Search Results - "Grand-Maı̂tre, Chantal" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Tetrahydrofuran-Based Transient Receptor Potential Ankyrin 1 (TRPA1) Antagonists: Ligand-Based Discovery, Activity in a Rodent Asthma Model, and Mechanism-of-Action via Cryogenic Electron Microscopy

Tetrahydrofuran-Based Transient Receptor Potential Ankyrin 1 (TRPA1) Antagonists: Ligand-Based Discovery, Activity in a Rodent Asthma Model, and Mechanism-of-Action via Cryogenic Electron Microscopy

by Terrett, Jack A, Chen, Huifen, Shore, Daniel G, Villemure, Elisia, Larouche-Gauthier, Robin, Déry, Martin, Beaumier, Francis, Constantineau-Forget, Léa, Grand-Maître, Chantal, Lépissier, Luce, Ciblat, Stéphane, Sturino, Claudio, Chen, Yong, Hu, Baihua, Lu, Aijun, Wang, Yunli, Cridland, Andrew P, Ward, Stuart I, Hackos, David H, Reese, Rebecca M, Shields, Shannon D, Chen, Jun, Balestrini, Alessia, Riol-Blanco, Lorena, Lee, Wyne P, Liu, John, Suto, Eric, Wu, Xiumin, Zhang, Juan, Ly, Justin Q, La, Hank, Johnson, Kevin, Baumgardner, Matt, Chou, Kang-Jye, Rohou, Alexis, Rougé, Lionel, Safina, Brian S, Magnuson, Steven, Volgraf, Matthew
Published in Journal of medicinal chemistry (08.04.2021)

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Novel Inhibitor Binding Site Discovery on HIV‑1 Capsid N‑Terminal Domain by NMR and X‑ray Crystallography

Novel Inhibitor Binding Site Discovery on HIV‑1 Capsid N‑Terminal Domain by NMR and X‑ray Crystallography

by Goudreau, Nathalie, Lemke, Christopher T, Faucher, Anne-Marie, Grand-Maître, Chantal, Goulet, Sylvie, Lacoste, Jean-Eric, Rancourt, Jean, Malenfant, Eric, Mercier, Jean-François, Titolo, Steve, Mason, Stephen W
Published in ACS chemical biology (17.05.2013)

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Discovery of a 1,5-dihydrobenzo[b][1,4]diazepine-2,4-dione series of inhibitors of HIV-1 capsid assembly

Discovery of a 1,5-dihydrobenzo[b][1,4]diazepine-2,4-dione series of inhibitors of HIV-1 capsid assembly

by Fader, Lee D., Bethell, Richard, Bonneau, Pierre, Bös, Michael, Bousquet, Yves, Cordingley, Michael G., Coulombe, René, Deroy, Patrick, Faucher, Anne-Marie, Gagnon, Alexandre, Goudreau, Nathalie, Grand-Maître, Chantal, Guse, Ingrid, Hucke, Oliver, Kawai, Stephen H., Lacoste, Jean-Eric, Landry, Serge, Lemke, Christopher T., Malenfant, Eric, Mason, Stephen, Morin, Sébastien, O’Meara, Jeff, Simoneau, Bruno, Titolo, Steve, Yoakim, Christiane
Published in Bioorganic & medicinal chemistry letters (01.01.2011)

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Discovery of Small-Molecule Inhibitors of the ATPase Activity of Human Papillomavirus E1 Helicase

Discovery of Small-Molecule Inhibitors of the ATPase Activity of Human Papillomavirus E1 Helicase

by Faucher, Anne-Marie, White, Peter W, Brochu, Christian, Grand-Maître, Chantal, Rancourt, Jean, Fazal, Gulrez
Published in Journal of medicinal chemistry (01.01.2004)

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Monitoring Binding of HIV-1 Capsid Assembly Inhibitors Using 19F Ligand-and 15N Protein-Based NMR and X-ray Crystallography: Early Hit Validation of a Benzodiazepine Series

