Identification of apoptosis signal-regulating kinase 1 (ASK1) inhibitors among the derivatives of benzothiazol-2-yl-3-hydroxy-5-phenyl-1,5-dihydro-pyrrol-2-one
Starosyla, Sergiy A., Volynets, Galyna P., Lukashov, Sergiy S., Gorbatiuk, Oksana B., Golub, Andriy G., Bdzhola, Volodymyr G., Yarmoluk, Sergiy M.
Published in Bioorganic & medicinal chemistry (15.05.2015)
Published in Bioorganic & medicinal chemistry (15.05.2015)
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Journal Article
Identification of 3H-Naphtho[1,2,3-de]quinoline-2,7-diones as Inhibitors of Apoptosis Signal-Regulating Kinase 1 (ASK1)
Volynets, Galyna P, Chekanov, Maksym O, Synyugin, Anatoliy R, Golub, Andriy G, Kukharenko, Oleksandr P, Bdzhola, Volodymyr G, Yarmoluk, Sergiy M
Published in Journal of medicinal chemistry (28.04.2011)
Published in Journal of medicinal chemistry (28.04.2011)
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Journal Article
Synthesis and biological evaluation of substituted (thieno[2,3-d]pyrimidin-4-ylthio)carboxylic acids as inhibitors of human protein kinase CK2
Golub, Andriy G., Bdzhola, Volodymyr G., Briukhovetska, Nadiia V., Balanda, Anatoliy O., Kukharenko, Olexander P., Kotey, Igor M., Ostrynska, Olga V., Yarmoluk, Sergiy M.
Published in European journal of medicinal chemistry (01.03.2011)
Published in European journal of medicinal chemistry (01.03.2011)
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Journal Article
Rational design of apoptosis signal-regulating kinase 1 inhibitors: Discovering novel structural scaffold
Volynets, Galyna P., Bdzhola, Volodymyr G., Golub, Andriy G., Synyugin, Anatoliy R., Chekanov, Maksym A., Kukharenko, Oleksandr P., Yarmoluk, Sergiy M.
Published in European journal of medicinal chemistry (01.03.2013)
Published in European journal of medicinal chemistry (01.03.2013)
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Journal Article
Structural Hypervariability of the Two Human Protein Kinase CK2 Catalytic Subunit Paralogs Revealed by Complex Structures with a Flavonol- and a Thieno[2,3-d]pyrimidine-Based Inhibitor
Niefind, Karsten, Bischoff, Nils, Golub, Andriy G, Bdzhola, Volodymyr G, Balanda, Anatoliy O, Prykhod'ko, Andriy O, Yarmoluk, Sergiy M
Published in Pharmaceuticals (Basel, Switzerland) (11.01.2017)
Published in Pharmaceuticals (Basel, Switzerland) (11.01.2017)
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Journal Article
Discovery of potent anti-tuberculosis agents targeting leucyl-tRNA synthetase
Gudzera, Olga I., Golub, Andriy G., Bdzhola, Volodymyr G., Volynets, Galyna P., Lukashov, Sergiy S., Kovalenko, Oksana P., Kriklivyi, Ivan A., Yaremchuk, Anna D., Starosyla, Sergiy A., Yarmoluk, Sergiy M., Tukalo, Michail A.
Published in Bioorganic & medicinal chemistry (01.03.2016)
Published in Bioorganic & medicinal chemistry (01.03.2016)
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Journal Article
A Note of Caution on the Role of Halogen Bonds for Protein Kinase/Inhibitor Recognition Suggested by High- And Low-Salt CK2α Complex Structures
Guerra, Barbara, Bischoff, Nils, Bdzhola, Volodymyr G, Yarmoluk, Sergiy M, Issinger, Olaf-Georg, Golub, Andriy G, Niefind, Karsten
Published in ACS chemical biology (17.07.2015)
Published in ACS chemical biology (17.07.2015)
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Journal Article
Discovery and characterization of synthetic 4′-hydroxyflavones—New CK2 inhibitors from flavone family
Golub, Andriy G., Bdzhola, Volodymyr G., Ostrynska, Olga V., Kyshenia, Iaroslav V., Sapelkin, Vladislav M., Prykhod’ko, Andriy O., Kukharenko, Olexander P., Yarmoluk, Sergiy M.
