Discovery of (3S,3aR)-2-(3-Chloro-4-cyanophenyl)-3-cyclopentyl-3,3a,4,5-tetrahydro-2H-benzo[g]indazole-7-carboxylic Acid (PF-3882845), an Orally Efficacious Mineralocorticoid Receptor (MR) Antagonist for Hypertension and Nephropathy
Meyers, Marvin J, Arhancet, Graciela B, Hockerman, Susan L, Chen, Xiangyang, Long, Scott A, Mahoney, Matthew W, Rico, Joseph R, Garland, Danny J, Blinn, James. R, Collins, Joe T, Yang, Shengtian, Huang, Horng-Chih, McGee, Kevin F, Wendling, Jay M, Dietz, Jessica D, Payne, Maria A, Homer, Bruce L, Heron, Marcia I, Reitz, David B, Hu, Xiao
Published in Journal of medicinal chemistry (26.08.2010)
Published in Journal of medicinal chemistry (26.08.2010)
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Discovery and SAR of PF-4693627, a potent, selective and orally bioavailable mPGES-1 inhibitor for the potential treatment of inflammation
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Published in Bioorganic & medicinal chemistry letters (15.02.2013)
Published in Bioorganic & medicinal chemistry letters (15.02.2013)
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Stereochemical Requirements for the Mineralocorticoid Receptor Antagonist Activity of Dihydropyridines
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Published in Journal of medicinal chemistry (27.05.2010)
Published in Journal of medicinal chemistry (27.05.2010)
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Identification of (R)‑6-(1-(4-Cyano-3-methylphenyl)-5-cyclopentyl-4,5-dihydro‑1H‑pyrazol-3-yl)-2-methoxynicotinic Acid, a Highly Potent and Selective Nonsteroidal Mineralocorticoid Receptor Antagonist
Casimiro-Garcia, Agustin, Piotrowski, David W, Ambler, Catherine, Arhancet, Graciela B, Banker, Mary Ellen, Banks, Tereece, Boustany-Kari, Carine M, Cai, Cuiman, Chen, Xiangyang, Eudy, Rena, Hepworth, David, Hulford, Catherine A, Jennings, Sandra M, Loria, Paula M, Meyers, Marvin J, Petersen, Donna N, Raheja, Neil K, Sammons, Matthew, She, Li, Song, Kun, Vrieze, Derek, Wei, Liuqing
Published in Journal of medicinal chemistry (22.05.2014)
Published in Journal of medicinal chemistry (22.05.2014)
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Discovery of Novel Cyanodihydropyridines as Potent Mineralocorticoid Receptor Antagonists
Arhancet, Graciela B, Woodard, Scott S, Iyanar, Kaliappan, Case, Brenda L, Woerndle, Rhonda, Dietz, Jessica D, Garland, Danny J, Collins, Joe T, Payne, Maria A, Blinn, James R, Pomposiello, Silvia I, Hu, Xiao, Heron, Marcia I, Huang, Horng-Chih, Lee, Len F
Published in Journal of medicinal chemistry (26.08.2010)
Published in Journal of medicinal chemistry (26.08.2010)
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Synthesis and biological evaluation of substituted benzoxazoles as inhibitors of mPGES-1: Use of a conformation-based hypothesis to facilitate compound design
Walker, Daniel P., Arhancet, Graciela B., Lu, Hwang-Fun, Heasley, Steven E., Metz, Sue, Kablaoui, Natasha M., Franco, Francisco M., Hanau, Cathleen E., Scholten, Jeffrey A., Springer, John R., Fobian, Yvette M., Carter, Jeffrey S., Xing, Li, Yang, Shengtian, Shaffer, Alexander F., Jerome, Gina M., Baratta, Michael T., Moore, William M., Vazquez, Michael L.
Published in Bioorganic & medicinal chemistry letters (15.02.2013)
Published in Bioorganic & medicinal chemistry letters (15.02.2013)
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Synthesis and Characterization of Novel Surfactants Based on 2-Hydroxy-4-(Methylthio)Butanoic Acid: 1. Anionic Surfactants
Yu, Guangzhe, Long, Scott A., Karinshak, Kyle A., Grady, Brian P., Harwell, Jeff H., Arhancet, Graciela B.
