Discovery of Novel Boron-Containing N-Substituted Oseltamivir Derivatives as Anti-Influenza A Virus Agents for Overcoming N1-H274Y Oseltamivir-Resistant
Jia, Ruifang, Zhang, Jiwei, Zhang, Jian, Bertagnin, Chiara, Bonomini, Anna, Guizzo, Laura, Gao, Zhen, Ji, Xiangkai, Li, Zhuo, Liu, Chuanfeng, Ju, Han, Ma, Xiuli, Loregian, Arianna, Huang, Bing, Zhan, Peng, Liu, Xinyong
Published in Molecules (Basel, Switzerland) (29.09.2022)
Published in Molecules (Basel, Switzerland) (29.09.2022)
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A novel N-heterocycles substituted oseltamivir derivatives as potent inhibitors of influenza virus neuraminidase: discovery, synthesis and biological evaluation
Zhang, Jiwei, Liu, Chuanfeng, Jia, Ruifang, Zhang, Xujie, Zhang, Jian, Bertagnin, Chiara, Bonomini, Anna, Guizzo, Laura, Jiang, Yuanmin, Jia, Huinan, Jia, Shuzhen, Ma, Xiuli, Loregian, Arianna, Huang, Bing, Zhan, Peng, Liu, Xinyong
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2023)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2023)
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Journal Article
Identification of C5-NH2 Modified Oseltamivir Derivatives as Novel Influenza Neuraminidase Inhibitors with Highly Improved Antiviral Activities and Favorable Druggability
Ju, Han, Murugan, N. Arul, Hou, Lingxin, Li, Ping, Guizzo, Laura, Zhang, Ying, Bertagnin, Chiara, Kong, Xiujie, Kang, Dongwei, Jia, Ruifang, Ma, Xiuli, Du, Ruikun, Poongavanam, Vasanthanathan, Loregian, Arianna, Huang, Bing, Liu, Xinyong, Zhan, Peng
Published in Journal of medicinal chemistry (23.12.2021)
Published in Journal of medicinal chemistry (23.12.2021)
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Iterative Optimization and Structure–Activity Relationship Studies of Oseltamivir Amino Derivatives as Potent and Selective Neuraminidase Inhibitors via Targeting 150-Cavity
Ju, Han, Hou, Lingxin, Zhao, Fabao, Zhang, Ying, Jia, Ruifang, Guizzo, Laura, Bonomini, Anna, Zhang, Jiwei, Gao, Zhen, Liang, Ruipeng, Bertagnin, Chiara, Kong, Xiujie, Ma, Xiuli, Kang, Dongwei, Loregian, Arianna, Huang, Bing, Liu, Xinyong, Zhan, Peng
Published in Journal of medicinal chemistry (08.09.2022)
Published in Journal of medicinal chemistry (08.09.2022)
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Journal Article
Identification of C5-NH 2 Modified Oseltamivir Derivatives as Novel Influenza Neuraminidase Inhibitors with Highly Improved Antiviral Activities and Favorable Druggability
Ju, Han, Murugan, N Arul, Hou, Lingxin, Li, Ping, Guizzo, Laura, Zhang, Ying, Bertagnin, Chiara, Kong, Xiujie, Kang, Dongwei, Jia, Ruifang, Ma, Xiuli, Du, Ruikun, Poongavanam, Vasanthanathan, Loregian, Arianna, Huang, Bing, Liu, Xinyong, Zhan, Peng
Published in Journal of medicinal chemistry (23.12.2021)
Published in Journal of medicinal chemistry (23.12.2021)
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Journal Article
Discovery of Novel Boron-Containing IN/I-Substituted Oseltamivir Derivatives as Anti-Influenza A Virus Agents for Overcoming N1-H274Y Oseltamivir-Resistant
Jia, Ruifang, Zhang, Jiwei, Zhang, Jian, Bertagnin, Chiara, Bonomini, Anna, Guizzo, Laura, Gao, Zhen, Ji, Xiangkai, Li, Zhuo, Liu, Chuanfeng, Ju, Han, Ma, Xiuli, Loregian, Arianna, Huang, Bing, Zhan, Peng, Liu, Xinyong
Published in Molecules (Basel, Switzerland) (01.09.2022)
Published in Molecules (Basel, Switzerland) (01.09.2022)
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Journal Article