Monitoring Binding of HIV-1 Capsid Assembly Inhibitors Using 19F Ligand-and 15N Protein-Based NMR and X-ray Crystallography: Early Hit Validation of a Benzodiazepine Series

by Goudreau, Nathalie, Coulombe, René, Faucher, Anne-Marie, Grand-Maître, Chantal, Lacoste, Jean-Eric, Lemke, Christopher T., Malenfant, Eric, Bousquet, Yves, Fader, Lee, Simoneau, Bruno, Mercier, Jean-François, Titolo, Steve, Mason, Stephen W.
Published in ChemMedChem (01.03.2013)

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Discovery of TRPA1 Antagonist GDC-6599: Derisking Preclinical Toxicity and Aldehyde Oxidase Metabolism with a Potential First-in-Class Therapy for Respiratory Disease

Discovery of TRPA1 Antagonist GDC-6599: Derisking Preclinical Toxicity and Aldehyde Oxidase Metabolism with a Potential First-in-Class Therapy for Respiratory Disease

by Terrett, Jack A., Ly, Justin Q., Katavolos, Paula, Hasselgren, Catrin, Laing, Steven, Zhong, Fiona, Villemure, Elisia, Déry, Martin, Larouche-Gauthier, Robin, Chen, Huifen, Shore, Daniel G., Lee, Wyne P., Suto, Eric, Johnson, Kevin, Brooks, Marjory, Stablein, Alyssa, Beaumier, Francis, Constantineau-Forget, Léa, Grand-Maître, Chantal, Lépissier, Luce, Ciblat, Stéphane, Sturino, Claudio, Chen, Yong, Hu, Baihua, Elstrott, Justin, Gandham, Vineela, Joseph, Victory, Booler, Helen, Cain, Gary, Chou, Carolina, Fullerton, Aaron, Lepherd, Michelle, Stainton, Shannon, Torres, Elizabeth, Urban, Konnie, Yu, Lanlan, Zhong, Yu, Bao, Linda, Chou, Kang-Jye, Lin, Jessica, Zhang, Wei, La, Hank, Liu, Liling, Mulder, Teresa, Chen, Jun, Chernov-Rogan, Tania, Johnson, Adam R., Hackos, David H., Leahey, Rebecca, Shields, Shannon D., Balestrini, Alessia, Riol-Blanco, Lorena, Safina, Brian S., Volgraf, Matthew, Magnuson, Steven, Kakiuchi-Kiyota, Satoko
Published in Journal of medicinal chemistry (14.03.2024)

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Discovery and Structural Characterization of a New Inhibitor Series of HIV-1 Nucleocapsid Function: NMR Solution Structure Determination of a Ternary Complex Involving a 2:1 Inhibitor/NC Stoichiometry

Discovery and Structural Characterization of a New Inhibitor Series of HIV-1 Nucleocapsid Function: NMR Solution Structure Determination of a Ternary Complex Involving a 2:1 Inhibitor/NC Stoichiometry

by Goudreau, Nathalie, Hucke, Oliver, Faucher, Anne-Marie, Grand-Maître, Chantal, Lepage, Olivier, Bonneau, Pierre R., Mason, Stephen W., Titolo, Steve
Published in Journal of molecular biology (12.06.2013)

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Structure−Activity Study on a Novel Series of Macrocyclic Inhibitors of the Hepatitis C Virus NS3 Protease Leading to the Discovery of BILN 2061

Structure−Activity Study on a Novel Series of Macrocyclic Inhibitors of the Hepatitis C Virus NS3 Protease Leading to the Discovery of BILN 2061

by Llinàs-Brunet, Montse, Bailey, Murray D, Bolger, Gordon, Brochu, Christian, Faucher, Anne-Marie, Ferland, Jean Marie, Garneau, Michel, Ghiro, Elise, Gorys, Vida, Grand-Maître, Chantal, Halmos, Ted, Lapeyre-Paquette, Nicole, Liard, Francine, Poirier, Martin, Rhéaume, Manon, Tsantrizos, Youla S, Lamarre, Daniel
Published in Journal of medicinal chemistry (25.03.2004)

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Design, synthesis and biological evaluation of novel aminothiazoles as antiviral compounds acting against human rhinovirus

