Revisiting Proteasome Inhibitors: Molecular Underpinnings of Their Development, Mechanisms of Resistance and Strategies to Overcome Anti-Cancer Drug Resistance
Leonardo-Sousa, Carlota, Carvalho, Andreia Neves, Guedes, Romina A, Fernandes, Pedro M P, Aniceto, Natália, Salvador, Jorge A R, Gama, Maria João, Guedes, Rita C
Published in Molecules (Basel, Switzerland) (28.03.2022)
Published in Molecules (Basel, Switzerland) (28.03.2022)
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Journal Article
Highlights in USP7 inhibitors for cancer treatment
Oliveira, Rita I., Guedes, Romina A., Salvador, Jorge A. R.
Published in Frontiers in chemistry (15.09.2022)
Published in Frontiers in chemistry (15.09.2022)
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Journal Article
Disclosing the antitumour potential of the marine bromoditerpene sphaerococcenol A on distinct cancer cellular models
Alves, Celso, Silva, Joana, Afonso, Marta B., Guedes, Romina A., Guedes, Rita C., Alvariño, Rebeca, Pinteus, Susete, Gaspar, Helena, Goettert, Márcia I., Alfonso, Amparo, Rodrigues, Cecília M.P., Alpoím, Maria C., Botana, Luis, Pedrosa, Rui
Published in Biomedicine & pharmacotherapy (01.05.2022)
Published in Biomedicine & pharmacotherapy (01.05.2022)
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Bromoditerpenes from the Red Seaweed Sphaerococcus coronopifolius as Potential Cytotoxic Agents and Proteasome Inhibitors and Related Mechanisms of Action
Alves, Celso, Silva, Joana, Pintéus, Susete, Guedes, Romina A., Guedes, Rita C., Alvariño, Rebeca, Freitas, Rafaela, Goettert, Márcia I., Gaspar, Helena, Alfonso, Amparo, Alpoím, Maria C., Botana, Luis M., Pedrosa, Rui
Published in Marine drugs (20.10.2022)
Published in Marine drugs (20.10.2022)
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Journal Article
Computational Approaches for the Discovery of Human Proteasome Inhibitors: An Overview
Guedes, Romina A, Serra, Patrícia, Salvador, Jorge A R, Guedes, Rita C
Published in Molecules (Basel, Switzerland) (16.07.2016)
Published in Molecules (Basel, Switzerland) (16.07.2016)
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New Scaffolds of Proteasome Inhibitors: Boosting Anticancer Potential by Exploiting the Synergy of In Silico and In Vitro Methodologies
Guedes, Romina A, Grilo, Jorge H, Carvalho, Andreia N, Fernandes, Pedro M. P, Ressurreição, Ana S, Brito, Vanessa, Santos, Adriana O, Silvestre, Samuel, Gallerani, Eleonora, Gama, Maria João, Gavioli, Riccardo, Salvador, Jorge A. R, Guedes, Rita C
Published in Pharmaceuticals (Basel, Switzerland) (01.08.2023)
Published in Pharmaceuticals (Basel, Switzerland) (01.08.2023)
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Journal Article
Artificial intelligence for prediction of biological activities and generation of molecular hits using stereochemical information
Pereira, Tiago O., Abbasi, Maryam, Oliveira, Rita I., Guedes, Romina A., Salvador, Jorge A. R., Arrais, Joel P.
Published in Journal of computer-aided molecular design (01.12.2023)
Published in Journal of computer-aided molecular design (01.12.2023)
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Journal Article
Optimization of O 3‑Acyl Kojic Acid Derivatives as Potent and Selective Human Neutrophil Elastase Inhibitors
Lucas, Susana D, Gonçalves, Lídia M, Carvalho, Luís A. R, Correia, Henrique F, Da Costa, Eduardo M. R, Guedes, Romina A, Moreira, Rui, Guedes, Rita C
Published in Journal of medicinal chemistry (12.12.2013)
Published in Journal of medicinal chemistry (12.12.2013)
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Journal Article
3-Hydroxypyrrolidine and (3,4)-dihydroxypyrrolidine derivatives: Inhibition of rat intestinal α-glucosidase
Carreiro, Elisabete P., Louro, Patrícia, Adriano, Gizé, Guedes, Romina A., Vannuchi, Nicholas, Costa, Ana R., Antunes, Célia M.M., Guedes, Rita C., Burke, A.J.
Published in Bioorganic chemistry (01.06.2014)
Published in Bioorganic chemistry (01.06.2014)
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Journal Article
Optimization of O3-acyl kojic acid derivatives as potent and selective human neutrophil elastase inhibitors
Lucas, Susana D, Gonçalves, Lídia M, Carvalho, Luís A R, Correia, Henrique F, Da Costa, Eduardo M R, Guedes, Romina A, Moreira, Rui, Guedes, Rita C
Published in Journal of medicinal chemistry (12.12.2013)
Published in Journal of medicinal chemistry (12.12.2013)
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