Riluzole Series. Synthesis and in Vivo “Antiglutamate” Activity of 6-Substituted-2-benzothiazolamines and 3-Substituted-2-imino-benzothiazolines
Jimonet, Patrick, Audiau, François, Barreau, Michel, Blanchard, Jean-Charles, Boireau, Alain, Bour, Yvette, Coléno, Marie-Annick, Doble, Adam, Doerflinger, Gilles, Do Huu, Claudine, Donat, Marie-Hélène, Duchesne, Jean Marie, Ganil, Pierre, Guérémy, Claude, Honoré, Eliane, Just, Bernard, Kerphirique, Roselyne, Gontier, Sylvie, Hubert, Philippe, Laduron, Pierre M, Le Blevec, Joseph, Meunier, Mireille, Miquet, Jean-Marie, Nemecek, Conception, Pasquet, Martine, Piot, Odile, Pratt, Jeremy, Rataud, Jean, Reibaud, Michel, Stutzmann, Jean-Marie, Mignani, Serge
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Published in Journal of medicinal chemistry (29.07.1999)
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Electrophysiological and pharmacological characterization of peripheral benzodiazepine receptors in a guinea pig heart preparation
Mestre, M, Carriot, T, Belin, C, Uzan, A, Renault, C, Dubroeucq, M C, Guérémy, C, Le Fur, G
Published in Life sciences (1973) (27.08.1984)
Published in Life sciences (1973) (27.08.1984)
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Electrophysiological and pharmacological evidence that peripheral type benzodiazepine receptors are coupled to calcium channels in the heart
Mestre, M, Carriot, T, Belin, C, Uzan, A, Renault, C, Dubroeucq, M C, Guérémy, C, Doble, A, Le Fur, G
Published in Life sciences (1973) (01.01.1985)
Published in Life sciences (1973) (01.01.1985)
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Labelling of peripheral-type benzodiazepine binding sites in human brain with [3H]PK 11195: anatomical and subcellular distribution
Doble, A, Malgouris, C, Daniel, M, Daniel, N, Imbault, F, Basbaum, A, Uzan, A, Guérémy, C, Le Fur, G
Published in Brain research bulletin (01.01.1987)
Published in Brain research bulletin (01.01.1987)
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Peripheral benzodiazepine binding sites: effect of PK 11195, 1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)-3-isoquinolinecarboxamide. I. In vitro studies
Le Fur, G, Perrier, M L, Vaucher, N, Imbault, F, Flamier, A, Benavides, J, Uzan, A, Renault, C, Dubroeucq, M C, Guérémy, C
Published in Life sciences (1973) (18.04.1983)
Published in Life sciences (1973) (18.04.1983)
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Peripheral benzodiazepine binding sites: effect of PK 11195, 1-(2-chlorophenyl)-N-methyl-(1-methylpropyl)-3 isoquinolinecarboxamide. II. In vivo studies
Le Fur, G, Guilloux, F, Rufat, P, Benavides, J, Uzan, A, Renault, C, Dubroeucq, M C, Guérémy, C
Published in Life sciences (1973) (18.04.1983)
Published in Life sciences (1973) (18.04.1983)
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New indole derivatives as potent and selective serotonin uptake inhibitors
Malleron, Jean Luc, Gueremy, Claude, Mignani, Serge, Peyronel, Jean Francois, Truchon, Alain, Blanchard, Jean Charles, Doble, Adam, Laduron, Pierre, Piot, Odile
Published in Journal of medicinal chemistry (30.04.1993)
Published in Journal of medicinal chemistry (30.04.1993)
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Quantitative autoradiography of [3H]indalpine binding sites in the rat brain: II. Regional distribution
Savaki, H, Malgouris, C, Bénavidès, J, Laplace, C, Uzan, A, Guérémy, C, Le Fur, G
Published in Journal of neurochemistry (01.08.1985)
Published in Journal of neurochemistry (01.08.1985)
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Quantitative autoradiography of [3H]indalpine binding sites in the rat brain: I. Pharmacological characterization
Bénavidès, J, Savaki, H E, Malgouris, C, Laplace, C, Margelidon, C, Daniel, M, Courteix, J, Uzan, A, Guérémy, C, Le Fur, G
