Evaluation of Substituted N-Phenylpiperazine Analogs as D3 vs. D2 Dopamine Receptor Subtype Selective Ligands
Lee, Boeun, Taylor, Michelle, Griffin, Suzy A., McInnis, Tamara, Sumien, Nathalie, Mach, Robert H., Luedtke, Robert R.
Published in Molecules (Basel, Switzerland) (26.05.2021)
Published in Molecules (Basel, Switzerland) (26.05.2021)
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N-(3-Fluoro-4-(4-(2-methoxy or 2,3-dichlorophenyl)piperazine-1-yl)butyl)arylcarboxamides as Selective Dopamine D3 Receptor Ligands: Critical Role of the Carboxamide Linker for D3 Receptor Selectivity
Banala, Ashwini K, Levy, Benjamin A, Khatri, Sameer S, Furman, Cheryse A, Roof, Rebecca A, Mishra, Yogesh, Griffin, Suzy A, Sibley, David R, Luedtke, Robert R, Newman, Amy Hauck
Published in Journal of medicinal chemistry (26.05.2011)
Published in Journal of medicinal chemistry (26.05.2011)
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Evaluation of the D3 dopamine receptor selective antagonist PG01037 on l-dopa-dependent abnormal involuntary movements in rats
Kumar, Rakesh, Riddle, Lindsay, Griffin, Suzy A., Grundt, Peter, Newman, Amy Hauck, Luedtke, Robert R.
Published in Neuropharmacology (01.05.2009)
Published in Neuropharmacology (01.05.2009)
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Design, synthesis, and evaluation of N-(4-(4-phenyl piperazin-1-yl)butyl)-4-(thiophen-3-yl)benzamides as selective dopamine D3 receptor ligands
Chen, Peng-Jen, Taylor, Michelle, Griffin, Suzy A., Amani, Armaghan, Hayatshahi, Hamed, Korzekwa, Kenneth, Ye, Min, Mach, Robert H., Liu, Jin, Luedtke, Robert R., Gordon, John C., Blass, Benjamin E.
Published in Bioorganic & medicinal chemistry letters (15.09.2019)
Published in Bioorganic & medicinal chemistry letters (15.09.2019)
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Design, synthesis, and evaluation of N-(4-(4-phenyl piperazin-1-yl) butyl)-4-(thiophen-3-yl) benzamides as selective dopamine D-3 receptor ligands
Chen, Peng-Jen, Taylor, Michelle, Griffin, Suzy A., Amani, Armaghan, Hayatshahi, Hamed, Korzekwa, Kenneth, Ye, Min, Mach, Robert H., Liu, Jin, Luedtke, Robert R., Gordon, John C., Blass, Benjamin E.
Published in Bioorganic & medicinal chemistry letters (15.09.2019)
Published in Bioorganic & medicinal chemistry letters (15.09.2019)
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Analogues of Arylamide Phenylpiperazine Ligands To Investigate the Factors Influencing D3 Dopamine Receptor Bitropic Binding and Receptor Subtype Selectivity
Hayatshahi, Hamed S, Xu, Kuiying, Griffin, Suzy A, Taylor, Michelle, Mach, Robert H, Liu, Jin, Luedtke, Robert R
Published in ACS chemical neuroscience (19.12.2018)
Published in ACS chemical neuroscience (19.12.2018)
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Design, synthesis, and evaluation of functionalized 5-(4-arylpiperazin-1-yl)-N-quinolinyl-pentanamides as selective dopamine D3 receptor ligands
Blass, Benjamin E., Chen, Peng-Jen, Taylor, Michelle, Griffin, Suzy A., Gordon, John C., Luedtke, Robert R.
Published in Medicinal chemistry research (01.05.2022)
Published in Medicinal chemistry research (01.05.2022)
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Synthesis and evaluation of cyclic diamino benzamide based D3 receptor ligands
Blass, Benjamin E., Chen, Peng-Jen, Taylor, Michelle, Griffin, Suzy A., Gordon, John C., Luedtke, Robert R.
Published in Medicinal chemistry research (01.03.2022)
Published in Medicinal chemistry research (01.03.2022)
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Design, synthesis, and evaluation of functionalized 5-(4-arylpiperazin-1-yl)-N-arylpentanamides as selective dopamine D3 receptor ligands
Blass, Benjamin E., Chen, Peng-Jen, Taylor, Michelle, Griffin, Suzy A., Gordon, John C., Luedtke, Robert R.
Published in Medicinal chemistry research (2022)
Published in Medicinal chemistry research (2022)
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The tetrahydroisoquinoline derivative SB269,652 is an allosteric antagonist at dopamine D3 and D2 receptors
Silvano, Elena, Millan, Mark J, Mannoury la Cour, Clotilde, Han, Yang, Duan, Lihua, Griffin, Suzy A, Luedtke, Robert R, Aloisi, Gabriella, Rossi, Mario, Zazzeroni, Francesca, Javitch, Jonathan A, Maggio, Roberto
Published in Molecular pharmacology (01.11.2010)
Published in Molecular pharmacology (01.11.2010)
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Evaluation of D2 and D3 dopamine receptor selective compounds on l-dopa-dependent abnormal involuntary movements in rats
Kumar, Rakesh, Riddle, Lindsay R., Griffin, Suzy A., Chu, Wenhua, Vangveravong, Suwanna, Neisewander, Janet, Mach, Robert H., Luedtke, Robert R.
