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HETEROCYCLIC INHIBITORS OF GLUTAMINASE
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HETEROCYCLIC INHIBITORS OF GLUTAMINASE
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Year of Publication 15.12.2016
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The Selective Proteasome Inhibitor Carfilzomib Is Well Tolerated in Experimental Animals with Dose Intensive Administration
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Published in Blood (16.11.2008)
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Anti-Tumor Activity of Immunoproteasome Selective Inhibitors
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Immunoproteasome-Selective Keto-Epoxide Inhibitors: Potential Therapeutic Agents for the Treatment of Hematological Disorders
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Identification of Peptide Epoxy-Ketone Proteasome Inhibitors with Differential Active Site Selectivity
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A Proteasome Specific Binding Assay for Quantitation of Constitutive and Immunoproteasome Active Sites
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Pharmacokinetics, Pharmacodynamics and Anti-Tumor Efficacy of PR-171, a Novel Inhibitor of the 20S Proteasome
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Published in Blood (16.11.2005)
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Biochemical and Cellular Characterization of the Novel Proteasome Inhibitor PR-171
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Published in Blood (16.11.2005)
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