The Ligands of Translocator Protein: Design and Biological Properties
Mokrov, Grigory V, Deeva, Olga A, Gudasheva, Tatiana A
Published in Current pharmaceutical design (2021)
Published in Current pharmaceutical design (2021)
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Novel Technologies for Dipeptide Drugs Design and their Implantation
Gudasheva, Tatiana A, Ostrovskaya, Rita U, Seredenin, Sergey B
Published in Current pharmaceutical design (01.01.2018)
Published in Current pharmaceutical design (01.01.2018)
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Сhronically Administered BDNF Dipeptide Mimetic GSB-106 Prevents the Depressive-like Behavior and Memory Impairments after Transient Middle Cerebral Artery Occlusion in Rats
Povarnina, Polina Y, Antipova, Tatyana A, Logvinov, Ilya O, Gudasheva, Tatiana A, Seredenin, Sergey B
Published in Current pharmaceutical design (2023)
Published in Current pharmaceutical design (2023)
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Journal Article
Analysis of Antidepressant-like Effects and Action Mechanisms of GSB-106, a Small Molecule, Affecting the TrkB Signaling
Vakhitova, Yulia V, Kalinina, Tatiana S, Zainullina, Liana F, Lusta, Anastasiya Yu, Volkova, Anna V, Kudryashov, Nikita V, Gudasheva, Tatiana A, Shimshirt, Alexander A, Kadnikov, Ilya A, Voronin, Mikhail V, Seredenin, Sergei B
Published in International journal of molecular sciences (13.12.2021)
Published in International journal of molecular sciences (13.12.2021)
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Journal Article
The New Dipeptide TSPO Ligands: Design, Synthesis and Structure-Anxiolytic Activity Relationship
Gudasheva, Tatiana A, Deeva, Olga A, Pantileev, Andrey S, Mokrov, Grigory V, Rybina, Inna V, Yarkova, Milada A, Seredenin, Sergei B
Published in Molecules (Basel, Switzerland) (04.11.2020)
Published in Molecules (Basel, Switzerland) (04.11.2020)
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Journal Article
Neuroregenerative Activity of the Dipeptide Mimetic of Brain-derived Neurotrophic Factor GSB-106 Under Experimental Ischemic Stroke
Gudasheva, Tatiana A, Povarnina, Polina Y, Antipova, Tatiana A, Kruglov, Sergey V, Logvinov, Ilya O, Nikiforov, Dmitry M, Seredenin, Sergey B
Published in CNS & neurological disorders drug targets (2021)
Published in CNS & neurological disorders drug targets (2021)
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Antidepressant-like Effects of BDNF and NGF Individual Loop Dipeptide Mimetics Depend on the Signal Transmission Patterns Associated with Trk
Mezhlumyan, Armen G, Tallerova, Anna V, Povarnina, Polina Y, Tarasiuk, Aleksey V, Sazonova, Nellya M, Gudasheva, Tatiana A, Seredenin, Sergey B
Published in Pharmaceuticals (Basel, Switzerland) (24.02.2022)
Published in Pharmaceuticals (Basel, Switzerland) (24.02.2022)
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Journal Article
Low-Molecular Weight BDNF Mimetic, Dimeric Dipeptide GSB-106, Reverses Depressive Symptoms in Mouse Chronic Social Defeat Stress
Gudasheva, Tatiana A, Tallerova, Anna V, Mezhlumyan, Armen G, Antipova, Tatyana A, Logvinov, Ilya O, Firsova, Yulia N, Povarnina, Polina Y, Seredenin, Sergey B
Published in Biomolecules (Basel, Switzerland) (10.02.2021)
Published in Biomolecules (Basel, Switzerland) (10.02.2021)
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Journal Article
Design, Synthesis and Anxiolytic Activity Evaluation of N-Acyltryptophanyl- Containing Dipeptides, Potential TSPO Ligands
Gudasheva, Tatiana A, Deeva, Olga A, Mokrov, Grigory V, Dyabina, Alina S, Yarkova, Milada A, Seredenin, Sergey B
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (2019)
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (2019)
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Low molecular weight NGF mimetic GK‐2 normalizes the parameters of glucose and lipid metabolism and exhibits a hepatoprotective effect on a prediabetes model in obese Wistar rats
Ivanov, Sergei V., Ostrovskaya, Rita U., Koliasnikova, Ksenia N., Alchinova, Irina B., Demorzhi, Marina S., Gudasheva, Tatiana A., Seredenin, Sergei B.