Published in Neuropharmacology (01.05.2009)
Published in Neuropharmacology (01.05.2009)
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Immunoblot and immunohistochemical comparison of murine monoclonal antibodies specific for the rat D1a and D1b dopamine receptor subtypes
Luedtke, Robert R, Griffin, Suzy A, Conroy, Susan S, Jin, Xialan, Pinto, Aline, Sesack, Susan R
Published in Journal of neuroimmunology (15.11.1999)
Published in Journal of neuroimmunology (15.11.1999)
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Evaluation of the D3 dopamine receptor selective agonist/partial agonist PG01042 on l-dopa dependent animal involuntary movements in rats
Riddle, Lindsay R., Kumar, Rakesh, Griffin, Suzy A., Grundt, Peter, Newman, Amy Hauck, Luedtke, Robert R.
Published in Neuropharmacology (01.02.2011)
Published in Neuropharmacology (01.02.2011)
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Dopamine D3 receptor selective ligands with varying intrinsic efficacies at adenylyl cyclase inhibition and mitogenic signaling pathways
Taylor, Michelle, Grundt, Peter, Griffin, Suzy A., Newman, Amy Hauck, Luedtke, Robert R.
Published in Synapse (New York, N.Y.) (01.03.2010)
Published in Synapse (New York, N.Y.) (01.03.2010)
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Comparison of the Binding and Functional Properties of Two Structurally Different D2 Dopamine Receptor Subtype Selective Compounds
Luedtke, Robert R, Mishra, Yogesh, Wang, Qi, Griffin, Suzy A, Bell-Horner, Cathy, Taylor, Michelle, Vangveravong, Suwanna, Dillon, Glenn H, Huang, Ren-Qi, Reichert, David E, Mach, Robert H
Published in ACS chemical neuroscience (19.12.2012)
Published in ACS chemical neuroscience (19.12.2012)
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The Effect of SV 293, a D2 Dopamine Receptor-Selective Antagonist, on D2 Receptor-Mediated GIRK Channel Activation and Adenylyl Cyclase Inhibition
Huang, Renqi, Griffin, Suzy A., Taylor, Michelle, Vangveravong, Suwanna, Mach, Robert H., Dillon, Glenn H., Luedtke, Robert R.
Published in Pharmacology (01.01.2013)
Published in Pharmacology (01.01.2013)
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The Tetrahydroisoquinoline Derivative SB269,652 Is an Allosteric Antagonist at Dopamine D 3 and D 2 Receptors
Silvano, Elena, Millan, Mark J., la Cour, Clotilde Mannoury, Han, Yang, Duan, Lihua, Griffin, Suzy A., Luedtke, Robert R., Aloisi, Gabriella, Rossi, Mario, Zazzeroni, Francesca, Javitch, Jonathan A., Maggio, Roberto
Published in Molecular pharmacology (01.11.2010)
Published in Molecular pharmacology (01.11.2010)
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Journal Article
N-(3-Fluoro-4-(4-(2-methoxy or 2,3-dichlorophenyl) piperazine-1-yl)-butyl)-aryl carboxamides as Selective Dopamine D3 Receptor Ligands: Critical Role of the Carboxamide Linker for D3 Receptor Selectivity
Banala, Ashwini K., Levy, Benjamin A., Khatri, Sameer S., Furman, Cheryse A., Roof, Rebecca A., Mishra, Yogesh, Griffin, Suzy A., Sibley, David R., Luedtke, Robert R., Newman, Amy Hauck
Published in Journal of medicinal chemistry (02.05.2011)
Published in Journal of medicinal chemistry (02.05.2011)
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Journal Article
The Tetrahydroisoquinoline Derivative SB269,652 Is an Allosteric Antagonist at Dopamine D3 and D2 ReceptorsS
Silvano, Elena, Millan, Mark J., la Cour, Clotilde Mannoury, Han, Yang, Duan, Lihua, Griffin, Suzy A., Luedtke, Robert R., Aloisi, Gabriella, Rossi, Mario, Zazzeroni, Francesca, Javitch, Jonathan A., Maggio, Roberto
Published in Molecular pharmacology (01.11.2010)
Published in Molecular pharmacology (01.11.2010)
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Journal Article
Molecular characterization of a mammalian smooth muscle myosin light chain kinase
GALLAGHER, P. J, HERRING, B. P, GRIFFIN, S. A, STULL, J. T
Published in The Journal of biological chemistry (15.12.1991)
Published in The Journal of biological chemistry (15.12.1991)
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