A First-in-Human Study of Novel Cereblon Modulator Avadomide (CC-122) in Advanced Malignancies
Rasco, Drew W, Papadopoulos, Kyriakos P, Pourdehnad, Michael, Gandhi, Anita K, Hagner, Patrick R, Li, Yan, Wei, Xin, Chopra, Rajesh, Hege, Kristen, DiMartino, Jorge, Shih, Kent
Published in Clinical cancer research (01.01.2019)
Published in Clinical cancer research (01.01.2019)
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CC-122, a pleiotropic pathway modifier, mimics an interferon response and has antitumor activity in DLBCL
Hagner, Patrick R., Man, Hon-Wah, Fontanillo, Celia, Wang, Maria, Couto, Suzana, Breider, Mike, Bjorklund, Chad, Havens, Courtney G., Lu, Gang, Rychak, Emily, Raymon, Heather, Narla, Rama Krishna, Barnes, Leo, Khambatta, Gody, Chiu, Hsiling, Kosek, Jolanta, Kang, Jian, Amantangelo, Michael D., Waldman, Michelle, Lopez-Girona, Antonia, Cai, Ti, Pourdehnad, Michael, Trotter, Matthew, Daniel, Thomas O., Schafer, Peter H., Klippel, Anke, Thakurta, Anjan, Chopra, Rajesh, Gandhi, Anita K.
Published in Blood (06.08.2015)
Published in Blood (06.08.2015)
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Hypoxia-inducible Factor-1α (HIF-1α) Promotes Cap-dependent Translation of Selective mRNAs through Up-regulating Initiation Factor eIF4E1 in Breast Cancer Cells under Hypoxia Conditions
Yi, Tingfang, Papadopoulos, Evangelos, Hagner, Patrick R., Wagner, Gerhard
Published in The Journal of biological chemistry (28.06.2013)
Published in The Journal of biological chemistry (28.06.2013)
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Journal Article
Phase I, multicenter, dose‐escalation study of avadomide in adult Japanese patients with advanced malignancies
Hatake, Kiyohiko, Chou, Takaaki, Doi, Toshihiko, Terui, Yasuhito, Kato, Harumi, Hirose, Takayuki, Seo, Sachiko, Pourdehnad, Michael, Ogaki, Yumi, Fujimoto, Hiroshi, Hagner, Patrick R., Yamamoto, Kazuhito
Published in Cancer science (01.01.2021)
Published in Cancer science (01.01.2021)
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Journal Article
Interactome of Aiolos/Ikaros Reveals Combination Rationale of Cereblon Modulators with HDAC Inhibitors in DLBCL
Hagner, Patrick R, Chiu, Hsiling, Chopra, Vivek S, Colombo, Martino, Patel, Nisha, Estevez, Maria Ortiz, Waldman, Michelle F, Loos, Remco, Towfic, Fadi, Gandhi, Anita K
Published in Clinical cancer research (02.08.2022)
Published in Clinical cancer research (02.08.2022)
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Journal Article
Extended exposure to low doses of azacitidine induces differentiation of leukemic stem cells through activation of myeloperoxidase
Jeyaraju, Danny V, Alapa, Maryam, Polonskaia, Ann, Risueño, Alberto, Subramanyam, Prakash, Anand, Amit, Ghosh, Kaushik, Kyriakopoulos, Charalampos, Hemerich, Daiane, Hurren, Rose, Wang, Xiaoming, Gronda, Marcela, Ahsan, Aarif, Chiu, Hsiling, Thomas, Geethu, Lind, Evan F, Menezes, Daniel L, Schimmer, Aaron D, Hagner, Patrick R, Gandhi, Anita, Thakurta, Anjan G
Published in Haematologica (Roma) (01.04.2024)
Published in Haematologica (Roma) (01.04.2024)
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Avadomide monotherapy in relapsed/refractory DLBCL: safety, efficacy, and a predictive gene classifier
Carpio, Cecilia, Bouabdallah, Reda, Ysebaert, Loïc, Sancho, Juan-Manuel, Salles, Gilles, Cordoba, Raul, Pinto, Antonio, Gharibo, Mecide, Rasco, Drew, Panizo, Carlos, Lopez-Martin, Jose A., Santoro, Armando, Salar, Antonio, Damian, Silvia, Martin, Alejandro, Verhoef, Gregor, Van den Neste, Eric, Wang, Maria, Couto, Suzana, Carrancio, Soraya, Weng, Andrew, Wang, Xuehai, Schmitz, Frank, Wei, Xin, Hege, Kristen, Trotter, Matthew W.B., Risueño, Alberto, Buchholz, Tonia J., Hagner, Patrick R., Gandhi, Anita K., Pourdehnad, Michael, Ribrag, Vincent
Published in Blood (26.03.2020)
Published in Blood (26.03.2020)
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Journal Article
Triggering interferon signaling in T cells with avadomide sensitizes CLL to anti-PD-L1/PD-1 immunotherapy
Ioannou, Nikolaos, Hagner, Patrick R., Stokes, Matt, Gandhi, Anita K., Apollonio, Benedetta, Fanous, Mariam, Papazoglou, Despoina, Sutton, Lesley-Ann, Rosenquist, Richard, Amini, Rose-Marie, Chiu, Hsiling, Lopez-Girona, Antonia, Janardhanan, Preethi, Awan, Farrukh T., Jones, Jeffrey, Kay, Neil E., Shanafelt, Tait D., Tallman, Martin S., Stamatopoulos, Kostas, Patten, Piers E.M., Vardi, Anna, Ramsay, Alan G.
