β-Turned Dipeptoids as Potent and Selective CCK1 Receptor Antagonists
Martín-Martínez, Mercedes, De la Figuera, Natalia, Latorre, Miriam, Herranz, Rosario, García-López, M. Teresa, Cenarruzabeitia, Edurne, Del Río, Joaquín, González-Muñiz, Rosario
Published in Journal of medicinal chemistry (05.10.2000)
Published in Journal of medicinal chemistry (05.10.2000)
Get full text
Journal Article
Highly constrained dipeptoid analogues containing a type II′ β-turn mimic as novel and selective CCK-A receptor ligands
Figuera, Natalia de la, Martín-Martínez, Mercedes, Herranz, Rosario, Teresa García-López, M., Latorre, Miriam, Cenarruzabeitia, Edurne, del Río, Joaquín, González-Muñiz, Rosario
Published in Bioorganic & medicinal chemistry letters (04.01.1999)
Published in Bioorganic & medicinal chemistry letters (04.01.1999)
Get full text
Journal Article
Boc-Trp-Orn(Z)-Asp-NH2 and derivatives: a new family of CCK antagonists
Gonzalez-Muniz, R, Bergeron, F, Marseigne, I, Durieux, C, Roques, Bernard P
Published in Journal of medicinal chemistry (01.12.1990)
Published in Journal of medicinal chemistry (01.12.1990)
Get full text
Journal Article
Entry to New Conformationally Constrained Amino Acids. First Synthesis of 3-Unsubstituted 4-Alkyl-4-carboxy-2-azetidinone Derivatives via an Intramolecular N α -C α-Cyclization Strategy
Gerona-Navarro, Guillermo, Bonache, Maria Angeles, Herranz, Rosario, García-López, Maria Teresa, González-Muñiz, Rosario
Published in Journal of organic chemistry (18.05.2001)
Published in Journal of organic chemistry (18.05.2001)
Get full text
Journal Article
From 1-Acyl-β-lactam Human Cytomegalovirus Protease Inhibitors to 1-Benzyloxycarbonylazetidines with Improved Antiviral Activity. A Straightforward Approach To Convert Covalent to Noncovalent Inhibitors
Gerona-Navarro, Guillermo, Pérez de Vega, M. Jesús, García-López, M. Teresa, Andrei, Graciela, Snoeck, Robert, De Clercq, Erik, Balzarini, Jan, González-Muñiz, Rosario
Published in Journal of medicinal chemistry (07.04.2005)
Published in Journal of medicinal chemistry (07.04.2005)
Get full text
Journal Article
Stereoselective synthesis of amino acid-derived β-lactams. Experimental evidence for TADDOL as a memory of chirality enhancer
Bonache, M. Angeles, López, Pilar, Martín-Martínez, Mercedes, García-López, M. Teresa, Cativiela, Carlos, González-Muñiz, Rosario
Published in Tetrahedron (02.01.2006)
Published in Tetrahedron (02.01.2006)
Get full text
Journal Article
Synthesis and anti-HCMV activity of 1-acyl-β-lactams and 1-acylazetidines derived from phenylalanine
GERONA-NAVARRO, Guillermo, PEREZ DE VEGA, Ma. Jesus, GARCIA-LOPEZ, Ma. Teresa, ANDREI, Graciela, SNOECK, Robert, BALZARINI, Jan, DE CLERCQ, Erik, GONZALEZ-MUNIZ, Rosario
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Published in Bioorganic & medicinal chemistry letters (03.05.2004)
Get full text
Journal Article
Solid phase synthesis of a fully active analogue of cholecystokinin using the acid-stable Boc-Phe (p-CH2) SO3H as a substitute for Boc-Tyr(SO3H) in CCK8
Gonzalez-Muniz, R, Cornille, F, Bergeron, F, Ficheux, D, Pothier, J, Durieux, C, Roques, B P
Published in International journal of peptide and protein research (01.04.1991)
Published in International journal of peptide and protein research (01.04.1991)
Get more information
Journal Article
Conformationally Constrained CCK4 Analogues Incorporating IBTM and BTD β-Turn Mimetics
