Triazine-Based Vanilloid 1 Receptor Open Channel Blockers: Design, Synthesis, Evaluation, and SAR Analysis
Vidal-Mosquera, Miquel, Fernández-Carvajal, Asia, Moure, Alejandra, Valente, Pierluigi, Planells-Cases, Rosa, González-Ros, José M, Bujons, Jordi, Ferrer-Montiel, Antonio, Messeguer, Angel
Published in Journal of medicinal chemistry (10.11.2011)
Published in Journal of medicinal chemistry (10.11.2011)
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Steady-state and time-resolved fluorescent methodologies to characterize the conformational landscape of the selectivity filter of K+ channels
Renart, María Lourdes, Giudici, Ana Marcela, González-Ros, José M., Poveda, José A.
Published in Methods (San Diego, Calif.) (01.05.2024)
Published in Methods (San Diego, Calif.) (01.05.2024)
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Towards understanding the molecular basis of ion channel modulation by lipids: Mechanistic models and current paradigms
Poveda, José A., Marcela Giudici, A., Lourdes Renart, M., Morales, Andrés, González-Ros, José M.
Published in Biochimica et biophysica acta. Biomembranes (01.09.2017)
Published in Biochimica et biophysica acta. Biomembranes (01.09.2017)
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Membranes: a meeting point for lipids, proteins and therapies
Escribá, Pablo V., González‐Ros, José M., Goñi, Félix M., Kinnunen, Paavo K. J., Vigh, Lászlo, Sánchez‐Magraner, Lissete, Fernández, Asia M., Busquets, Xavier, Horváth, Ibolya, Barceló‐Coblijn, Gwendolyn
Published in Journal of cellular and molecular medicine (01.06.2008)
Published in Journal of cellular and molecular medicine (01.06.2008)
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Differential binding of monovalent cations to KcsA: Deciphering the mechanisms of potassium channel selectivity
Montoya, Estefanía, Lourdes Renart, M., Marcela Giudici, A., Poveda, José A., Fernández, Asia M., Morales, Andrés, González-Ros, José M.
Published in Biochimica et biophysica acta. Biomembranes (01.05.2017)
Published in Biochimica et biophysica acta. Biomembranes (01.05.2017)
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Antifungal effects and mechanism of action of viscotoxin A3
Giudici, Marcela, Antonio Poveda, José, Molina, María Luisa, de la Canal, Laura, González‐Ros, José M., Pfüller, Karola, Pfüller, Uwe, Villalaín, José
Published in The FEBS journal (01.01.2006)
Published in The FEBS journal (01.01.2006)
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Journal Article
Clustering and Coupled Gating Modulate the Activity in KcsA, a Potassium Channel Model
Molina, Maria L., Barrera, Francisco N., Fernández, Asia M., Poveda, Jose A., Renart, Maria L., Encinar, Jose A., Riquelme, Gloria, González-Ros, Jose M.
Published in The Journal of biological chemistry (07.07.2006)
Published in The Journal of biological chemistry (07.07.2006)
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Journal Article
Modulation of the potassium channel KcsA by anionic phospholipids: Role of arginines at the non-annular lipid binding sites
Poveda, José A., Giudici, A. Marcela, Renart, M. Lourdes, Millet, Oscar, Morales, Andrés, González-Ros, José M., Oakes, Victoria, Furini, Simone, Domene, Carmen
Published in Biochimica et biophysica acta. Biomembranes (01.10.2019)
Published in Biochimica et biophysica acta. Biomembranes (01.10.2019)
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Journal Article
Probing the Structural Dynamics of the Activation Gate of KcsA Using Homo-FRET Measurements
Díaz-García, Clara, Renart, Maria Lourdes, Poveda, José Antonio, Giudici, Ana Marcela, González-Ros, José M, Prieto, Manuel, Coutinho, Ana
Published in International journal of molecular sciences (04.11.2021)
Published in International journal of molecular sciences (04.11.2021)
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Journal Article
Conformational plasticity in the KcsA potassium channel pore helix revealed by homo-FRET studies
Renart, M. Lourdes, Giudici, A. Marcela, Poveda, José A., Fedorov, Aleksander, Berberan-Santos, Mário N., Prieto, Manuel, Díaz-García, Clara, González-Ros, José M., Coutinho, Ana
Published in Scientific reports (17.04.2019)
