Isoform-Selective ATAD2 Chemical Probe with Novel Chemical Structure and Unusual Mode of Action
Fernández-Montalván, Amaury E, Berger, Markus, Kuropka, Benno, Koo, Seong Joo, Badock, Volker, Weiske, Joerg, Puetter, Vera, Holton, Simon J, Stöckigt, Detlef, ter Laak, Antonius, Centrella, Paolo A, Clark, Matthew A, Dumelin, Christoph E, Sigel, Eric A, Soutter, Holly H, Troast, Dawn M, Zhang, Ying, Cuozzo, John W, Keefe, Anthony D, Roche, Didier, Rodeschini, Vincent, Chaikuad, Apirat, Díaz-Sáez, Laura, Bennett, James M, Fedorov, Oleg, Huber, Kilian V. M, Hübner, Jan, Weinmann, Hilmar, Hartung, Ingo V, Gorjánácz, Mátyás
Published in ACS chemical biology (17.11.2017)
Published in ACS chemical biology (17.11.2017)
Get full text
Journal Article
Abstract 5084: Potent and isoform-selective ATAD2 bromodomain inhibitor with unprecedented chemical structure and mode of action
Fernández-Montalván, Amaury E., Berger, Markus, Kuropka, Benno, Koo, Seong Joo, Badock, Volker, Weiske, Joerg, Holton, Simon J., Chaikuad, Apirat, Díaz-Sáez, Laura, Bennett, James, Federov, Oleg, Huber, Kilian, Centrella, Paolo, Clark, Matthew A., Dumelin, Christoph E., Sigel, Eric A., Soutter, Holly S., Troast, Dawn M., Zhang, Ying, Cuozzo, John W., Keefe, Anthony D., Roche, Didier, Rodeschini, Vincent, Hübner, Jan, Weinmann, Hilmar, Hartung, Ingo V., Gorjanacz, Matyas
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Get full text
Journal Article
Furane derivatives as inhibitors of ATAD2
Hübner, Jan, Gorjanacz, Matyas, Berger, Markus, Rodeschini, Vincent, Ter Laak, Antonius, Roche, Didier, Fernandez-Montalvan, Amaury Ernesto
Year of Publication 19.05.2020
Get full text
Year of Publication 19.05.2020
Patent
FURANE DERIVATIVES AS INHIBITORS OF ATAD2
GORJANACZ, Matyas, ROCHE, Didier, FERNANDEZ-MONTALVAN, Amaury Ernesto, TER LAAK, Antonius, HÜBNER, Jan, BERGER, Markus, RODESCHINI, Vincent
Year of Publication 29.01.2020
Get full text
Year of Publication 29.01.2020
Patent
FURANE DERIVATIVES AS INHIBITORS OF ATAD2
GORJANACZ, Matyas, ROCHE, Didier, FERNANDEZ-MONTALVAN, Amaury Ernesto, TER LAAK, Antonius, HÜBNER, Jan, BERGER, Markus, RODESCHINI, Vincent
Year of Publication 18.07.2019
Get full text
Year of Publication 18.07.2019
Patent
FURANE DERIVATIVES AS INHIBITORS OF ATAD2
GORJANACZ, Matyas, ROCHE, Didier, FERNANDEZ-MONTALVAN, Amaury Ernesto, TER LAAK, Antonius, HÜBNER, Jan, BERGER, Markus, RODESCHINI, Vincent
Year of Publication 10.10.2018
Get full text
Year of Publication 10.10.2018
Patent
FURANE DERIVATIVES AS INHIBITORS OF ATAD2
GORJANNACZ, Matyas, ROCHE, Didier, FERNANDEZ-MONTALVAN, Amaury Ernesto, TER LAAK, Antonius, HÜBNER, Jan, BERGER, Markus, RODESCHINI, Vincent
Year of Publication 08.06.2017
Get full text
Year of Publication 08.06.2017
Patent
18 METHYL 6 7 METHYLENE 3 OXO 17 PREGN 4 ENE 21 17? CARBOLACTONES PHARMACEUTICAL PREPARATIONS COMPRISING SAID COMPOUNDS AND USE THEREOF IN THE TREATMENT OF ENDOMETRIOSIS
GALLUS NORBERT, TEREBESI ILDIKO, KUHNKE JOACHIM, HÜBNER JAN, BOHLMANN ROLF, GASHAW ISABELLA, NUBBEMEYER REINHARD, FISCHER OLIVER MARTIN
