Synthetic Study toward Total Synthesis of (±)-Germine: Synthesis of (±)-4-Methylenegermine
Stork, Gilbert, Yamashita, Ayako, Hanson, Robert M, Phan, Ly, Phillips, Eifion, Dubé, Daniel, Bos, Pieter H, Clark, Andrew J, Gough, Maxwell, Greenlee, Mark L, Jiang, Yimin, Jones, Keith, Kitamura, Masato, Leonard, John, Liu, Tongzhu, Parsons, Philip J, Venkatesan, Aranapakam M
Published in Organic letters (06.10.2017)
Published in Organic letters (06.10.2017)
Get full text
Journal Article
Ibrexafungerp: An orally active β-1,3-glucan synthesis inhibitor
Apgar, James M., Wilkening, Robert R., Parker, Dann L., Meng, Dongfang, Wildonger, Kenneth J., Sperbeck, Donald, Greenlee, Mark L., Balkovec, James M., Flattery, Amy M., Abruzzo, George K., Galgoci, Andrew M., Giacobbe, Robert A., Gill, Charles J., Hsu, Ming-Jo, Liberator, Paul, Misura, Andrew S., Motyl, Mary, Nielsen Kahn, Jennifer, Powles, Maryann, Racine, Fred, Dragovic, Jasminka, Fan, Weiming, Kirwan, Robin, Lee, Shu, Liu, Hao, Mamai, Ahmed, Nelson, Kingsley, Peel, Michael
Published in Bioorganic & medicinal chemistry letters (15.01.2021)
Published in Bioorganic & medicinal chemistry letters (15.01.2021)
Get full text
Journal Article
MK-5204: An orally active β-1,3-glucan synthesis inhibitor
Apgar, James M., Wilkening, Robert R., Parker, Dann L., Meng, Dongfang, Wildonger, Kenneth J., Sperbeck, Donald, Greenlee, Mark L., Balkovec, James M., Flattery, Amy M., Abruzzo, George K., Galgoci, Andrew M., Giacobbe, Robert A., Gill, Charles J., Hsu, Ming-Jo, Liberator, Paul, Misura, Andrew S., Motyl, Mary, Kahn, Jennifer Nielsen, Powles, Maryann, Racine, Fred, Dragovic, Jasminka, Fan, Weiming, Kirwan, Robin, Lee, Shu, Liu, Hao, Mamai, Ahmed, Nelson, Kingsley, Peel, Michael
Published in Bioorganic & medicinal chemistry letters (01.09.2020)
Published in Bioorganic & medicinal chemistry letters (01.09.2020)
Get full text
Journal Article
Novel orally active inhibitors of β-1,3-glucan synthesis derived from enfumafungin
Apgar, James M., Wilkening, Robert R., Greenlee, Mark L., Balkovec, James M., Flattery, Amy M., Abruzzo, George K., Galgoci, Andrew M., Giacobbe, Robert A., Gill, Charles J., Hsu, Ming Jo, Liberator, Paul, Misura, Andrew S., Motyl, Mary, Nielsen Kahn, Jennifer, Powles, Maryann, Racine, Fred, Dragovic, Jasminka, Habulihaz, Bahanu, Fan, Weiming, Kirwan, Robin, Lee, Shu, Liu, Hao, Mamai, Ahmed, Nelson, Kingsley, Peel, Michael
Published in Bioorganic & medicinal chemistry letters (15.12.2015)
Published in Bioorganic & medicinal chemistry letters (15.12.2015)
Get full text
Journal Article
Triazolo-tetrahydrofluorenones as selective estrogen receptor beta agonists
Parker, Dann L., Meng, Dongfang, Ratcliffe, Ronald W., Wilkening, Robert R., Sperbeck, Donald M., Greenlee, Mark L., Colwell, Lawrence F., Lambert, Sherrie, Birzin, Elizabeth T., Frisch, Katalin, Rohrer, Susan P., Nilsson, Stefan, Thorsell, Ann-Gerd, Hammond, Milton L.
Published in Bioorganic & medicinal chemistry letters (01.09.2006)
Published in Bioorganic & medicinal chemistry letters (01.09.2006)
Get full text
Journal Article
A unique reversal of regioselectivity in the photoaddition of 2-fluorocyclohexenone to isobutylene
Greenlee, Mark L, Fritzen, Edward L, Swenton, John S
Published in Journal of organic chemistry (01.11.1978)
Published in Journal of organic chemistry (01.11.1978)
Get full text
Journal Article
Inhibition of IMP-1 metallo-β-lactamase and sensitization of IMP-1-producing bacteria by thioester derivatives
Hammond, Gail G., Huber, Joann L., Greenlee, Mark L., Laub, Joanne B., Young, Katherine, Silver, Lynn L., Balkovec, James M., Pryor, KellyAnn D., Wu, Joseph K., Leiting, Barbara, Pompliano, David L., Toney, Jeffrey H.