Martín-Martínez, Mercedes, De la Figuera, Natalia, LaTorre, Miriam, García-López, M. Teresa, Cenarruzabeitia, Edurne, Del Río, Joaquín, González-Muñiz, Rosario
Published in Journal of medicinal chemistry (01.12.2005)
Published in Journal of medicinal chemistry (01.12.2005)
Get full text
Journal Article
Simple access to novel azetidine-containing conformationally restricted amino acids by chemoselective reduction of β-lactams
Gerona-Navarro, Guillermo, Bonache, M a Angeles, Alı́as, Miriam, Pérez de Vega, M a Jesús, Garcı́a-López, M a Teresa, López, Pilar, Cativiela, Carlos, González-Muñiz, Rosario
Published in Tetrahedron letters (01.03.2004)
Published in Tetrahedron letters (01.03.2004)
Get full text
Journal Article
Memory of chirality in the enantioselective synthesis of beta-lactams derived from amino acids. Influence of the reaction conditions
Bonache, MA, Gerona-Navarro, G, Martin-Martinez, M, Garcia-Lopez, MT, Lopez, P, Cativiela, C, Gonzalez-Muniz, R
Published in Synlett (02.06.2003)
Published in Synlett (02.06.2003)
Get more information
Journal Article
Prolonged antinociceptive activity of pseudodipeptide analogues of Lys-Trp(Nps) and Trp(Nps)-Lys
De Ceballos, M.L., Lopez, A.E., Harto, J.R., Bravo, A., Gomez-Monterrey, I., Gonzalez-Muñiz, R., Garcia-Lopez, M.T., Del Rio, J.
Published in Peptides (New York, N.Y. : 1980) (1992)
Published in Peptides (New York, N.Y. : 1980) (1992)
Get full text
Journal Article
Combination of Molecular Modeling, Site-Directed Mutagenesis, and SAR Studies To Delineate the Binding Site of Pyridopyrimidine Antagonists on the Human CCK1 Receptor
Martín-Martínez, Mercedes, Marty, Anne, Jourdan, Maud, Escrieut, Chantal, Archer, Elodie, González-Muñiz, Rosario, García-López, M. Teresa, Maigret, Bernard, Herranz, Rosario, Fourmy, Daniel
Published in Journal of medicinal chemistry (28.07.2005)
Published in Journal of medicinal chemistry (28.07.2005)
Get full text
Journal Article
Analogues of the neuroprotective tripeptide Gly-Pro-Glu (GPE): synthesis and structure–activity relationships
Alonso De Diego, Sergio A., Muñoz, Pilar, González-Muñiz, Rosario, Herranz, Rosario, Martín-Martínez, Mercedes, Cenarruzabeitia, Edurne, Frechilla, Diana, Del Río, Joaquín, Luisa Jimeno, M., Teresa García-López, M.
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
Published in Bioorganic & medicinal chemistry letters (02.05.2005)
Get full text
Journal Article
New Gly-Pro-Glu (GPE) analogues: Expedite solid-phase synthesis and biological activity
Alonso De Diego, Sergio A., Gutiérrez-Rodríguez, Marta, Pérez de Vega, M. Jesús, Casabona, Diego, Cativiela, Carlos, González-Muñiz, Rosario, Herranz, Rosario, Cenarruzabeitia, Edurne, Frechilla, Diana, Río, Joaquín Del, Luisa Jimeno, M., Teresa García-López, M.
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
Published in Bioorganic & medicinal chemistry letters (01.03.2006)
Get full text
Journal Article
Memory of chirality in the stereoselective synthesis of β-lactams: importance of the starting amino acid derivative
Bonache, M a̱ Angeles, Gerona-Navarro, Guillermo, Garcı́a-Aparicio, Carlos, Alı́as, Miriam, Martı́n-Martı́nez, Mercedes, Garcı́a-López, M a̱ Teresa, López, Pilar, Cativiela, Carlos, González-Muñiz, Rosario
Published in Tetrahedron: asymmetry (01.08.2003)
Published in Tetrahedron: asymmetry (01.08.2003)
Get full text
Journal Article