Year of Publication 03.07.2015
Get full text
Year of Publication 03.07.2015
Patent
ΠΑΡΑΓΩΓΑ 5-ΥΠΟΚΑΤΕΣΤΗΜΕΝΗΣ ΚΙΝΟΛΙΝΗΣ ΚΑΙ ΙΣΟΚΙΝΟΛΙΝΗΣ· ΜΕΘΟΔΟΣ ΓΙΑ ΤΗΝ ΠΑΡΑΓΩΓΗ ΤΟΥΣ ΚΑΙ Η ΧΡΗΣΗ ΤΟΥΣ ΩΣ ΑΝΤΙΦΛΕΓΜΟΝΩΔΗ
JAROCH STEFAN, PETROV ORLIN, HÜBNER JAN, DINTER CHRISTIAN, SCHÄCKE HEIKE, SCHNEIDER MATTHIAS, SCHMEES NORBERT, REHWINKEL HARTMUT, SKUBALA WERNER
Year of Publication 29.04.2015
Get full text
Year of Publication 29.04.2015
Patent
"17beta-alquil-17alfa-óxi-estratrienos"
JENS HOFFMANN, MICHAEL SANDER, ROLF BOHLMANN, SILKE KÖHR, TIM WINTERMANTEL, DIETER LANG, HERMANN KÜNZER, KARSTEN DENNER, GEORG KETTSCHAU, NIKOLAUS HEINRICH, PHILIP LIENAU, JAN HÜBNER, MICHAEL GERISCH
Year of Publication 29.03.2016
Get full text
Year of Publication 29.03.2016
Patent
18-METHYL-6,7-METHYLENE-3-OXO-17-PREGN-4-ENE-21,17B-CARBOLACTONES, PHARMACEUTICAL PREPARATIONS COMPRISING SAID COMPOUNDS AND USE THEREOF IN THE TREATMENT OF ENDOMETRIOSIS
GALLUS NORBERT, TEREBESI ILDIKO, KUHNKE JOACHIM, HÜBNER JAN, BOHLMANN ROLF, GASHAW ISABELLA, NUBBEMEYER REINHARD, FISCHER OLIVER MARTIN
Year of Publication 25.09.2014
Get full text
Year of Publication 25.09.2014
Patent
Derivado de 17-(-1'-propenil)-17-3'-oxidoestra-4-en-3-ona, seu uso e o medicamento contendo o derivado
HANS PETER MUHN, STEFFEN BORDEN, FREDERIK MENGES, KATJA PRELLE, THOMAS FRENZEL, ROLF BOHLMANN, SVEN RING, JAN HÜBNER, ULRICH KLAR, JOACHIM KUHNKE
Year of Publication 23.06.2015
Get full text
Year of Publication 23.06.2015
Patent
Derivado esteroide de gama-lactona de ácido 17-hidróxi-19-nor-21-carboxílico, uso do mesmo e medicamento que contém o derivado
HANS PETER MUHN, STEFFEN BORDEN, FREDERIK MENGES, KATJA PRELLE, THOMAS FRENZEL, ROLF BOHLMANN, SVEN RING, JAN HÜBNER, ULRICH KLAR, JOACHIM KUHNKE
Year of Publication 16.06.2015
Get full text
Year of Publication 16.06.2015
Patent
Derivados 19-nor-esteroides com um grupo 15alfa, 16alfa-metileno e um anel 17, 17-espirolactona saturado, uso deste e produtos medicinais contendo esses derivados
HANS-PETER MUHN, STEFFEN BORDEN, FREDERIK MENGES, KATJA PRELLE, THOMAS FRENZEL, ROLF BOHLMANN, SVEN RING, JAN HÜBNER, ULRICH KLAR, JOACHIM KUHNKE
Year of Publication 16.06.2015
Get full text
Year of Publication 16.06.2015
Patent
Derivado de gama-lactona esteroide de ácido 15,16-metileno-17-hidróxi-19-nor-21-carboxílico, seu uso e medicamentos contendo o derivado
HANS PETER MUHN, STEFFEN BORDEN, FREDERIK MENGES, KATJA PRELLE, THOMAS FRENZEL, ROLF BOHLMANN, SVEN RING, JAN HÜBNER, ULRICH KLAR, JOACHIM KUHNKE
Year of Publication 16.06.2015
Get full text
Year of Publication 16.06.2015
Patent
Derivado de 15, 16-metileno-17-(1'-propenil)-17,3'-oxidoestra-4-em-3-on a, seu uso e medicamentos contendo o derivado
HANS PETER MUHN, STEFFEN BORDEN, FREDERIK MENGES, KATJA PRELLE, THOMAS FRENZEL, ROLF BOHLMANN, SVEN RING, JAN HÜBNER, ULRICH KLAR, JOACHIM KUHNKE
Year of Publication 16.06.2015
Get full text
Year of Publication 16.06.2015
Patent