Synthesis and Structure−Activity Relationship of Acrylamides as KCNQ2 Potassium Channel Openers
Wu, Yong-Jin, He, Huan, Sun, Li-Qiang, L'Heureux, Alexandre, Chen, Jie, Dextraze, Pierre, Starrett, John E, Boissard, Christopher G, Gribkoff, Valentin K, Natale, Joanne, Dworetzky, Steven I
Published in Journal of medicinal chemistry (20.05.2004)
Published in Journal of medicinal chemistry (20.05.2004)
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Targeted disruption of the mouse Mel(1b) melatonin receptor
Jin, Xiaowei, von Gall, Charlotte, Pieschl, Rick L, Gribkoff, Valentin K, Stehle, Jorg H, Reppert, Steven M, Weaver, David R
Published in Molecular and cellular biology (01.02.2003)
Published in Molecular and cellular biology (01.02.2003)
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Long-Lasting Functional Disabilities in Middle-Aged Rats with Small Cerebral Infarcts
Lindner, Mark D, Gribkoff, Valentin K, Donlan, Nicole A, Jones, Theresa A
Published in The Journal of neuroscience (26.11.2003)
Published in The Journal of neuroscience (26.11.2003)
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Synthesis and Structure−Activity Relationships of 3-Aryloxindoles: A New Class of Calcium-Dependent, Large Conductance Potassium (Maxi-K) Channel Openers with Neuroprotective Properties
Hewawasam, Piyasena, Erway, Matthew, Moon, Sandra L, Knipe, Jay, Weiner, Harvey, Boissard, Christopher G, Post-Munson, Debra J, Gao, Qi, Huang, Stella, Gribkoff, Valentin K, Meanwell, Nicholas A
Published in Journal of medicinal chemistry (28.03.2002)
Published in Journal of medicinal chemistry (28.03.2002)
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The synthesis and characterization of BMS-204352 (MaxiPost) and related 3-fluorooxindoles as openers of maxi-K potassium channels
HEWAWASAM, Piyasena, GRIBKOFF, Valentin K, PAJOR, Lorraine M, KNIPE, Jay, QI GAO, PERRONE, Robert, STARRETT, John E, PENDRI, Yadagiri, DWORETZKY, Steven I, MEANWELL, Nicholas A, MARTINEZ, Eduardo, BOISSARD, Christopher G, POST-MUNSON, Debra J, TROJNACKI, Joanne T, YELESWARAM, Krishnaswamy
Published in Bioorganic & medicinal chemistry letters (08.04.2002)
Published in Bioorganic & medicinal chemistry letters (08.04.2002)
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An Assessment of the Effects of Serotonin 6 (5-HT6) Receptor Antagonists in Rodent Models of Learning
Lindner, Mark D, Hodges, Jr, Donald B, Hogan, John B, Orie, Anitra F, Corsa, Jason A, Barten, Donna M, Polson, Craig, Robertson, Barbara J, Guss, Valerie L, Gillman, Kevin W, Starrett, Jr, John E, Gribkoff, Valentin K
Published in The Journal of pharmacology and experimental therapeutics (01.11.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.11.2003)
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4-Aryl-3-(hydroxyalkyl)quinolin-2-ones: Novel Maxi-K Channel Opening Relaxants of Corporal Smooth Muscle Targeted for Erectile Dysfunction
Hewawasam, Piyasena, Fan, Wenhong, Ding, Min, Flint, Kim, Cook, Deborah, Goggins, Gregory D, Myers, Robert A, Gribkoff, Valentin K, Boissard, Christopher G, Dworetzky, Steven I, Starrett, John E, Lodge, Nicholas J
Published in Journal of medicinal chemistry (03.07.2003)
Published in Journal of medicinal chemistry (03.07.2003)
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Voltage-gated cation channel modulators for the treatment of stroke
Gribkoff, Valentin K, Winquist, Raymond J
Published in Expert opinion on investigational drugs (01.05.2005)
Published in Expert opinion on investigational drugs (01.05.2005)
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Phenotypic Alteration of a Human BK ( hSlo ) Channel by hSloβ Subunit Coexpression: Changes in Blocker Sensitivity, Activation/Relaxation and Inactivation Kinetics, and Protein Kinase A Modulation
Dworetzky, Steven I., Boissard, Christopher G., Lum-Ragan, Janet T., McKay, M. Craig, Post-Munson, Debra J., Trojnacki, Joanne T., Chang, Chia-Ping, Gribkoff, Valentin K.
Published in The Journal of neuroscience (01.08.1996)
Published in The Journal of neuroscience (01.08.1996)
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(S)-N-[1-(3-Morpholin-4-ylphenyl)ethyl]-3phenylacrylamide: An orally bioavailable KCNQ2 opener with significant activity in a cortical spreading depression model of migraine
Wu, YJ, Boissard, CG, Greco, C, Gribkoff, VK, Harden, DG, He, H, L'Heureux, A, Kang, SH, Kinney, GG, Knox, RJ, Natale, J, Newton, AE, Lehtinen-Oboma, S, Sinz, MW, Sivarao, DV, Starrett, JE, Sun, LQ, Tertyshnikova, S, Thompson, MW, Weaver, D, Wong, HS, Zhang, L, Dworetzky, SL
Published in Journal of medicinal chemistry (17.07.2003)
Published in Journal of medicinal chemistry (17.07.2003)
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Formation of intermediate-conductance calcium-activated potassium channels by interaction of Slack and Slo subunits
Kaczmarek, Leonard K, Joiner, William J, Tang, Michael D, Wang, Lu-Yang, Dworetzky, Steven I, Boissard, Christopher G, Gan, Li, Gribkoff, Valentin K
Published in Nature neuroscience (01.10.1998)
Published in Nature neuroscience (01.10.1998)
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3-Thio-quinolinone maxi-K openers for the treatment of erectile dysfunction
BOY, Kenneth M, GUERNON, Jason M, STARRETT, John E, SIT, Sing-Yuen, XIE, Kai, HEWAWASAM, Piyasena, BOISSARD, Christopher G, DWORETZKY, Steven I, NATALE, Joanne, GRIBKOFF, Valentin K, LODGE, Nicholas
Published in Bioorganic & medicinal chemistry letters (18.10.2004)
Published in Bioorganic & medicinal chemistry letters (18.10.2004)
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4-Aryl-3-(mercapto)quinolin-2-ones: novel maxi-K channel opening relaxants of corporal smooth muscle
Hewawasam, Piyasena, Fan, Wenhong, Cook, Deborah A., Newberry, Kimberly S., Boissard, Christopher G., Gribkoff, Valentin K., Starrett, John, Lodge, Nicholas J.
Published in Bioorganic & medicinal chemistry letters (06.09.2004)
Published in Bioorganic & medicinal chemistry letters (06.09.2004)
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Journal Article
Effects of channel modulators on cloned large-conductance calcium-activated potassium channels
V K Gribkoff, J T Lum-Ragan, C G Boissard, D J Post-Munson, N A Meanwell, J E Starrett, Jr, E S Kozlowski, J L Romine, J T Trojnacki, M C Mckay, J Zhong, S I Dworetzky
Published in Molecular pharmacology (01.07.1996)
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Published in Molecular pharmacology (01.07.1996)
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