Published in FEMS microbiology letters (01.10.1999)
Published in FEMS microbiology letters (01.10.1999)
Get full text
Journal Article
Inhibition of IMP-1 metallo-β-lactamase and sensitization of IMP-1-producing bacteria by thioester derivatives
Hammond, Gail G., Huber, Joann L., Greenlee, Mark L., Laub, Joanne B., Young, Katherine, Silver, Lynn L., Balkovec, James M., Pryor, KellyAnn D., Wu, Joseph K., Leiting, Barbara, Pompliano, David L., Toney, Jeffrey H.
Published in FEMS microbiology letters (01.10.1999)
Published in FEMS microbiology letters (01.10.1999)
Get full text
Journal Article
Succinic acids as potent inhibitors of plasmid-borne IMP-1 metallo-beta-lactamase
Toney, J H, Hammond, G G, Fitzgerald, P M, Sharma, N, Balkovec, J M, Rouen, G P, Olson, S H, Hammond, M L, Greenlee, M L, Gao, Y D
Published in The Journal of biological chemistry (24.08.2001)
Published in The Journal of biological chemistry (24.08.2001)
Get full text
Journal Article
X-ray and theoretical analysis of the relationship between substituent steric effects and the structure of bicyclo[1.1.0]butane. The unexpected flexibility of the bicyclo[1.1.0]butane skeleton
Gassman, Paul G, Greenlee, Mark L, Dixon, David A, Richtsmeier, Steven, Gougoutas, J. Zanos
Published in Journal of the American Chemical Society (01.09.1983)
Published in Journal of the American Chemical Society (01.09.1983)
Get full text
Journal Article
Erratum to “Triazolo-tetrahydrofluorenones as selective estrogen receptor beta agonists” [Bioorg. Med. Chem. Lett. 16 (2006) 4652–4656]
Parker, Dann L., Meng, Dongfang, Ratcliffe, Ronald W., Wilkening, Robert R., Sperbeck, Donald M., Greenlee, Mark L., Colwell, Lawrence F., Lambert, Sherrie, Birzin, Elizabeth T., Frisch, Katalin, Rohrer, Susan P., Nilsson, Stefan, Thorsell, Ann-Gerd, Hammond, Milton L.
Published in Bioorganic & medicinal chemistry letters (15.10.2006)
Published in Bioorganic & medicinal chemistry letters (15.10.2006)
Get full text
Journal Article
Inhibition of IMP-1 metallo-β-lactamase and sensitization of IMP-1-producing bacteria by thioester derivatives
Hammond, Gail G., Huber, Joann L., Greenlee, Mark L., Laub, Joanne B., Young, Katherine, Silver, Lynn L., Balkovec, James M., Pryor, KellyAnn D., Wu, Joseph K., Leiting, Barbara, Pompliano, David L., Toney, Jeffrey H.
Published in FEMS microbiology letters (15.10.1999)
Published in FEMS microbiology letters (15.10.1999)
Get full text
Journal Article
Synthesis and SAR of thioester and thiol inhibitors of IMP-1 Metallo-β-Lactamase
Greenlee, Mark L., Laub, Joanne B., Balkovec, James M., Hammond, Milton L., Hammond, Gail G., Pompliano, David L., Epstein-Toney, Jeffrey H.
Published in Bioorganic & medicinal chemistry letters (06.09.1999)
Published in Bioorganic & medicinal chemistry letters (06.09.1999)
Get full text
Journal Article
Dicationic 2-fluorenonylcarbapenems: Potent anti-MRS agents with improved solubility and pharmacokinetic properties
Greenlee, Mark L., Laub, Joanne B., Rouen, Gregory P., DiNinno, Frank, Hammond, Milton L., Huber, Joann L., Sundelof, Jon G., Hammond, Gail G.
Published in Bioorganic & medicinal chemistry letters (15.11.1999)
Published in Bioorganic & medicinal chemistry letters (15.11.1999)
Get full text
Journal Article
Succinic Acids as Potent Inhibitors of Plasmid-borne IMP-1 Metallo-β-lactamase
Jeffrey H. Toney, Gail G. Hammond, Paula M. D. Fitzgerald, Nandini Sharma, James M. Balkovec, Gregory P. Rouen, Steven H. Olson, Milton L. Hammond, Mark L. Greenlee, Ying-Duo Gao
Published in The Journal of biological chemistry (24.08.2001)
Published in The Journal of biological chemistry (24.08.2001)
Get full text
Journal Article
ESTROGEN RECEPTOR MODULATORS
MENG, Dongfang, SPERBECK, Donald, M, WILDONGER, Kenneth, J, GREENLEE, Mark, L
Year of Publication 27.09.2017
Get full text
Year of Publication 27.09.2017
Patent