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FUNCTIONALIZED POLYMER COMPOSITION
WANG XIAOJUN, GRACIELA B ARHANCET, MATTHEW MAHONEY, RANGARANI KARNATI
Year of Publication 08.02.2018
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Year of Publication 08.02.2018
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Insulin sensitizing pharmacology of thiazolidinediones correlates with mitochondrial gene expression rather than activation of PPAR gamma
Bolten, Charles W, Blanner, Patrick M, McDonald, William G, Staten, Nicholas R, Mazzarella, Richard A, Arhancet, Graciela B, Meier, Martin F, Weiss, David J, Sullivan, Patrick M, Hromockyj, Alexander E, Kletzien, Rolf F, Colca, Jerry R
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Thiazolidinediones inhibit the progression of established hypertension in the Dahl salt-sensitive rat
Bolten, Charles W, Payne, Maria A, McDonald, William G, Blanner, Patrick M, Chott, Robert C, Ghosh, Sarbani, Arhancet, Graciela B, Staten, Nicholas R, Gulve, Eric A, Sullivan, Patrick M, Hromockyj, Alexander E, Colca, Jerry R
Published in Diabetes & vascular disease research (01.06.2007)
Published in Diabetes & vascular disease research (01.06.2007)
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Discovery of (3 S ,3a R )-2-(3-Chloro-4-cyanophenyl)-3-cyclopentyl-3,3a,4,5-tetrahydro-2 H -benzo[ g ]indazole-7-carboxylic Acid (PF-3882845), an Orally Efficacious Mineralocorticoid Receptor (MR) Antagonist for Hypertension and Nephropathy
Meyers, Marvin J., Arhancet, Graciela B., Hockerman, Susan L., Chen, Xiangyang, Long, Scott A., Mahoney, Matthew W., Rico, Joseph R., Garland, Danny J., Blinn, James. R., Collins, Joe T., Yang, Shengtian, Huang, Horng-Chih, McGee, Kevin F., Wendling, Jay M., Dietz, Jessica D., Payne, Maria A., Homer, Bruce L., Heron, Marcia I., Reitz, David B., Hu, Xiao
Published in Journal of medicinal chemistry (26.08.2010)
Published in Journal of medicinal chemistry (26.08.2010)
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Journal Article
Identification of ( R )-6-(1-(4-Cyano-3-methylphenyl)-5-cyclopentyl-4,5-dihydro-1 H -pyrazol-3-yl)-2-methoxynicotinic Acid, a Highly Potent and Selective Nonsteroidal Mineralocorticoid Receptor Antagonist
Casimiro-Garcia, Agustin, Piotrowski, David W., Ambler, Catherine, Arhancet, Graciela B., Banker, Mary Ellen, Banks, Tereece, Boustany-Kari, Carine M., Cai, Cuiman, Chen, Xiangyang, Eudy, Rena, Hepworth, David, Hulford, Catherine A., Jennings, Sandra M., Loria, Paula M., Meyers, Marvin J., Petersen, Donna N., Raheja, Neil K., Sammons, Matthew, She, Li, Song, Kun, Vrieze, Derek, Wei, Liuqing
Published in Journal of medicinal chemistry (22.05.2014)
Published in Journal of medicinal chemistry (22.05.2014)
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P.J. LENNON P.J. LENNON, R.J. BRINKER R.J. BRINKER, S. HENKE S. HENKE, X. CHEN X. CHEN, HENRY E. AGBAJE HENRY E. AGBAJE, JEFFREY A. GRAHAM JEFFREY A. GRAHAM, M. D. MAHONEY M. D. MAHONEY, W. ABRAHAM W. ABRAHAM, DAVID Z. BECHER DAVID Z. BECHER, N. PALLAS N. PALLAS, X.C. XU X.C. XU, JEANETTE L. GLAENZER JEANETTE L. GLAENZER, GRACIELA B. ARHANCET GRACIELA B. ARHANCET, JANE L. GILLESPIE JANE L. GILLESPIE, A. S. WIDEMAN A. S. WIDEMAN, DANIEL R. WRIGHT DANIEL R. WRIGHT
Year of Publication 31.07.2001
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Year of Publication 31.07.2001
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