Carboxylic Acid Derivatives of Amlexanox Display Enhanced Potency toward TBK1 and IKK ε and Reveal Mechanisms for Selective Inhibition
Beyett, Tyler S, Gan, Xinmin, Reilly, Shannon M, Chang, Louise, Gomez, Andrew V, Saltiel, Alan R, Showalter, Hollis D, Tesmer, John J G
Published in Molecular pharmacology (01.10.2018)
Published in Molecular pharmacology (01.10.2018)
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Inhibition of IKKɛ and TBK1 Improves Glucose Control in a Subset of Patients with Type 2 Diabetes
Oral, Elif A., Reilly, Shannon M., Gomez, Andrew V., Meral, Rasimcan, Butz, Laura, Ajluni, Nevin, Chenevert, Thomas L., Korytnaya, Evgenia, Neidert, Adam H., Hench, Rita, Rus, Diana, Horowitz, Jeffrey F., Poirier, BreAnne, Zhao, Peng, Lehmann, Kim, Jain, Mohit, Yu, Ruth, Liddle, Christopher, Ahmadian, Maryam, Downes, Michael, Evans, Ronald M., Saltiel, Alan R.
Published in Cell metabolism (05.07.2017)
Published in Cell metabolism (05.07.2017)
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FGF21 is required for the metabolic benefits of IKKε/TBK1 inhibition
Reilly, Shannon M, Abu-Odeh, Mohammad, Ameka, Magdalene, DeLuca, Julia H, Naber, Meghan C, Dadpey, Benyamin, Ebadat, Nima, Gomez, Andrew V, Peng, Xiaoling, Poirier, BreAnne, Walk, Elyse, Potthoff, Matthew J, Saltiel, Alan R
Published in The Journal of clinical investigation (17.05.2021)
Published in The Journal of clinical investigation (17.05.2021)
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2043-P: The Biphasic Antiobesogenic Effects of Amlexanox
GOMEZ, ANDREW V., REILLY, SHANNON, ODEH, MOHAMMAD ABU, WALK, ELYSE, SALTIEL, ALAN
Published in Diabetes (New York, N.Y.) (01.06.2019)
Published in Diabetes (New York, N.Y.) (01.06.2019)
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Design, synthesis, and biological activity of substituted 2-amino-5-oxo-5H-chromeno[2,3-b]pyridine-3-carboxylic acid derivatives as inhibitors of the inflammatory kinases TBK1 and IKKε for the treatment of obesity
Beyett, Tyler S., Gan, Xinmin, Reilly, Shannon M., Gomez, Andrew V., Chang, Louise, Tesmer, John J.G., Saltiel, Alan R., Showalter, Hollis D.
Published in Bioorganic & medicinal chemistry (01.11.2018)
Published in Bioorganic & medicinal chemistry (01.11.2018)
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Lipid-coated mesoporous silica nanoparticles for anti-viral applications via delivery of CRISPR-Cas9 ribonucleoproteins
LaBauve, Annette E, Saada, Edwin A, Jones, Iris K A, Mosesso, Richard, Noureddine, Achraf, Techel, Jessica, Gomez, Andrew, Collette, Nicole, Sherman, Michael B, Serda, Rita E, Butler, Kimberly S, Brinker, C Jeffery, Schoeniger, Joseph S, Sasaki, Darryl, Negrete, Oscar A
Published in Scientific reports (27.04.2023)
Published in Scientific reports (27.04.2023)
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Self-assembly/disassembly of giant double-hydrophilic polymersomes at biologically-relevant pH
Shin, Sun Hae Ra, McAninch, Patrick T, Henderson, Ian M, Gomez, Andrew, Greene, Adrienne C, Carnes, Eric C, Paxton, Walter F
Published in Chemical communications (Cambridge, England) (2018)
Published in Chemical communications (Cambridge, England) (2018)
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Journal Article
ERRγ Preserves Brown Fat Innate Thermogenic Activity
Ahmadian, Maryam, Liu, Sihao, Reilly, Shannon M., Hah, Nasun, Fan, Weiwei, Yoshihara, Eiji, Jha, Pooja, De Magalhaes Filho, C. Daniel, Jacinto, Sandra, Gomez, Andrew V., Dai, Yang, Yu, Ruth T., Liddle, Christopher, Atkins, Annette R., Auwerx, Johan, Saltiel, Alan R., Downes, Michael, Evans, Ronald M.
Published in Cell reports (Cambridge) (13.03.2018)
Published in Cell reports (Cambridge) (13.03.2018)
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The Role of Membrane Fluidization in the Gel-Assisted Formation of Giant Polymersomes
Greene, Adrienne C, Henderson, Ian M, Gomez, Andrew, Paxton, Walter F, VanDelinder, Virginia, Bachand, George D
Published in PloS one (13.07.2016)
Published in PloS one (13.07.2016)
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Catecholamines suppress fatty acid re-esterification and increase oxidation in white adipocytes via STAT3
Reilly, Shannon M, Hung, Chao-Wei, Ahmadian, Maryam, Zhao, Peng, Keinan, Omer, Gomez, Andrew V, DeLuca, Julia H, Dadpey, Benyamin, Lu, Donald, Zaid, Jessica, Poirier, BreAnne, Peng, Xiaoling, Yu, Ruth T, Downes, Michael, Liddle, Christopher, Evans, Ronald M, Murphy, Anne N, Saltiel, Alan R
Published in Nature metabolism (01.07.2020)
Published in Nature metabolism (01.07.2020)
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Angiotensin Converting Enzyme (ACE) expression in microglia reduces amyloid β deposition and neurodegeneration by increasing SYK signaling and endolysosomal trafficking
Gomez, Andrew R, Byun, Hyae Ran, Wu, Shaogen, Muhammad, Akm Ghulam, Ikbariyeh, Jasmine, Chen, Jaelin, Muro, Alek, Li, Lin, Bernstein, Kenneth E, Ainsworth, Richard, Tourtellotte, Warren G
Published in bioRxiv : the preprint server for biology (21.05.2024)
Published in bioRxiv : the preprint server for biology (21.05.2024)
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Dancing pharynx
Liew, Yew, Junior, Andrew, Bakri, Adzreil, Narayanan, Prepageran
Published in Ci ji yi xue za zhi (01.07.2020)
Published in Ci ji yi xue za zhi (01.07.2020)
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Modulating amyloid‐beta proteostasis in the brain of 5xFAD mice by selective expression of angiotensin converting enzyme in microglia
Gomez, Andrew, Wu, Shaogen, Byun, Hyae Ran, Muro, Alek, Muhammad, AKM Ghulam, Li, Lin, Tourtellotte, Warren G
Published in Alzheimer's & dementia (01.12.2023)
Published in Alzheimer's & dementia (01.12.2023)
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