, Sheridan, Robert P, Suen, Linda M, Verras, Andreas, Walji, Abbas, Joshi, Elizabeth M, Bueters, Tjerk
Published in Journal of medicinal chemistry (24.08.2017)
Published in Journal of medicinal chemistry (24.08.2017)
Get full text
Journal Article
Overcoming Mutagenicity and Ion Channel Activity: Optimization of Selective Spleen Tyrosine Kinase Inhibitors
Ellis, J. Michael, Altman, Michael D, Bass, Alan, Butcher, John W, Byford, Alan J, Donofrio, Anthony, Galloway, Sheila, Haidle, Andrew M, Jewell, James, Kelly, Nancy, Leccese, Erica K, Lee, Sandra, Maddess, Matthew, Miller, J. Richard, Moy, Lily Y, Osimboni, Ekundayo, Otte, Ryan D, Reddy, M. Vijay, Spencer, Kerrie, Sun, Binyuan, Vincent, Stella H, Ward, Gwendolyn J, Woo, Grace H. C, Yang, Chiming, Houshyar, Hani, Northrup, Alan B
Published in Journal of medicinal chemistry (26.02.2015)
Published in Journal of medicinal chemistry (26.02.2015)
Get full text
Journal Article
MARK inhibitors: Declaring a No-Go decision on a chemical series based on extensive DMPK experimentation
Haidle, Andrew M., Childers, Kaleen K., Zabierek, Anna A., Katz, Jason D., Jewell, James P., Hou, Yongquan, Altman, Michael D., Szewczak, Alexander, Chen, Dapeng, Harsch, Andreas, Hayashi, Mansuo, Warren, Lee, Hutton, Michael, Nuthall, Hugh, Stanton, Matt G., Davies, Ian W., Munoz, Ben, Northrup, Alan
Published in Bioorganic & medicinal chemistry letters (01.01.2017)
Published in Bioorganic & medicinal chemistry letters (01.01.2017)
Get full text
Journal Article
Carboxamide Spleen Tyrosine Kinase (Syk) Inhibitors: Leveraging Ground State Interactions To Accelerate Optimization
Ellis, J. Michael, Altman, Michael D, Cash, Brandon, Haidle, Andrew M, Kubiak, Rachel L, Maddess, Matthew L, Yan, Youwei, Northrup, Alan B
Published in ACS medicinal chemistry letters (08.12.2016)
Published in ACS medicinal chemistry letters (08.12.2016)
Get full text
Journal Article
Thiophene carboxamide inhibitors of JAK2 as potential treatments for myleoproliferative neoplasms
Haidle, Andrew M., Zabierek, Anna A., Childers, Kaleen K., Rosenstein, Craig, Mathur, Anjili, Altman, Michael D., Chan, Grace, Xu, Lin, Bachman, Eric, Mo, Jan-Rung, Bouthillette, Melaney, Rush, Thomas, Tempest, Paul, Marshall, C. Gary, Young, Jonathan R.
Published in Bioorganic & medicinal chemistry letters (15.04.2014)
Published in Bioorganic & medicinal chemistry letters (15.04.2014)
Get full text
Journal Article
IL4I1 억제제 및 사용 방법
CASH BRANDON D, LARSEN MATTHEW A, LIU PING, MCGOWAN MEREDETH A, SILIPHAIVANH PHIENG, LESBURG CHARLES A, HOPKINS BRETT A, YAN XIN, HAIDLE ANDREW M, FU WENLANG, SANYAL SULAGNA, WHITE CATHERINE M, PU QINGLIN, GIAMBASU GEORGE MADALIN
Year of Publication 11.01.2023
Get full text
Year of Publication 11.01.2023
Patent
STING 효능제로서의 벤조[b]티오펜 화합물
CASH BRANDON D, CUMMING JARED N, JEWELL JAMES P, LARSEN MATTHEW A, ALTMAN MICHAEL D, LIM JONGWON, HENDERSON TIMOTHY J, LU MIN, CHANG WONSUK, TYAGARAJAN SRIRAM, HAIDLE ANDREW M, LIANG RUI, OTTE RYAN D, SIU TONY, TROTTER BENJAMIN WESLEY
Year of Publication 24.05.2019
Get full text
Year of Publication 24.05.2019
Patent
AMINOPYRIMIDINES AS SYK INHIBITORS
DI FRANCESCO MARIA EMILIA, ZHOU HUA, GRIMM JONATHAN, CHILDERS KALEEN KONRAD, SCHELL ADAM J, ALTMAN MICHAEL D, HAIDLE ANDREW M, ELLIS JOHN MICHAEL, OTTE RYAN D, PETROCCHI ALESSIA, FISCHER CHRISTIAN, NORTHRUP ALAN B, KATTAR SOLOMON D
Year of Publication 07.03.2014
Get full text
Year of Publication 07.03.2014
Patent
A practical, two-step synthesis of 1-alkyl-4-aminopyrazoles
Zabierek, Anna A., Konrad, Kaleen M., Haidle, Andrew M.
Published in Tetrahedron letters (28.04.2008)
Published in Tetrahedron letters (28.04.2008)
Get full text
Journal Article
AMINOPYRIMIDINES AS SYK INHIBITORS
DONOFRIO ANTHONY, GUAY DANIEL, DI FRANCESCO MARIA EMILIA, ZHOU HUA, CHILDERS KALEEN KONRAD, KNOWLES SANDRA LEE, SCHELL ADAM J, SPENCER KERRIE B, ALTMAN MICHAEL D, TAOKA BRANDON M, ANDRESEN BRIAN M, O'BOYLE BRENDAN M, GAUTHIER JACQUES YVES, REUTERSHAN MICHAEL H, HAIDLE ANDREW M, TROTTER B. WESLEY, OTTE RYAN D, GUERIN DAVID JOSEPH, BHAT SATHESH, PETROCCHI ALESSIA, SIU TONY, LI CHAOMIN, DUPONT GAUDET KRISTINA, MACHACEK MICHELLE R, WOO, HYUN CHONG, COTE BERNARD, GRIMM JONATHAN, ARRINGTON KENNETH L, ROBICHAUD JOEL S, KATTAR SOLOMON, MADDESS MATTHEW L, ROMEO ERIC, BURCH JASON, FOURNIER JEAN FRANCOIS, ELLIS JOHN MICHAEL, LIM, JONG WON, FISCHER CHRISTIAN, NORTHRUP ALAN B
Year of Publication 04.09.2012
Get full text
Year of Publication 04.09.2012
Patent