Hybrid topoisomerase I and HDAC inhibitors as dual action anticancer agents
Cincinelli, Raffaella, Musso, Loana, Artali, Roberto, Guglielmi, Mario B, La Porta, Ilaria, Melito, Carmela, Colelli, Fabiana, Cardile, Francesco, Signorino, Giacomo, Fucci, Alessandra, Frusciante, Martina, Pisano, Claudio, Dallavalle, Sabrina
Published in PloS one (09.10.2018)
Published in PloS one (09.10.2018)
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Journal Article
Antitumor activity of novel POLA1-HDAC11 dual inhibitors
Dallavalle, Sabrina, Musso, Loana, Cincinelli, Raffaella, Darwiche, Nadine, Gervasoni, Silvia, Vistoli, Giulio, Guglielmi, Mario B., La Porta, Ilaria, Pizzulo, Maddalena, Modica, Elisa, Prosperi, Federica, Signorino, Giacomo, Colelli, Fabiana, Cardile, Francesco, Fucci, Alessandra, D'Andrea, Egildo Luca, Riccio, Assunta, Pisano, Claudio
Published in European journal of medicinal chemistry (15.01.2022)
Published in European journal of medicinal chemistry (15.01.2022)
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Journal Article
Alkyl-guanidine Compounds as Potent Broad-Spectrum Antibacterial Agents: Chemical Library Extension and Biological Characterization
Pasero, Carolina, D’Agostino, Ilaria, De Luca, Filomena, Zamperini, Claudio, Deodato, Davide, Truglio, Giuseppina I, Sannio, Filomena, Del Prete, Rosita, Ferraro, Teresa, Visaggio, Daniela, Mancini, Arianna, Guglielmi, Mario B, Visca, Paolo, Docquier, Jean-Denis, Botta, Maurizio
Published in Journal of medicinal chemistry (25.10.2018)
Published in Journal of medicinal chemistry (25.10.2018)
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Synthesis and Evaluation of New Hsp90 Inhibitors Based on a 1,4,5-Trisubstituted 1,2,3-Triazole Scaffold
Taddei, Maurizio, Ferrini, Serena, Giannotti, Luca, Corsi, Massimo, Manetti, Fabrizio, Giannini, Giuseppe, Vesci, Loredana, Milazzo, Ferdinando M, Alloatti, Domenico, Guglielmi, Mario B, Castorina, Massimo, Cervoni, Maria L, Barbarino, Marcella, Foderà, Rosanna, Carollo, Valeria, Pisano, Claudio, Armaroli, Silvia, Cabri, Walter
Published in Journal of medicinal chemistry (27.03.2014)
Published in Journal of medicinal chemistry (27.03.2014)
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Journal Article
Novel adamantyl retinoid-related molecules with POLA1 inhibitory activity
Cincinelli, Raffaella, Musso, Loana, Guglielmi, Mario B., La Porta, Ilaria, Fucci, Alessandra, Luca D'Andrea, Egildo, Cardile, Francesco, Colelli, Fabiana, Signorino, Giacomo, Darwiche, Nadine, Gervasoni, Silvia, Vistoli, Giulio, Pisano, Claudio, Dallavalle, Sabrina
Published in Bioorganic chemistry (01.11.2020)
Published in Bioorganic chemistry (01.11.2020)
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Journal Article
Novel Combretastatin Analogues Endowed with Antitumor Activity
Simoni, Daniele, Romagnoli, Romeo, Baruchello, Riccardo, Rondanin, Riccardo, Rizzi, Michele, Pavani, Maria Giovanna, Alloatti, Domenico, Giannini, Giuseppe, Marcellini, Marcella, Riccioni, Teresa, Castorina, Massimo, Guglielmi, Mario B, Bucci, Federica, Carminati, Paolo, Pisano, Claudio
Published in Journal of medicinal chemistry (01.06.2006)
Published in Journal of medicinal chemistry (01.06.2006)
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Journal Article
Novel 3,4-Isoxazolediamides as Potent Inhibitors of Chaperone Heat Shock Protein 90
Baruchello, Riccardo, Simoni, Daniele, Grisolia, Giuseppina, Barbato, Giuseppina, Marchetti, Paolo, Rondanin, Riccardo, Mangiola, Stefania, Giannini, Giuseppe, Brunetti, Tiziana, Alloatti, Domenico, Gallo, Grazia, Ciacci, Andrea, Vesci, Loredana, Castorina, Massimo, Milazzo, Ferdinando M, Cervoni, Maria L, Guglielmi, Mario B, Barbarino, Marcella, Foderà, Rosanna, Pisano, Claudio, Cabri, Walter
Published in Journal of medicinal chemistry (22.12.2011)
