Oral administration of GW788388, an inhibitor of TGF-β type I and II receptor kinases, decreases renal fibrosis
Petersen, M., Thorikay, M., Deckers, M., van Dinther, M., Grygielko, E.T., Gellibert, F., de Gouville, A.C., Huet, S., ten Dijke, P., Laping, N.J.
Published in Kidney international (01.03.2008)
Published in Kidney international (01.03.2008)
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Discovery of 4-{4-[3-(Pyridin-2-yl)-1H-pyrazol-4-yl]pyridin-2-yl}-N-(tetrahydro-2H- pyran-4-yl)benzamide (GW788388): A Potent, Selective, and Orally Active Transforming Growth Factor-β Type I Receptor Inhibitor
Gellibert, Françoise, de Gouville, Anne-Charlotte, Woolven, James, Mathews, Neil, Nguyen, Van-Loc, Bertho-Ruault, Cécile, Patikis, Angela, Grygielko, Eugene T, Laping, Nicholas J, Huet, Stéphane
Published in Journal of medicinal chemistry (06.04.2006)
Published in Journal of medicinal chemistry (06.04.2006)
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Osmolality: a physiological long-term regulator of lumbar sympathetic nerve activity and arterial pressure
Scrogin, Karie E, Grygielko, Eugene T, Brooks, Virginia L
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.06.1999)
Published in American journal of physiology. Regulatory, integrative and comparative physiology (01.06.1999)
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Role of caspases in human renal proximal tubular epithelial cell apoptosis
Wong, Victoria Y, Keller, Paul M, Nuttall, Mark E, Kikly, Kristine, DeWolf, Walter E, Lee, Dennis, Ali, Shujath M, Nadeau, Daniel P, Grygielko, Eugene T, Laping, Nicholas J, Brooks, David P
Published in European journal of pharmacology (21.12.2001)
Published in European journal of pharmacology (21.12.2001)
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Oral administration of GW788388, an inhibitor of TGF-[beta] type I and II receptor kinases, decreases renal fibrosis
Petersen, M, Thorikay, M, Deckers, M, Van Dinther, M, Grygielko, E T, Gellibert, F, De Gouville, A C, Huet, S, Ten Dijke, P, Laping, N J
Published in Kidney international (01.03.2008)
Published in Kidney international (01.03.2008)
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Inhibition of gene markers of fibrosis with a novel inhibitor of transforming growth factor-beta type I receptor kinase in puromycin-induced nephritis
Grygielko, Eugene T, Martin, William M, Tweed, Christopher, Thornton, Peter, Harling, John, Brooks, David P, Laping, Nicholas J
Published in The Journal of pharmacology and experimental therapeutics (01.06.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.06.2005)
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The Angiotensin Type 1 Receptor Antagonist, Eprosartan, Attenuates the Progression of Renal Disease in Spontaneously Hypertensive Stroke-Prone Rats with Accelerated Hypertension
Abrahamsen, Christian T, Barone, Frank C, Campbell, Jr, Wallace G, Nelson, Allen H, Contino, Lisa C, Pullen, Mark A, Grygielko, Eugene T, Edwards, Richard M, Laping, Nicholas J, Brooks, David P
Published in The Journal of pharmacology and experimental therapeutics (01.04.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2002)
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Effects of Angiotensins II and IV on Blood Pressure, Renal Function, and PAI-1 Expression in the Heart and Kidney of the Rat
Abrahamsen, Christian T., Pullen, Mark A., Schnackenberg, Christine G., Grygielko, Eugene T., Edwards, Richard M., Laping, Nicholas J., Brooks, David P.
Published in Pharmacology (01.09.2002)
Published in Pharmacology (01.09.2002)
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