Metabolism, Excretion, and Mass Balance of the HIV-1 Integrase Inhibitor Dolutegravir in Humans
CASTELLINO, Stephen, MOSS, Lee, PISCITELLI, Stephen C, SAVINA, Paul M, WAGNER, David, BORLAND, Julie, SONG, Ivy, SHUGUANG CHEN, YU LOU, MIN, Sherene S, GOLJER, Igor, CULP, Amanda
Published in Antimicrobial Agents and Chemotherapy (01.08.2013)
Published in Antimicrobial Agents and Chemotherapy (01.08.2013)
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Enantiomeric separation and determination of absolute stereochemistry of asymmetric molecules in drug discovery-Building chiral technology toolboxes
McConnell, Oliver, Bach II, Alvin, Balibar, Carl, Byrne, Neal, Cai, Yanxuan, Carter, Guy, Chlenov, Michael, Di, Li, Fan, Kristi, Goljer, Igor, He, Yanan, Herold, Don, Kagan, Michael, Kerns, Edward, Koehn, Frank, Kraml, Christina, Marathias, Vasilios, Marquez, Brian, McDonald, Leonard, Nogle, Lisa, Petucci, Christopher, Schlingmann, Gerhard, Tawa, Gregory, Tischler, Mark, Williamson, R. Thomas, Sutherland, Alan, Watts, William, Young, Mairead, Zhang, Mei-Yi, Zhang, Yingru, Zhou, Dahui, Ho, Douglas
Published in Chirality (New York, N.Y.) (01.09.2007)
Published in Chirality (New York, N.Y.) (01.09.2007)
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The metabolism and disposition of GSK2140944 in healthy human subjects
Negash, Kitaw, Andonian, Clara, Felgate, Clive, Chen, Cathy, Goljer, Igor, Squillaci, Bianca, Nguyen, Dung, Pirhalla, Jill, Lev, Mally, Schubert, Ernest, Tiffany, Courtney, Hossain, Mohammad, Ho, May
Published in Xenobiotica (02.08.2016)
Published in Xenobiotica (02.08.2016)
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Journal Article
Regioselective Synthesis of Substituted Pyrroles: Efficient Palladium-Catalyzed Cyclization of Internal Alkynes and 2-Amino-3-iodoacrylate Derivatives
Crawley, Matthew L, Goljer, Igor, Jenkins, Douglas J, Mehlmann, John F, Nogle, Lisa, Dooley, Rebecca, Mahaney, Paige E
Published in Organic letters (07.12.2006)
Published in Organic letters (07.12.2006)
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Modulation of Wnt Signaling Through Inhibition of Secreted Frizzled-Related Protein I (sFRP-1) with N-Substituted Piperidinyl Diphenylsulfonyl Sulfonamidest
Moore, William J., Kern, Jeffrey C., Bhat, Ramesh, Commons, Thomas J., Fukayama, Shoichi, Goljer, Igor, Krishnamurthy, Girija, Magolda, Ronald L., Nogle, Lisa, Pitts, Keith, Stauffer, Barb, Trybulski, Eugene J., Welmaker, Gregory S., Wilson, Matthew, Bodine, Peter V. N.