Published in Journal of neurochemistry (01.08.1985)
Published in Journal of neurochemistry (01.08.1985)
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Multiple benzodiazepine receptors: evidence of dissociation between anticonflict and anticonvulsant properties by PK 8165 and PK 9084 (two quinoline derivatives)
Le Fur, G, Mizoule, J, Burgevin, M C, Ferris, O, Heaulme, M, Gauthier, A, Guérémy, C, Uzan, A
Published in Life sciences (1973) (30.03.1981)
Published in Life sciences (1973) (30.03.1981)
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PK 11195, an antagonist of peripheral type benzodiazepine receptors, modulates Bay K8644 sensitive but not beta- or H2-receptor sensitive voltage operated calcium channels in the guinea pig heart
Mestre, M, Carriot, T, Néliat, G, Uzan, A, Renault, C, Dubroeucq, M C, Guérémy, C, Doble, A, Le Fur, G
Published in Life sciences (1973) (28.07.1986)
Published in Life sciences (1973) (28.07.1986)
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Autoradiographic localization of peripheral benzodiazepine binding sites in the cat brain with [3H]PK 11195
Bénavidès, J, Savaki, H E, Malgouris, C, Laplace, C, Daniel, M, Begassat, F, Desban, M, Uzan, A, Dubroeucq, M C, Renault, C
Published in Brain research bulletin (01.07.1984)
Published in Brain research bulletin (01.07.1984)
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Labelling of "peripheral-type" benzodiazepine binding sites in the rat brain by using [3H]PK 11195, an isoquinoline carboxamide derivative: kinetic studies and autoradiographic localization
Benavides, J, Quarteronet, D, Imbault, F, Malgouris, C, Uzan, A, Renault, C, Dubroeucq, M C, Gueremy, C, Le Fur, G
Published in Journal of neurochemistry (01.12.1983)
Published in Journal of neurochemistry (01.12.1983)
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Pharmacological characterization of RP 62203, a novel 5‐hydroxytryptamine 5‐HT2 receptor antagonist
Doble, A., Girdlestone, D., Piot, O., Allam, D., Betschart, J., Boireau, A., Dupuy, A., Guérémy, C., Ménager, J., Zundel, J.L., Blanchard, J.C.
Published in British journal of pharmacology (01.01.1992)
Published in British journal of pharmacology (01.01.1992)
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Stereospecificity of the in vitro and in vivo blockade of beta-receptors by FM 24, a slowly reversible ligand
Le Fur, G, Canton, T, Malgouris, C, Paillard, J J, Hardy, J C, Guérémy, C, Uzan, A
Published in Life sciences (1973) (14.12.1981)
Published in Life sciences (1973) (14.12.1981)
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Photoaffinity labeling of peripheral-type benzodiazepine-binding sites
DOBLE, A, FERRIS, O, BURGEVIN, M. C, MENAGER, J, UZAN, A, DUBRŒUCQ, M. C, RENAULT, C, GUEREMY, C, LE FUR, G
Published in Molecular pharmacology (01.01.1987)
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Published in Molecular pharmacology (01.01.1987)
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2-Amino-6-trifluoromethoxy benzothiazole, a possible antagonist of excitatory amino acid neurotransmission--II. Biochemical properties
Benavides, J, Camelin, J C, Mitrani, N, Flamand, F, Uzan, A, Legrand, J J, Gueremy, C, Le Fur, G
Published in Neuropharmacology (01.11.1985)
Published in Neuropharmacology (01.11.1985)
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Opposite effects of two ligands for peripheral type benzodiazepine binding sites, PK 11195 and RO5-4864, in a conflict situation in the rat
Mizoule, J, Gauthier, A, Uzan, A, Renault, C, Dubroeucq, M C, Guérémy, C, Le Fur, G
Published in Life sciences (1973) (18.03.1985)
Published in Life sciences (1973) (18.03.1985)
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