Published in Blood (14.01.2021)
Published in Blood (14.01.2021)
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Journal Article
Activity of lenalidomide in mantle cell lymphoma can be explained by NK cell‐mediated cytotoxicity
Hagner, Patrick R., Chiu, Hsiling, Ortiz, Maria, Apollonio, Benedetta, Wang, Maria, Couto, Suzana, Waldman, Michelle F., Flynt, Erin, Ramsay, Alan G., Trotter, Matthew, Gandhi, Anita K., Chopra, Rajesh, Thakurta, Anjan
Published in British journal of haematology (01.11.2017)
Published in British journal of haematology (01.11.2017)
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Journal Article
Combination lenalidomide‐rituximab immunotherapy activates anti‐tumour immunity and induces tumour cell death by complementary mechanisms of action in follicular lymphoma
Chiu, Hsiling, Trisal, Preeti, Bjorklund, Chad, Carrancio, Soraya, Toraño, Estela G., Guarinos, Carla, Papazoglou, Despoina, Hagner, Patrick R., Beldi‐Ferchiou, Asma, Tarte, Karin, Delfau‐Larue, Marie‐Hélène, Morschhauser, Franck, Ramsay, Alan G., Gandhi, Anita K.
Published in British journal of haematology (01.04.2019)
Published in British journal of haematology (01.04.2019)
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Overcoming IMiD resistance in T-cell lymphomas through potent degradation of ZFP91 and IKZF1
Wu, Wenchao, Nelson, Geoffrey M., Koch, Raphael, Donovan, Katherine A., Nowak, Radosław P., Heavican-Foral, Tayla B., Nirmal, Ajit J., Liu, Huiyun, Yang, Lei, Duffy, Jessica, Powers, Foster, Stevenson, Kristen E., Jones, Marcus Kenneth, Ng, Samuel Y., Wu, Gongwei, Jain, Salvia, Xu, Ran, Amaka, Sam, Trevisani, Christopher, Donaldson, Nicholas L., Hagner, Patrick R., de Leval, Laurence, Gaulard, Philippe, Iqbal, Javeed, Thakurta, Anjan, Fischer, Eric S., Adelman, Karen, Weinstock, David M.
Published in Blood (31.03.2022)
Published in Blood (31.03.2022)
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Journal Article
Leveraging gene expression subgroups to classify DLBCL patients and select for clinical benefit from a novel agent
Risueño, Alberto, Hagner, Patrick R., Towfic, Fadi, Fontanillo, Celia, Djebbari, Amira, Parker, Joel S., Drew, Clifton P., Nowakowski, Grzegorz S., Maurer, Matthew J., Cerhan, James R., Wei, Xin, Ren, Yan, Lee, Chung-Wein, Couto, Suzana, Wang, Maria, Pourdehnad, Michael, Gandhi, Anita K., Trotter, Matthew W.B.
Published in Blood (26.03.2020)
Published in Blood (26.03.2020)
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Journal Article
Transcriptomic classification of diffuse large B-cell lymphoma identifies a high-risk activated B-cell-like subpopulation with targetable MYC dysregulation
Stokes, Matthew E., Wenzl, Kerstin, Huang, C. Chris, Ortiz, María, Hsu, Chih-Chao, Maurer, Matthew J., Stong, Nicholas, Nakayama, Yumi, Wu, Lei, Chiu, Hsiling, Polonskaia, Ann, Danziger, Samuel A., Towfic, Fadi, Parker, Joel, King, Rebecca L., Link, Brian K., Slager, Susan L., Sarangi, Vivekananda, Asmann, Yan W., Novak, Joseph P., Sudhindra, Akshay, Ansell, Stephen M., Habermann, Thomas M., Hagner, Patrick R., Nowakowski, Grzegorz S., Cerhan, James R., Novak, Anne J., Gandhi, Anita K.
