Discovery and structure–activity relationships of novel sulfonamides as potent PTP1B inhibitors
Holmes, Christopher P., Li, Xianfeng, Pan, Yijun, Xu, Caiding, Bhandari, Ashok, Moody, Claire M., Miguel, Joy A., Ferla, Steven W., De Francisco, M. Nuria, Frederick, Brian T., Zhou, Siqun, Macher, Natalie, Jang, Larry, Irvine, Jennifer D., Grove, J. Russell
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
Published in Bioorganic & medicinal chemistry letters (01.10.2005)
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Designing better coumarin-based fluorogenic substrates for PTP1B
Holmes, Christopher P., Macher, Natalie, Grove, J. Russell, Jang, Larry, Irvine, Jennifer D.
Published in Bioorganic & medicinal chemistry (01.06.2008)
Published in Bioorganic & medicinal chemistry (01.06.2008)
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Journal Article
TNFα-Mediated Inhibition and Reversal of Adipocyte Differentiation Is Accompanied by Suppressed Expression of PPARγ without Effects on Pref-1 Expression
Xing, Hong, Northrop, Jeffrey P., Grove, J. Russell, Kilpatrick, Katherine E., Su, Jui-Lan, Ringold, Gordon M.
Published in Endocrinology (Philadelphia) (01.07.1997)
Published in Endocrinology (Philadelphia) (01.07.1997)
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Journal Article
PTP1B inhibitors: Synthesis and evaluation of difluoro-methylenephosphonate bioisosteres on a sulfonamide scaffold
Holmes, Christopher P., Li, Xianfeng, Pan, Yijun, Xu, Caiding, Bhandari, Ashok, Moody, Claire M., Miguel, Joy A., Ferla, Steven W., De Francisco, M. Nuria, Frederick, Brian T., Zhou, Siqun, Macher, Natalie, Jang, Larry, Irvine, Jennifer D., Grove, J. Russell
Published in Bioorganic & medicinal chemistry (15.04.2008)
Published in Bioorganic & medicinal chemistry (15.04.2008)
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Journal Article
Multiple independent inputs are required for activation of the p70 S6 kinase
Weng, Qing-Ping, Andrabi, Khurshid, Kozlowski, Mark T., Grove, J. Russell, Avruch, Joseph
Published in Molecular and Cellular Biology (01.05.1995)
Published in Molecular and Cellular Biology (01.05.1995)
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A new and direct approach to functionalized biaryl α-ketophosphonic acids via aqueous Suzuki coupling on solid support
Li, Xianfeng, Szardenings, Anna Katrin, Holmes, Christopher P., Wang, Liang, Bhandari, Ashok, Shi, Lihong, Navre, Marc, Jang, Larry, Grove, J. Russell
Published in Tetrahedron letters (02.01.2006)
Published in Tetrahedron letters (02.01.2006)
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Potent Inhibitory Ligands of the GRB2 SH2 Domain from Recombinant Peptide Libraries
Hart, Charles P., Martin, Jennifer E., Reed, Margaret A., Keval, Aftab A., Pustelnik, Matthew J., Northrop, Jeffrey P., Patel, Dinesh V., Grove, J.Russell
Published in Cellular signalling (01.06.1999)
Published in Cellular signalling (01.06.1999)
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Membrane localization of the pertussis toxin-sensitive G-protein subunits alpha i-2 and alpha i-3 and expression of a metallothionein-alpha i-2 fusion gene in LLC-PK1 cells
Ercolani, L, Stow, J L, Boyle, J F, Holtzman, E J, Lin, H, Grove, J R, Ausiello, D A
Published in Proceedings of the National Academy of Sciences - PNAS (01.06.1990)
Published in Proceedings of the National Academy of Sciences - PNAS (01.06.1990)
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Journal Article
TNFα-Mediated Inhibition and Reversal of Adipocyte Differentiation Is Accompanied by Suppressed Expression of PPARγ without Effects on Pref-1 Expression1
Xing, Hong, Northrop, Jeffrey P, Grove, J. Russell, Kilpatrick, Katherine E, Su, Jui-Lan, Ringold, Gordon M
Published in Endocrinology (Philadelphia) (01.07.1997)
Published in Endocrinology (Philadelphia) (01.07.1997)
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Journal Article
Correction: Membrane Localization of the Pertussis Toxin-Sensitive G- Protein Subunits αi-2and αi-3and Expression of a Metallothionein-αi-2Fusion Gene in LLC-PK1Cells
Ercolani, Louis, Stow, Jennifer L., Boyle, Jane F., Holtzman, Eliezer J., Lin, Herbert, Grove, J. Russell, Ausiello, Dennis A.
Published in Proceedings of the National Academy of Sciences - PNAS (01.09.1990)
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Published in Proceedings of the National Academy of Sciences - PNAS (01.09.1990)
Journal Article
Membrane Localization of the Pertussis Toxin-Sensitive G-Protein Subunits αi-2and αi-3and Expression of a Metallothionein- αi-2Fusion Gene in LLC-PK1Cells
Ercolani, Louis, Stow, Jennifer L., Boyle, Jane F., Holtzman, Eliezer J., Lin, Herbert, Grove, J. Russell, Ausiello, Dennis A.
Published in Proceedings of the National Academy of Sciences - PNAS (01.06.1990)
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Published in Proceedings of the National Academy of Sciences - PNAS (01.06.1990)
Journal Article
Isolation of glucocorticoid-unresponsive rat hepatoma cells by fluorescence-activated cell sorting
Grove, J.Russell, Dieckmann, Barbara S., Schroer, Trina A., Ringold, Gordon M.
Published in Cell (01.08.1980)
Published in Cell (01.08.1980)
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Journal Article
Cloning and Expression of Two Human p70 S6 Kinase Polypeptides Differing Only at Their Amino Termini
Grove, J. Russell, Banerjee, Papia, Balasubramanyam, Ashok, Coffer, Paul J., Price, Daniel J., Avruch, Joseph, Woodgett, James R.
Published in Molecular and cellular biology (01.11.1991)
Published in Molecular and cellular biology (01.11.1991)
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