Blocking an N-terminal acetylation-dependent protein interaction inhibits an E3 ligase
Scott, Daniel C, Hammill, Jared T, Min, Jaeki, Rhee, David Y, Connelly, Michele, Sviderskiy, Vladislav O, Bhasin, Deepak, Chen, Yizhe, Ong, Su-Sien, Chai, Sergio C, Goktug, Asli N, Huang, Guochang, Monda, Julie K, Low, Jonathan, Kim, Ho Shin, Paulo, Joao A, Cannon, Joe R, Shelat, Anang A, Chen, Taosheng, Kelsall, Ian R, Alpi, Arno F, Pagala, Vishwajeeth, Wang, Xusheng, Peng, Junmin, Singh, Bhuvanesh, Harper, J Wade, Schulman, Brenda A, Guy, R Kip
Published in Nature chemical biology (01.08.2017)
Published in Nature chemical biology (01.08.2017)
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Journal Article
High-throughput assays for promiscuous inhibitors
Guy, R Kip, Shoichet, Brian K, Feng, Brian Y, Shelat, Anang, Doman, Thompson N
Published in Nature chemical biology (01.08.2005)
Published in Nature chemical biology (01.08.2005)
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Journal Article
Planarity and Constraint of the Carbonyl Groups in 1,2-Diones Are Determinants for Selective Inhibition of Human Carboxylesterase 1
Hyatt, Janice L, Wadkins, Randy M, Tsurkan, Lyudmila, Hicks, Latorya D, Hatfield, M. Jason, Edwards, Carol C, Ross, Charles R, Cantalupo, Stephanie A, Crundwell, Guy, Danks, Mary K, Guy, R. Kip, Potter, Philip M
Published in Journal of medicinal chemistry (15.11.2007)
Published in Journal of medicinal chemistry (15.11.2007)
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Journal Article
Chemical approaches to nuclear receptors in metabolism
Margolis, Ronald N, Moore, David D, Willson, Timothy M, Guy, R Kip
Published in Science signaling (04.08.2009)
Published in Science signaling (04.08.2009)
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Journal Article
A New Script to Refill the Pharmacy Pipeline
Hudspeth, Brooke, Howington, Gavin, Matson, Adrienne W., Edwards, Jason, Mejia-Cruz, Rosa, Jones, Mandy, Guy, R. Kip
Published in American journal of pharmaceutical education (01.08.2023)
Published in American journal of pharmaceutical education (01.08.2023)
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Journal Article
An Integrated In Vitro and In Vivo High-Throughput Screen Identifies Treatment Leads for Ependymoma
Atkinson, Jennifer M., Shelat, Anang A., Carcaboso, Angel Montero, Kranenburg, Tanya A., Arnold, Leggy A., Boulos, Nidal, Wright, Karen, Johnson, Robert A., Poppleton, Helen, Mohankumar, Kumarasamypet M., Féau, Clementine, Phoenix, Timothy, Gibson, Paul, Zhu, Liqin, Tong, Yiai, Eden, Chris, Ellison, David W., Priebe, Waldemar, Koul, Dimpy, Yung, W. K. Alfred, Gajjar, Amar, Stewart, Clinton F., Guy, R. Kiplin, Gilbertson, Richard J.
Published in Cancer cell (13.09.2011)
Published in Cancer cell (13.09.2011)
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Journal Article
PCM-22A NEW APPROACH OF PRECLINICAL TESTING OF CHEMOTHERAPIES - AN EXAMPLE OF BRAIN TUMOUR THERAPY
Nimmervoll, Birgit, Patel, Yogesh, Bianski, Brandon, DeCuypere, Michael, Shelat, Anang, Stewart, Clinton, Merchant, Tom, Guy, R. Kip, Gilbertson, Richard
Published in Neuro-oncology (Charlottesville, Va.) (01.06.2016)
Published in Neuro-oncology (Charlottesville, Va.) (01.06.2016)
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Journal Article
Abstract 4522: Identification of small molecule agonists/activators of BMP-2, 4, 7 signaling
Vrijens, Karen, Lin, Wenwei, Cui, Jimmy, Shelat, Anang, Taylor, Michael, Guy, Kip R., Chen, Taosheng, Roussel, Martine F.
Published in Cancer research (Chicago, Ill.) (15.04.2011)
Published in Cancer research (Chicago, Ill.) (15.04.2011)
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Journal Article
Abstract A52: An interspecies genomics based high-throughput screen for novel treatments of ependymoma
Atkinson, Jennifer M., Shelat, Anang, Johnson, Robert, Wright, Karen, Poppleton, Helen, Mohankumar, Kumarasamypet M., Feau, Clementine, Arnold, Alexander, White, Elsie, Kranenburg, Tanya, Guy, R. Kip, Gilbertson, Richard J.
Published in Molecular cancer therapeutics (10.12.2009)
Published in Molecular cancer therapeutics (10.12.2009)
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Journal Article
Tetrahydroquinoline-based bromodomain inhibitors
Boyd, Vincent A, Shelat, Anang, Shadrick, William Robert, Slavish, P Jake, Guy, R. Kip, Bharatham, Nagakumar, Young, Brandon M, Price, Jeanine E
Year of Publication 17.10.2023
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Year of Publication 17.10.2023
Patent
TETRAHYDROQUINOLINE-BASED BROMODOMAIN INHIBITORS
Boyd, Vincent A, Shelat, Anang, Shadrick, William Robert, Slavish, P. Jake, Guy, R. Kip, Bharatham, Nagakumar, Young, Brandon M, Price, Jeanine E
Year of Publication 24.06.2021
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Year of Publication 24.06.2021
Patent
Tetrahydroquinoline-based bromodomain inhibitors
Boyd, Vincent A, Shelat, Anang, Shadrick, William Robert, Slavish, P. Jake, Guy, R. Kip, Bharatham, Nagakumar, Young, Brandon M, Price, Jeanine E
Year of Publication 08.06.2021
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Year of Publication 08.06.2021
Patent
TETRAHYDROQUINOLINE-BASED BROMODOMAIN INHIBITORS
Boyd, Vincent A, Shelat, Anang, Shadrick, William Robert, Slavish, P. Jake, Guy, R. Kip, Bharatham, Nagakumar, Young, Brandon M, Price, Jeanine E
Year of Publication 12.03.2020
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Year of Publication 12.03.2020
Patent
Method for treating ocular cancer
JOSEN AART GERRIT, ZHU FANGYI, MARINE JEANRISTOPHE, GUY R. KIP, DYER MICHAEL A
Year of Publication 25.06.2013
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Year of Publication 25.06.2013
Patent