Published in Nature communications (08.08.2024)
Published in Nature communications (08.08.2024)
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Journal Article
ATM regulates a DNA damage response posttranscriptional RNA operon in lymphocytes
Mazan-Mamczarz, Krystyna, Hagner, Patrick R., Zhang, Yongqing, Dai, Bojie, Lehrmann, Elin, Becker, Kevin G., Keene, Jack D., Gorospe, Myriam, Liu, Zhenqui, Gartenhaus, Ronald B.
Published in Blood (24.02.2011)
Published in Blood (24.02.2011)
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Prolyl-tRNA synthetase as a novel therapeutic target in multiple myeloma
Kurata, Keiji, James-Bott, Anna, Tye, Mark A, Yamamoto, Leona, Samur, Mehmet K, Tai, Yu-Tzu, Dunford, James, Johansson, Catrine, Senbabaoglu, Filiz, Philpott, Martin, Palmer, Charlotte, Ramasamy, Karthik, Gooding, Sarah, Smilova, Mihaela, Gaeta, Giorgia, Guo, Manman, Christianson, John C, Payne, N Connor, Singh, Kritika, Karagoz, Kubra, Stokes, Matthew E, Ortiz, Maria, Hagner, Patrick, Thakurta, Anjan, Cribbs, Adam, Mazitschek, Ralph, Hideshima, Teru, Anderson, Kenneth C, Oppermann, Udo
Published in Blood cancer journal (New York) (12.01.2023)
Published in Blood cancer journal (New York) (12.01.2023)
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Journal Article
Functional and molecular interactions between ERK and CHK2 in diffuse large B-cell lymphoma
Dai, Bojie, Zhao, X Frank, Mazan-Mamczarz, Krystyna, Hagner, Patrick, Corl, Sharon, Bahassi, El Mustapha, Lu, Song, Stambrook, Peter J, Shapiro, Paul, Gartenhaus, Ronald B
Published in Nature communications (19.07.2011)
Published in Nature communications (19.07.2011)
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The C-Terminal Domain of Eukaryotic Initiation Factor 5 Promotes Start Codon Recognition by Its Dynamic Interplay with eIF1 and eIF2β
Luna, Rafael E., Arthanari, Haribabu, Hiraishi, Hiroyuki, Nanda, Jagpreet, Martin-Marcos, Pilar, Markus, Michelle A., Akabayov, Barak, Milbradt, Alexander G., Luna, Lunet E., Seo, Hee-Chan, Hyberts, Sven G., Fahmy, Amr, Reibarkh, Mikhail, Miles, David, Hagner, Patrick R., O'Day, Elizabeth M., Yi, Tingfang, Marintchev, Assen, Hinnebusch, Alan G., Lorsch, Jon R., Asano, Katsura, Wagner, Gerhard
Published in Cell reports (Cambridge) (28.06.2012)
Published in Cell reports (Cambridge) (28.06.2012)
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P997: FEDRATINIB IS EFFECTIVE IN RUXOLITINIB‐RESISTANT CELLS: CLINICAL AND PRECLINICAL CORRELATIONS
Jeyaraju, Danny, Hayati, Sheida, Polonskaia, Ann, Browne, Andrew, Risueño, Alberto, Hagner, Patrick, Gupta, Vikas, Talpaz, Moshe, Hernandez, Christopher, Chia, Vincent, Brown, Patrick, De Menezes, Daniel Lopes, La Motte‐Mohs, Ross, Nvs Suragani, Rajasekhar, Gandhi, Anita
Published in HemaSphere (08.08.2023)
Published in HemaSphere (08.08.2023)
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Journal Article
Phase Ib study of combinations of avadomide (CC‐122), CC‐223, CC‐292, and rituximab in patients with relapsed/refractory diffuse large B‐cell lymphoma
Ribrag, Vincent, Chavez, Julio C., Boccomini, Carola, Kaplan, Jason, Chandler, Jason C., Santoro, Armando, Corradini, Paolo, Flinn, Ian W., Advani, Ranjana, Cassier, Philippe A., Sangha, Randeep, Kenkre, Vaishalee P., Isufi, Iris, Uttamsingh, Shailaja, Hagner, Patrick R., Gandhi, Anita K., Shen, Frank, Michelliza, Sophie, Haeske, Harald, Hege, Kristen, Pourdehnad, Michael, Kuruvilla, John
Published in EJHaem (01.02.2022)
Published in EJHaem (01.02.2022)
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