Published in Journal of medicinal chemistry (08.01.2009)
Published in Journal of medicinal chemistry (08.01.2009)
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Identification of Phenylsulfone-Substituted Quinoxaline (WYE-672) as a Tissue Selective Liver X-receptor (LXR) Agonist
Hu, Baihua, Unwalla, Rayomand J, Goljer, Igor, Jetter, James W, Quinet, Elaine M, Berrodin, Thomas J, Basso, Michael D, Feingold, Irene B, Nilsson, Annika Goos, Wilhelmsson, Anna, Evans, Mark J, Wrobel, Jay E
Published in Journal of medicinal chemistry (22.04.2010)
Published in Journal of medicinal chemistry (22.04.2010)
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Journal Article
Modulation of Wnt Signaling Through Inhibition of Secreted Frizzled-Related Protein I (sFRP-1) with N-Substituted Piperidinyl Diphenylsulfonyl Sulfonamides
Moore, William J, Kern, Jeffrey C, Bhat, Ramesh, Commons, Thomas J, Fukayama, Shoichi, Goljer, Igor, Krishnamurthy, Girija, Magolda, Ronald L, Nogle, Lisa, Pitts, Keith, Stauffer, Barb, Trybulski, Eugene J, Welmaker, Gregory S, Wilson, Matthew, Bodine, Peter V. N
Published in Journal of medicinal chemistry (08.01.2009)
Published in Journal of medicinal chemistry (08.01.2009)
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Journal Article
Metabolism of Intravenous Methylnaltrexone in Mice, Rats, Dogs, and Humans
CHANDRASEKARAN, Appavu, TONG, Zeen, SCATINA, Joann, HONGSHAN LI, ERVE, John C. L, DEMAIO, William, GOLJER, Igor, MCCONNELL, Oliver, ROTSHTEYN, Yakov, HULTIN, Theresa, TALAAT, Rasmy
Published in Drug metabolism and disposition (01.04.2010)
Published in Drug metabolism and disposition (01.04.2010)
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Journal Article
Evaluating Indole-Related Derivatives as Precursors in the Directed Biosynthesis of Diazepinomicin Analogues
Ratnayake, Anokha S, Janso, Jeffrey E, Feng, Xidong, Schlingmann, Gerhard, Goljer, Igor, Carter, Guy T
Published in Journal of natural products (Washington, D.C.) (27.03.2009)
Published in Journal of natural products (Washington, D.C.) (27.03.2009)
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Journal Article
Efficient, Regioselective Palladium-Catalyzed Tandem Heck-Isomerization Reaction of Aryl Bromides and Non-Allylic Benzyl Alcohols
Crawley, Matthew L, Phipps, Kristin M, Goljer, Igor, Mehlmann, John F, Lundquist, Joseph T, Ullrich, John W, Yang, Cuijian, Mahaney, Paige E
Published in Organic letters (05.03.2009)
Published in Organic letters (05.03.2009)
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Journal Article
Unexpected rearrangement of enantiomerically pure 3-aminoquinuclidine as a simple way of preparing diastereomeric octahydropyrrolo[2,3-c]pyridine derivatives
Goljer, Igor, Molinari, Albert, He, Yanan, Nogle, Lisa, Sun, Weilin, Campbell, Brandon, McConnell, Oliver
Published in Chirality (New York, N.Y.) (01.07.2009)
Published in Chirality (New York, N.Y.) (01.07.2009)
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Journal Article
Proton NMR spectroscopy shows lipids accumulate in skeletal muscle in response to burn trauma-induced apoptosis
Astrakas, Loukas G, Goljer, Igor, Yasuhara, Shingo, Padfield, Katie E, Zhang, Qunhao, Gopalan, Suresh, Mindrinos, Michael N, Dai, George, Yu, Yong-Ming, Martyn, J. A. Jeevendra, Tompkins, Ronald G, Rahme, Laurence G, Tzika, A. Aria
Published in The FASEB journal (01.09.2005)
Published in The FASEB journal (01.09.2005)
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Simultaneous determination of 1 H– 1 H and 1 H– 13 C residual dipolar couplings in a chiral liquid crystal solvent using a natural abundance HSQC experiment
Marathias, Vasilios M., Goljer, Igor, Bach II, Alvin C.
Published in Magnetic resonance in chemistry (01.07.2005)
Published in Magnetic resonance in chemistry (01.07.2005)
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3-(Arylamino)-3-phenylpropan-2-olamines as a new series of dual norepinephrine and serotonin reuptake inhibitors
Vu, An T., Cohn, Stephen T., Terefenko, Eugene A., Moore, William J., Zhang, Puwen, Mahaney, Paige E., Trybulski, Eugene J., Goljer, Igor, Dooley, Rebecca, Bray, Jenifer A., Johnston, Grace H., Leiter, Jennifer, Deecher, Darlene C.
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
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Journal Article
Solution Structure of a Duplex DNA with an Abasic Site in a dA Tract
Wang, Ke Yu, Parker, Sharon A, Goljer, Igor, Bolton, Philip H
Published in Biochemistry (Easton) (30.09.1997)
Published in Biochemistry (Easton) (30.09.1997)
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