A Novel Bioactivation Pathway for 2-[2-(2,6-Dichlorophenyl)aminophenyl]ethanoic Acid (Diclofenac) Initiated by Cytochrome P450-Mediated Oxidative Decarboxylation
GRILLO, Mark P, JI MA, TEFFERA, Yohannes, WALDON, Daniel J
Published in Drug metabolism and disposition (01.09.2008)
Published in Drug metabolism and disposition (01.09.2008)
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Journal Article
In vitro and in vivo pharmacokinetic characterization of mavacamten, a first-in-class small molecule allosteric modulator of beta cardiac myosin
Grillo, Mark P., Erve, John C. L., Dick, Ryan, Driscoll, James P., Haste, Nicole, Markova, Svetlana, Brun, Priscilla, Carlson, Timothy J., Evanchik, Marc
Published in Xenobiotica (03.06.2019)
Published in Xenobiotica (03.06.2019)
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Journal Article
Acyl-CoA thioesters as chemically-reactive intermediates of carboxylic acid-containing drugs
Grillo, Mark P., Li, Chunze, Benet, Leslie Z.
Published in Medicinal chemistry research (01.09.2023)
Published in Medicinal chemistry research (01.09.2023)
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Journal Article
STUDIES ON THE CHEMICAL REACTIVITY OF DICLOFENAC ACYL GLUCURONIDE WITH GLUTATHIONE: IDENTIFICATION OF DICLOFENAC-S-ACYL-GLUTATHIONE IN RAT BILE
GRILLO, Mark P, KNUTSON, Charles G, SANDERS, Phillip E, WALDON, Daniel J, FENGMEI HUA, WARE, Joseph A
Published in Drug metabolism and disposition (01.11.2003)
Published in Drug metabolism and disposition (01.11.2003)
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Journal Article
Preclinical in vitro and in vivo pharmacokinetic properties of danicamtiv, a new targeted myosin activator for the treatment of dilated cardiomyopathy
Grillo, Mark P., Markova, Svetlana, Evanchik, Marc, Trellu, Marc, Moliner, Patricia, Brun, Priscilla, Perreard-Dumaine, Anne, Vicat, Pascale, Yang, Chun, Driscoll, James P., Carlson, Tim J.
Published in Xenobiotica (01.02.2021)
Published in Xenobiotica (01.02.2021)
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Journal Article
Constituents in Kava Extracts Potentially Involved in Hepatotoxicity: A Review
Olsen, Line R, Grillo, Mark P, Skonberg, Christian
Published in Chemical research in toxicology (18.07.2011)
Published in Chemical research in toxicology (18.07.2011)
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Journal Article
Metabolic activation of carboxylic acids
Skonberg, Christian, Olsen, Jørgen, Madsen, Kim Grimstrup, Hansen, Steen Honoré, Grillo, Mark P
Published in Expert opinion on drug metabolism & toxicology (01.04.2008)
Published in Expert opinion on drug metabolism & toxicology (01.04.2008)
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Journal Article
Enantioselective Covalent Binding of 2-Phenylpropionic Acid to Protein in Vitro in Rat Hepatocytes
Li, Chunze, Benet, Leslie Z, Grillo, Mark P
Published in Chemical research in toxicology (01.11.2002)
Published in Chemical research in toxicology (01.11.2002)
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Journal Article