Design and synthesis of a folate-receptor targeted diazepine-ring-opened pyrrolobenzodiazepine prodrug conjugate
Vlahov, Iontcho R., Qi, Longwu, Santhapuram, Hari Krishna R., Felten, Albert, Parham, Garth L., Zou, Ning, Wang, Kevin, You, Fei, Vaughn, Jeremy F., Hahn, Spencer J., Klein, Hanna F., Kleindl, Paul J., Reddy, Joe, Reno, Dan, Nicoson, Jeff, Leamon, Christopher P.
Published in Bioorganic & medicinal chemistry letters (01.04.2020)
Published in Bioorganic & medicinal chemistry letters (01.04.2020)
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Latent Warheads for Targeted Cancer Therapy: Design and Synthesis of pro-Pyrrolobenzodiazepines and Conjugates
Vlahov, Iontcho R, Qi, Longwu, Kleindl, Paul J, Santhapuram, Hari K, Felten, Albert, Parham, Garth L, Wang, Kevin, You, Fei, Vaughn, Jeremy F, Hahn, Spencer J, Klein, Hanna F, Vetzel, Marilynn, Reddy, Joseph A, Nelson, Melissa, Nicoson, Jeff, Leamon, Christopher P
Published in Bioconjugate chemistry (20.12.2017)
Published in Bioconjugate chemistry (20.12.2017)
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Antiinflammatory Activity of a Novel Folic Acid Targeted Conjugate of the mTOR Inhibitor Everolimus
Lu, Yingjuan, Parker, Nikki, Kleindl, Paul J, Cross, Vicky A, Wollak, Kristin, Westrick, Elaine, Stinnette, Torian W, Gehrke, Mark A, Wang, Kevin, Santhapuram, Hari Krishna R, You, Fei, Hahn, Spencer J, Vaughn, Jeremy F, Klein, Patrick J, Vlahov, Iontcho R, Low, Philip S, Leamon, Christopher P
Published in Molecular medicine (Cambridge, Mass.) (08.07.2015)
Published in Molecular medicine (Cambridge, Mass.) (08.07.2015)
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Carbohydrate-Based Synthetic Approach to Control Toxicity Profiles of Folate−Drug Conjugates
Vlahov, Iontcho R, Santhapuram, Hari Krishna R, You, Fei, Wang, Yu, Kleindl, Paul J, Hahn, Spencer J, Vaughn, Jeremy F, Reno, Daniel S, Leamon, Christopher P
Published in Journal of organic chemistry (04.06.2010)
Published in Journal of organic chemistry (04.06.2010)
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Folate receptor-targeted aminopterin therapy is highly effective and specific in experimental models of autoimmune uveitis and autoimmune encephalomyelitis
Lu, Yingjuan, Wollak, Kristin N, Cross, Vicky A, Westrick, Elaine, Wheeler, Leroy W, Stinnette, Torian W, Vaughn, Jeremy F, Hahn, Spencer J, Xu, Le-Cun, Vlahov, Iontcho R, Leamon, Christopher P
Published in Clinical immunology (Orlando, Fla.) (01.01.2014)
Published in Clinical immunology (Orlando, Fla.) (01.01.2014)
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Design and regioselective synthesis of a new generation of targeted therapeutics. Part 3: Folate conjugates of aminopterin hydrazide for the treatment of inflammation
Vlahov, Iontcho R., You, Fei, Santhapuram, Hari Krishna R., Wang, Yu, Vaughn, Jeremy F., Hahn, Spencer J., Kleindl, Paul J., Fan, Mingjin, Leamon, Christopher P.
Published in Bioorganic & medicinal chemistry letters (15.02.2011)
Published in Bioorganic & medicinal chemistry letters (15.02.2011)
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Journal Article
Abstract 216: pro -Pyrrolobenzodiazepine ( pro -PBD) bioconjugates, the legacy: Design and synthesis of pro -PBD conjugates containing self-immolative substituted disulfide linkers
Vlahov, Iontcho, Qi, Longwu, Santhapuram, Hari K., Parham, Garth, Wang, Kevin, Vaughn, Jeremy F., Hahn, Spencer J., Vetzel, Marilynn, Nelson, Melissa, Reddy, Joseph A., Leamon, Christopher P.
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
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PBD CONJUGATES FOR TREATING DISEASES
REDDY, Joseph Anand, LU, Yingjuan J, YOU, Fei, VLAHOV, Iontcho Radoslavov, FELTEN, Albert E, PARHAM, Garth L, LEAMON, Christopher Paul, QI, Longwu, WANG, Kevin Yu, SANTHAPURAM, Hari Krishna R, WHEELER, II, Leroy W, ZOU, Ning, HAHN, Spencer J
Year of Publication 15.10.2020
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Year of Publication 15.10.2020
Patent
FOLATE CONJUGATE FOR USE IN TARGETING TUMOR ASSOCIATED MACROPHAGES
REDDY, Joseph Anand, LU, Yingjuan J, YOU, Fei, VLAHOV, Iontcho Radoslavov, FELTEN, Albert E, PARHAM, Garth L, LEAMON, Christopher Paul, QI, Longwu, WANG, Kevin Yu, SANTHAPURAM, Hari Krishna R, WHEELER, II, Leroy W, ZOU, Ning, HAHN, Spencer J
Year of Publication 06.02.2020
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Year of Publication 06.02.2020
Patent
FOLATE CONJUGATE FOR USE IN TARGETING TUMOR ASSOCIATED MACROPHAGES
REDDY, Joseph Anand, LU, Yingjuan J, YOU, Fei, VLAHOV, Iontcho Radoslavov, FELTEN, Albert E, PARHAM, Garth L, LEAMON, Christopher Paul, QI, Longwu, WANG, Kevin Yu, SANTHAPURAM, Hari Krishna R, WHEELER, II, Leroy W, ZOU, Ning, HAHN, Spencer J
Year of Publication 05.02.2020
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Year of Publication 05.02.2020
Patent
FOLATE CONJUGATE FOR USE IN TARGETING TUMOR ASSOCIATED MACROPHAGES
REDDY, Joseph Anand, LU, Yingjuan J, YOU, Fei, VLAHOV, Iontcho Radoslavov, FELTEN, Albert E, PARHAM, Garth L, WHEELER, II, LEAMON, Christopher Paul, QI, Longwu, WANG, Kevin Yu, SANTHAPURAM, Hari Krishna R, ZOU, Ning, HAHN, Spencer J
Year of Publication 04.10.2018
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Year of Publication 04.10.2018
Patent
PBD CONJUGATES FOR TREATING DISEASES
REDDY, Joseph Anand, LU, Yingjuan J, YOU, Fei, VLAHOV, Iontcho Radoslavov, FELTEN, Albert E, PARHAM, Garth L, LEAMON, Christopher Paul, QI, Longwu, WANG, Kevin Yu, SANTHAPURAM, Hari Krishna R, WHEELER, II, Leroy W, ZOU, Ning, HAHN, Spencer J
Year of Publication 05.10.2017
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Year of Publication 05.10.2017
Patent
FOLATE CONJUGATE FOR USE IN TARGETING TUMOR ASSOCIATED MACROPHAGES
REDDY JOSEPH ANAND, ZOU NING, WANG KEVIN YU, LU YINGJUAN J, VLAHOV IONTCHO RADOSLAVOV, PARHAM GARTH L, WHEELER II, HAHN SPENCER J, QI LONGWU, SANTHAPURAM HARI KRISHNA R, YOU FEI, LEAMON CHRISTOPHER PAUL, FELTEN ALBERT E
Year of Publication 10.01.2020
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Year of Publication 10.01.2020
Patent