Metabotropic glutamate receptor 1 acts as a dependence receptor creating a requirement for glutamate to sustain the viability and growth of human melanomas
Gelb, T, Pshenichkin, S, Rodriguez, O C, Hathaway, H A, Grajkowska, E, DiRaddo, J O, Wroblewska, B, Yasuda, R P, Albanese, C, Wolfe, B B, Wroblewski, J T
Published in Oncogene (21.05.2015)
Published in Oncogene (21.05.2015)
Get full text
Journal Article
JS01.5.A PHASE 2 TRIAL OF CARBOPLATIN AND BEVACIZUMAB FOR RECURRENT ADULT EPENDYMOMA. A CERN STUDY
Gilbert, M R, Omuro, A, Yuan, Y, Mendoza, T, Wall, K, Grajkowska, E, Vera, E, Reyes, J, Aldape, K, Penas-Prado, M, Walbert, T, Mikkelsen, T, Weathers, S, O'Brien, B, DeGroot, J, Puduvalli, V, Pentsova, E, DeAngelis, L, Kaley, T, Gavrilovic, I, Batchelor, T, Armstrong, T S
Published in Neuro-oncology (Charlottesville, Va.) (08.09.2023)
Published in Neuro-oncology (Charlottesville, Va.) (08.09.2023)
Get full text
Journal Article
P09.10.B THE COVID-19 PANDEMIC EXPERIENCE FOR PATIENTS WITH CENTRAL NERVOUS SYSTEM (CNS) TUMORS: DIFFERENCES IN MOOD AND ASSOCIATED HEALTH STATUS WITH RECOMMENDATIONS FOR PRACTICE
King, A L, Roche, K N, Pillai, V, Polskin, L, Acquaye-Mallory, A A, Boris, L, Burton, E, Choi, A, Grajkowska, E, Lollo, N, Ozer, B, Panzer, M, Penas-Prado, M, Reyes, J, Sahebjam, S, Theeler, B J, Wu, J, Gilbert, M R, Vera, E, Armstrong, T S
Published in Neuro-oncology (Charlottesville, Va.) (08.09.2023)
Published in Neuro-oncology (Charlottesville, Va.) (08.09.2023)
Get full text
Journal Article
Synthesis of Urea-Based Inhibitors as Active Site Probes of Glutamate Carboxypeptidase II: Efficacy as Analgesic Agents
Kozikowski, Alan P, Zhang, Jiazhong, Nan, Fajun, Petukhov, Pavel A, Grajkowska, Ewa, Wroblewski, Jarda T, Yamamoto, Tatsuo, Bzdega, Tomasz, Wroblewska, Barbara, Neale, Joseph H
Published in Journal of medicinal chemistry (25.03.2004)
Published in Journal of medicinal chemistry (25.03.2004)
Get full text
Journal Article
Antinociceptive effects of N-acetylaspartylglutamate (NAAG) peptidase inhibitors ZJ-11, ZJ-17 and ZJ-43 in the rat formalin test and in the rat neuropathic pain model
Yamamoto, Tatsuo, Hirasawa, Serabi, Wroblewska, Barbara, Grajkowska, Ewa, Zhou, Jia, Kozikowski, Alan, Wroblewski, Jarda, Neale, Joseph H.
Published in The European journal of neuroscience (01.07.2004)
Published in The European journal of neuroscience (01.07.2004)
Get full text
Journal Article
l-Homocysteine Sulfinic Acid and Other Acidic Homocysteine Derivatives Are Potent and Selective Metabotropic Glutamate Receptor Agonists
Shi, Qi, Savage, Jason E, Hufeisen, Sandra J, Rauser, Laura, Grajkowska, Ewa, Ernsberger, Paul, Wroblewski, Jarda T, Nadeau, Joseph H, Roth, Bryan L
Published in The Journal of pharmacology and experimental therapeutics (01.04.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.04.2003)
Get full text
Journal Article
Synthesis and receptor assay of aromatic–ethynyl–aromatic derivatives with potent mGluR5 antagonist activity
Alagille, David, Baldwin, Ronald M., Roth, Bryan L., Wroblewski, Jarda T., Grajkowska, Ewa, Tamagnan, Gilles D.
Published in Bioorganic & medicinal chemistry (03.01.2005)
Published in Bioorganic & medicinal chemistry (03.01.2005)
Get full text
Journal Article
Functionalization at position 3 of the phenyl ring of the potent mGluR5 noncompetitive antagonists MPEP
Alagille, David, Baldwin, Ronald M., Roth, Bryan L., Wroblewski, Jarda T., Grajkowska, Ewa, Tamagnan, Gilles D.
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
Published in Bioorganic & medicinal chemistry letters (15.02.2005)
Get full text
Journal Article
Synthesis of N(1)-substituted analogues of (2R,4R)-4-amino-pyrrolidine-2,4-dicarboxylic acid as agonists, partial agonists, and antagonists of group II metabotropic glutamate receptors
Mukhopadhyaya, J K, Kozikowski, A P, Grajkowska, E, Pshenichkin, S, Wroblewski, J T
Published in Bioorganic & medicinal chemistry letters (23.07.2001)
Published in Bioorganic & medicinal chemistry letters (23.07.2001)
Get full text
Journal Article
Synthesis of N 1 -substituted analogues of (2 R ,4 R )-4-amino-pyrrolidine-2,4-dicarboxylic acid as agonists, partial agonists, and antagonists of group II metabotropic glutamate receptors
Mukhopadhyaya, Jayanta Kumar, Kozikowski, Alan P., Grajkowska, Ewa, Pshenichkin, Sergey, Wroblewski, Jarda T.
Published in Bioorganic & medicinal chemistry letters (23.07.2001)
Published in Bioorganic & medicinal chemistry letters (23.07.2001)
Get full text
Journal Article