Design, synthesis and biological evaluation of novel aminothiazoles as antiviral compounds acting against human rhinovirus

by Décor, Anne, Grand-Maître, Chantal, Hucke, Oliver, O’Meara, Jeff, Kuhn, Cyrille, -Forget, Léa Constantineau, Brochu, Christian, Malenfant, Eric, Bertrand-Laperle, Mégan, Bordeleau, Josée, Ghiro, Elise, Pesant, Marc, Fazal, Gulrez, Gorys, Vida, Little, Michael, Boucher, Colette, Bordeleau, Sylvain, Turcotte, Pascal, Guo, Tim, Garneau, Michel, Spickler, Catherine, Gauthier, Annick
Published in Bioorganic & medicinal chemistry letters (01.07.2013)

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Chemo-enzymatic synthesis of chiral 2-substituted succinic acid derivatives

Chemo-enzymatic synthesis of chiral 2-substituted succinic acid derivatives

by Bailey, Murray D., Halmos, Ted, Adamson, Dan, Bordeleau, Josée, Grand-Maı̂tre, Chantal
Published in Tetrahedron: asymmetry (27.08.1999)

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Potent Inhibitors of the Hepatitis C Virus NS3 Protease: Design and Synthesis of Macrocyclic Substrate-Based β-Strand Mimics

Potent Inhibitors of the Hepatitis C Virus NS3 Protease: Design and Synthesis of Macrocyclic Substrate-Based β-Strand Mimics

by Goudreau, Nathalie, Brochu, Christian, Cameron, Dale R, Duceppe, Jean-Simon, Faucher, Anne-Marie, Ferland, Jean-Marie, Grand-Maître, Chantal, Poirier, Martin, Simoneau, Bruno, Tsantrizos, Youla S
Published in Journal of organic chemistry (17.09.2004)

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Characterization of the Human Cytomegalovirus Protease As an Induced-Fit Serine Protease and the Implications to the Design of Mechanism-Based Inhibitors

Characterization of the Human Cytomegalovirus Protease As an Induced-Fit Serine Protease and the Implications to the Design of Mechanism-Based Inhibitors

by LaPlante, Steven R, Bonneau, Pierre R, Aubry, Norman, Cameron, Dale R, Déziel, Robert, Grand-Maître, Chantal, Plouffe, Céline, Tong, Liang, Kawai, Stephen H
Published in Journal of the American Chemical Society (07.04.1999)

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Preparation of 3-O-aryl chloramphenicol derivatives via chemoselective copper-catalyzed O-arylation of (1R,2R)-(-)-N-BOC2-amino-1-(4-nitropheny1)-1,3-propanediol using triarylbismuthines

Preparation of 3-O-aryl chloramphenicol derivatives via chemoselective copper-catalyzed O-arylation of (1R,2R)-(-)-N-BOC2-amino-1-(4-nitropheny1)-1,3-propanediol using triarylbismuthines

by Ahmad, Tabinda, Dansereau, Julien, Hebert, Martin, Grand-Maitre, Chantal, Larivee, Alexandre, Siddiqui, Arshad, Gagnon, Alexandre
Published in Tetrahedron letters (21.09.2016)

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Preparation of 3-O-aryl chloramphenicol derivatives via chemoselective copper-catalyzed O-arylation of (1R,2R)-(−)-N-BOC-2-amino-1-(4-nitrophenyl)-1,3-propanediol using triarylbismuthines

Preparation of 3-O-aryl chloramphenicol derivatives via chemoselective copper-catalyzed O-arylation of (1R,2R)-(−)-N-BOC-2-amino-1-(4-nitrophenyl)-1,3-propanediol using triarylbismuthines

by Ahmad, Tabinda, Dansereau, Julien, Hébert, Martin, Grand-Maître, Chantal, Larivée, Alexandre, Siddiqui, Arshad, Gagnon, Alexandre
Published in Tetrahedron letters (21.09.2016)

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Evidence of a Conformational Change in the Human Cytomegalovirus Protease upon Binding of Peptidyl-Activated Carbonyl Inhibitors