Published in Scientific reports (17.04.2019)
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Journal Article
Tetraoctylammonium, a Long Chain Quaternary Ammonium Blocker, Promotes a Noncollapsed, Resting-Like Inactivated State in KcsA
Giudici, Ana Marcela, Díaz-García, Clara, Renart, Maria Lourdes, Coutinho, Ana, Prieto, Manuel, González-Ros, José M, Poveda, José Antonio
Published in International journal of molecular sciences (06.01.2021)
Published in International journal of molecular sciences (06.01.2021)
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Journal Article
Modulation of Function, Structure and Clustering of K + Channels by Lipids: Lessons Learnt from KcsA
Renart, María Lourdes, Giudici, Ana Marcela, Díaz-García, Clara, Molina, María Luisa, Morales, Andrés, González-Ros, José M, Poveda, José Antonio
Published in International journal of molecular sciences (07.04.2020)
Published in International journal of molecular sciences (07.04.2020)
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Journal Article
Partitioning of liquid-ordered/liquid-disordered membrane microdomains induced by the fluidifying effect of 2-hydroxylated fatty acid derivatives
Ibarguren, Maitane, López, David J., Encinar, José A., González-Ros, José M., Busquets, Xavier, Escribá, Pablo V.
Published in Biochimica et biophysica acta (01.11.2013)
Published in Biochimica et biophysica acta (01.11.2013)
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Journal Article
Selective exclusion and selective binding both contribute to ion selectivity in KcsA, a model potassium channel
Renart, M. Lourdes, Montoya, Estefanía, Giudici, A. Marcela, Poveda, José A., Fernández, Asia M., Morales, Andrés, González-Ros, José M.
Published in The Journal of biological chemistry (15.09.2017)
Published in The Journal of biological chemistry (15.09.2017)
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Journal Article
Competing Lipid-Protein and Protein-Protein Interactions Determine Clustering and Gating Patterns in the Potassium Channel from Streptomyces lividans (KcsA)
Molina, M. Luisa, Giudici, A. Marcela, Poveda, José A., Fernández-Ballester, Gregorio, Montoya, Estefanía, Renart, M. Lourdes, Fernández, Asia M., Encinar, José A., Riquelme, Gloria, Morales, Andrés, González-Ros, José M.
Published in The Journal of biological chemistry (16.10.2015)
Published in The Journal of biological chemistry (16.10.2015)
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Journal Article
Unfolding and Refolding in Vitro of a Tetrameric, α-Helical Membrane Protein: The Prokaryotic Potassium Channel KcsA
Barrera, Francisco N, Renart, M. Lourdes, Molina, M. Luisa, Poveda, José A, Encinar, José A, Fernández, Asia M, Neira, José L, González-Ros, José M
Published in Biochemistry (Easton) (01.11.2005)
Published in Biochemistry (Easton) (01.11.2005)
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Journal Article
Anionic Phospholipids Shift the Conformational Equilibrium of the Selectivity Filter in the KcsA Channel to the Conductive Conformation: Predicted Consequences on Inactivation
Renart, María Lourdes, Giudici, Ana Marcela, Coll-Díez, Carlos, González-Ros, José M, Poveda, José A
Published in Biomedicines (05.05.2023)
Published in Biomedicines (05.05.2023)
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Journal Article
Proteomic Analysis of Apical Microvillous Membranes of Syncytiotrophoblast Cells Reveals A High Degree of Similarity with Lipid Rafts
Paradela, Alberto, Bravo, Susana B, Henríquez, Mauricio, Riquelme, Gloria, Gavilanes, Francisco, González-Ros, José M, Albar, Juan P
Published in Journal of proteome research (01.11.2005)
Published in Journal of proteome research (01.11.2005)
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Journal Article
Mechanisms Underlying the Strong Inhibition of Muscle-Type Nicotinic Receptors by Tetracaine
Cobo, Raúl, Nikolaeva, Magdalena, Alberola-Die, Armando, Fernández-Ballester, Gregorio, González-Ros, José M, Ivorra, Isabel, Morales, Andrés
Published in Frontiers in molecular neuroscience (08.08.2018)
Published in Frontiers in molecular neuroscience (08.08.2018)
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