Published in Journal of medicinal chemistry (22.12.2011)
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Journal Article
Synthesis and Biological Activity of Fluorinated Combretastatin Analogues
Alloatti, Domenico, Giannini, Giuseppe, Cabri, Walter, Lustrati, Isabella, Marzi, Mauro, Ciacci, Andrea, Gallo, Grazia, Tinti, M. Ornella, Marcellini, Marcella, Riccioni, Teresa, Guglielmi, Mario B, Carminati, Paolo, Pisano, Claudio
Published in Journal of medicinal chemistry (08.05.2008)
Published in Journal of medicinal chemistry (08.05.2008)
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Journal Article
Abstract 3096: Host antitumor immune response activated by Dual POLA1-HDAC11 inhibitors endowed with a large spectrum of antitumor activity
Pisano, Claudio, Merlini, Lucio, Penco, Sergio, Cincinelli, Raffaella, Darwiche, Nadine, Guglielmi, Mario B., Porta, Ilaria La, Pizzulo, Maddalena, Prosperi, Federica, Signorino, Giacomo, Colelli, Fabiana, Cardile, Francesco, Focareta, Laura, Fucci, Alessandra, D'Andrea, Egildo L., Riccio, Assunta, Dallavalle, Sabrina
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
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Journal Article
Abstract 4848: Preclinical antitumor activity of novel DNA polymerase 1 (POLA1) inhibitors
Pisano, Claudio, Merlini, Lucio, Penco, Sergio, Cincinelli, Raffaella, Darwiche, Nadine, Guglielmi, Mario B., Porta, Ilaria La, Signorino, Giacomo, Rubis, Gabriele De, Colelli, Fabiana, Cardile, Francesco, Fucci, Alessandra, D'Andrea, Egildo L., Dallavalle, Sabrina
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Abstract 2936: Molecular profiling of primary malignant pleuralmesothelioma histotypes cell lines reveals relationship between GDF15overexpression and cisplatin resistance both in in vitro and in vivo models
Pisano, Claudio, Carletta, Gianluca, D’Angelo, Fulvio, Esposito, Antonietta, Bianchino, Erminia, Riccio, Assunta, Festa, Michela, Cardile, Francesco, Carchia, Emanuele, D’Acunto, Walter, Signorino, Giacomo, Guglielmi, Mario B., De Luca, Pasquale
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Journal Article
Abstract 4195: MIR002: a new POLA1 inhibitor endowed with a large spectrum of antitumor activity
Pisano, Claudio, Merlini, Lucio, Penco, Sergio, Cincinelli, Raffaella, Darwiche, Nadine, Guglielmi, Mario B., Esposito, Antonietta, Porta, Ilaria La, Signorino, Giacomo, Rubis, Gabriele De, Colelli, Fabiana, Cardile, Francesco, Fucci, Alessandra, D'Andrea, Egildo L., Dallavalle, Sabrina
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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Journal Article
Abstract 1774: Dihydroartemisinin (DHA): A potent enhancer of PARP inhibitors and DNA-damaging agents activity in human tumor models
Pisano, Claudio, Vesci, Loredana, Milazzo, Ferdinando M., Guglielmi, Mario B., Barbarino, Marcella, Beghetto, Elisa, Brughera, Marco M.
Published in Cancer research (Chicago, Ill.) (15.04.2012)
Published in Cancer research (Chicago, Ill.) (15.04.2012)
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Journal Article
Abstract 2623: ST3595, a new histone deacetylase (HDAC) inhibitor endowed with a peculiar mechanism of action
Pisano, Claudio, Vesci, Loredana, Milazzo, Ferdinando M., Guglielmi, Mario B., Barbarino, Marcella, Foderà, Rosanna, Zuco, Valentina, Zunino, Franco
Published in Cancer research (Chicago, Ill.) (15.04.2011)
Published in Cancer research (Chicago, Ill.) (15.04.2011)
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Journal Article
The role of the tumor suppressor gene p53 in cardiomyocyte apoptosis: Apoptosis
CROW, M. T, XILIN LONG, GUGIIELMI, M. B, ASAI, T, LAKATTA, E. G
Published in Heart failure reviews (1998)
Published in Heart failure reviews (1998)
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