Evidence of a Conformational Change in the Human Cytomegalovirus Protease upon Binding of Peptidyl-Activated Carbonyl Inhibitors

by Bonneau, Pierre R, Grand-Maître, Chantal, Greenwood, Daniel J, Lagacé, Lisette, LaPlante, Steven R, Massariol, Marie-Josée, Ogilvie, William W, O'Meara, Jeff A, Kawai, Stephen H
Published in Biochemistry (Easton) (14.10.1997)

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The Conformation of a Peptidyl Methyl Ketone Inhibitor Bound to the Human Cytomegalovirus Protease

The Conformation of a Peptidyl Methyl Ketone Inhibitor Bound to the Human Cytomegalovirus Protease

by LaPlante, Steven R., Cameron, Dale R., Aubry, Norman, Bonneau, Pierre R., Déziel, Robert, Grand-Maître, Chantal, Ogilvie, William W., Kawai, Stephen H.
Published in Angewandte Chemie International Edition (16.10.1998)

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1-Thiazol-2-yl-N-3-methyl-1H-pyrozole-5-carboxylic acid derivatives as antitumor agents

1-Thiazol-2-yl-N-3-methyl-1H-pyrozole-5-carboxylic acid derivatives as antitumor agents

by Cooper, Alan B., Ciblat, Stephane, Shipps, Gerald, Levine, Jedd, Kostura, Matthew, Oza, Vibha, Constantineau-Forget, Lea, Dery, Martin, Grand-Maitre, Chantal, Bruneau-Latour, Nicolas, Bellavance, Edith, Patane, Michael, Siddiqui, Arshad, Luther, Michael
Published in Bioorganic & medicinal chemistry letters (15.09.2017)

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Corrigendum to “1-Thiazol-2-yl-N-3-methyl-1H-pyrozole-5-carboxylic acid derivatives as antitumor agents” [Bioorg. Med. Chem. Lett. 27 (2017) 4471–4477]

Corrigendum to “1-Thiazol-2-yl-N-3-methyl-1H-pyrozole-5-carboxylic acid derivatives as antitumor agents” [Bioorg. Med. Chem. Lett. 27 (2017) 4471–4477]

by Cooper, Alan B., Ciblat, Stephane, Shipps, Gerald, Levine, Jedd, Kostura, Matthew, Oza, Vibha, Constantineau-Forget, Lea, Dery, Martin, Grand-Maitre, Chantal, Bruneau-Latour, Nicolas, Bellavance, Edith, Patane, Michael, Siddiqui, Arshad, Luther, Michael
Published in Bioorganic & medicinal chemistry letters (01.03.2018)

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Monitoring binding of HIV-1 capsid assembly inhibitors using (19)F ligand-and (15)N protein-based NMR and X-ray crystallography: early hit validation of a benzodiazepine series

Monitoring binding of HIV-1 capsid assembly inhibitors using (19)F ligand-and (15)N protein-based NMR and X-ray crystallography: early hit validation of a benzodiazepine series

by Goudreau, Nathalie, Coulombe, René, Faucher, Anne-Marie, Grand-Maître, Chantal, Lacoste, Jean-Eric, Lemke, Christopher T, Malenfant, Eric, Bousquet, Yves, Fader, Lee, Simoneau, Bruno, Mercier, Jean-François, Titolo, Steve, Mason, Stephen W
Published in ChemMedChem (01.03.2013)

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Monitoring Binding of HIV‐1 Capsid Assembly Inhibitors Using 19 F Ligand‐and 15 N Protein‐Based NMR and X‐ray Crystallography: Early Hit Validation of a Benzodiazepine Series

Monitoring Binding of HIV‐1 Capsid Assembly Inhibitors Using 19 F Ligand‐and 15 N Protein‐Based NMR and X‐ray Crystallography: Early Hit Validation of a Benzodiazepine Series

by Goudreau, Nathalie, Coulombe, René, Faucher, Anne‐Marie, Grand‐Maître, Chantal, Lacoste, Jean‐Eric, Lemke, Christopher T., Malenfant, Eric, Bousquet, Yves, Fader, Lee, Simoneau, Bruno, Mercier, Jean‐François, Titolo, Steve, Mason, Stephen W.
Published in ChemMedChem (01.03.2013)

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