Published in Clinical and experimental pharmacology & physiology (01.10.2022)
Published in Clinical and experimental pharmacology & physiology (01.10.2022)
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Journal Article
Design, Synthesis and Anticonvulsant Activity of Cinnamoyl Derivatives of 3,4,6,7,8,9-hexahydrodibenzo[ b,d ]furan-1-(2H)-one Oxime
Mokrov, Grigory V, Biryukova, Valentina E, Vorobieva, Tatiana Y, Pantileev, Andry S, Grigorkevich, Oksana S, Zhmurenko, Ludmila A, Rebeko, Alexey G, Bayburtskiy, Felix S, Litvinova, Svetlana A, Voronina, Tatiana A, Gudasheva, Tatiana A, Seredenin, Sergei B
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (2024)
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (2024)
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Role of the interfaces and the charge of a molecule in the non-equilibrium crystallization of dipeptide nanomaterials onto solid substrates
Loskutov, Alexander I, Lokshin, Boris V, Gudasheva, Tatiana A, Oshurko, Vadim B, Solis Pinargote, Nestor, Sazonova, Nellya M, Romanov, Vadim A
Published in CrystEngComm (2018)
Published in CrystEngComm (2018)
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Neuroprotective effect of novel cognitive enhancer noopept on AD-related cellular model involves the attenuation of apoptosis and tau hyperphosphorylation
Ostrovskaya, Rita U, Vakhitova, Yulia V, Kuzmina, Uliyana Sh, Salimgareeva, Milyausha Kh, Zainullina, Liana F, Gudasheva, Tatiana A, Vakhitov, Vener A, Seredenin, Sergey B
Published in Journal of biomedical science (06.08.2014)
Published in Journal of biomedical science (06.08.2014)
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Journal Article
GVS‐111 prevents oxidative damage and apoptosis in normal and Down's syndrome human cortical neurons
Pelsman, Alejandra, Hoyo‐Vadillo, Carlos, Gudasheva, Tatiana A., Seredenin, Sergei B., Ostrovskaya, Rita U., Busciglio, Jorge
Published in International journal of developmental neuroscience (01.05.2003)
Published in International journal of developmental neuroscience (01.05.2003)
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Journal Article
Design of N-Acylprolyltyrosine “Tripeptoid” Analogues of Neurotensin as Potential Atypical Antipsychotic Agents
Gudasheva, Tatiana A, Voronina, Tatiana A, Ostrovskaya, Rita U, Zaitseva, Natalya I, Bondarenko, Nina A, Briling, Vera K, Asmakova, Ludmila S, Rozantsev, Grigory G, Seredenin, Sergei B
Published in Journal of medicinal chemistry (29.01.1998)
Published in Journal of medicinal chemistry (29.01.1998)
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Preclinical and Clinical Pharmacokinetics of a Novel Dipeptide Anxiolytic GB-115
Bochkov, Pavel O, Kolik, Larisa G, Zherdev, Vladimir P, Kolyvanov, Gennadiy B, Litvin, Alexander A, Raskin, Sergei Yu, Shevchenko, Roman V, Grybakina, Oxana G, Gudasheva, Tatiana A, Seredenin, Sergei B
Published in Proceedings for Annual Meeting of The Japanese Pharmacological Society (2018)
Published in Proceedings for Annual Meeting of The Japanese Pharmacological Society (2018)
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Journal Article
The study of the spectrum of pharmacological activity of the new original NT-3 mimetic dipeptide GTS-302
Nikiforov, Dmitrii M., Povarnina, Polina Y., Gudasheva, Tatiana A., Nadorova, Anna V., Kolik, Larisa G., Valdman, Elena A., Vakhitova, Julia V., Seredenin, Sergey B.
Published in Medical academic journal (25.08.2023)
Published in Medical academic journal (25.08.2023)
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