Published in Bioorganic & medicinal chemistry (01.11.2013)
Published in Bioorganic & medicinal chemistry (01.11.2013)
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Journal Article
Identification of Mycobacterium tuberculosis leucyl-tRNA synthetase (LeuRS) inhibitors among the derivatives of 5-phenylamino-2H-[1,2,4]triazin-3-one
Gudzera, Olga I., Golub, Andriy G., Bdzhola, Volodymyr G., Volynets, Galyna P., Kovalenko, Oksana P., Boyarshin, Konstantin S., Yaremchuk, Anna D., Protopopov, Mykola V., Yarmoluk, Sergiy M., Tukalo, Michail A.
Published in Journal of enzyme inhibition and medicinal chemistry (02.11.2016)
Published in Journal of enzyme inhibition and medicinal chemistry (02.11.2016)
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Journal Article
Discovery of new scaffolds for rational design of HCV NS5B polymerase inhibitors
Golub, Andriy G., Gurukumar, K.R., Basu, Amartya, Bdzhola, Volodymyr G., Bilokin, Yaroslav, Yarmoluk, Sergiy M., Lee, Jin-Ching, Talele, Tanaji T., Nichols, Daniel B., Kaushik-Basu, Neerja
Published in European journal of medicinal chemistry (01.12.2012)
Published in European journal of medicinal chemistry (01.12.2012)
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Journal Article
Structure-based discovery of novel flavonol inhibitors of human protein kinase CK2
Golub, Andriy G., Bdzhola, Volodymyr G., Kyshenia, Yaroslav V., Sapelkin, Vladislav M., Prykhod’ko, Andriy O., Kukharenko, Olexander P., Ostrynska, Olga V., Yarmoluk, Sergiy M.
Published in Molecular and cellular biochemistry (01.10.2011)
Published in Molecular and cellular biochemistry (01.10.2011)
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Journal Article
Design and synthesis of novel protein kinase CK2 inhibitors on the base of 4-aminothieno[2,3-d]pyrimidines
Ostrynska, Olga V., Balanda, Anatoliy O., Bdzhola, Volodymyr G., Golub, Andriy G., Kotey, Igor M., Kukharenko, Olexander P., Gryshchenko, Andrii A., Briukhovetska, Nadiia V., Yarmoluk, Sergiy M.
Published in European journal of medicinal chemistry (10.06.2016)
Published in European journal of medicinal chemistry (10.06.2016)
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Journal Article
In vitro Activation of heme oxygenase-2 by menadione and its analogs
Vukomanovic, Dragic, Rahman, Mona N, Bilokin, Yaroslav, Golub, Andriy G, Brien, James F, Szarek, Walter A, Jia, Zongchao, Nakatsu, Kanji
Published in Medical gas research (18.02.2014)
Published in Medical gas research (18.02.2014)
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Journal Article
Identification of 3 H -Naphtho[1,2,3- de ]quinoline-2,7-diones as Inhibitors of Apoptosis Signal-Regulating Kinase 1 (ASK1)
Volynets, Galyna P., Chekanov, Maksym O., Synyugin, Anatoliy R., Golub, Andriy G., Kukharenko, Oleksandr P., Bdzhola, Volodymyr G., Yarmoluk, Sergiy M.
Published in Journal of medicinal chemistry (28.04.2011)
Published in Journal of medicinal chemistry (28.04.2011)
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Journal Article
In vitroActivation of heme oxygenase-2 by menadione and its analogs
Vukomanovic, Dragic, Rahman, Mona N, Bilokin, Yaroslav, Golub, Andriy G, Brien, James F, Szarek, Walter A, Jia, Zongchao, Nakatsu, Kanji
Published in Medical gas research (18.02.2014)
Published in Medical gas research (18.02.2014)
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Journal Article