Constrained Peptides with Target-Adapted Cross-Links as Inhibitors of a Pathogenic Protein-Protein Interaction
Glas, Adrian, Bier, David, Hahne, Gernot, Rademacher, Christoph, Ottmann, Christian, Grossmann, Tom N.
Published in Angewandte Chemie (International ed.) (24.02.2014)
Published in Angewandte Chemie (International ed.) (24.02.2014)
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Journal Article
Adapting free energy perturbation simulations for large macrocyclic ligands: how to dissect contributions from direct binding and free ligand flexibility
Wallraven, Kerstin, Holmelin, Fredrik L, Glas, Adrian, Hennig, Sven, Frolov, Andrey I, Grossmann, Tom N
Published in Chemical science (Cambridge) (28.02.2020)
Published in Chemical science (Cambridge) (28.02.2020)
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Structure-Based Design of Non-natural Macrocyclic Peptides That Inhibit Protein–Protein Interactions
Krüger, Dennis M, Glas, Adrian, Bier, David, Pospiech, Nicole, Wallraven, Kerstin, Dietrich, Laura, Ottmann, Christian, Koch, Oliver, Hennig, Sven, Grossmann, Tom N
Published in Journal of medicinal chemistry (09.11.2017)
Published in Journal of medicinal chemistry (09.11.2017)
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Adapting free energy perturbation simulations for large macrocyclic ligands: how to dissect contributions from direct binding and free ligand flexibility† †Electronic supplementary information (ESI) available. See DOI: 10.1039/c9sc04705k
Wallraven, Kerstin, Holmelin, Fredrik L., Glas, Adrian, Hennig, Sven, Frolov, Andrey I., Grossmann, Tom N.
Published in Chemical science (Cambridge) (22.01.2020)
Published in Chemical science (Cambridge) (22.01.2020)
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Constraining an Irregular Peptide Secondary Structure through Ring-Closing Alkyne Metathesis
Cromm, Philipp M., Wallraven, Kerstin, Glas, Adrian, Bier, David, Fürstner, Alois, Ottmann, Christian, Grossmann, Tom N.
Published in Chembiochem : a European journal of chemical biology (17.10.2016)
Published in Chembiochem : a European journal of chemical biology (17.10.2016)
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Cover Feature: Increased Conformational Flexibility of a Macrocycle–Receptor Complex Contributes to Reduced Dissociation Rates (Chem. Eur. J. 64/2017)
Glas, Adrian, Wamhoff, Eike‐Christian, Krüger, Dennis M., Rademacher, Christoph, Grossmann, Tom N.
Published in Chemistry : a European journal (16.11.2017)
Published in Chemistry : a European journal (16.11.2017)
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Back Cover: Constrained Peptides with Target-Adapted Cross-Links as Inhibitors of a Pathogenic Protein-Protein Interaction (Angew. Chem. Int. Ed. 9/2014)
Glas, Adrian, Bier, David, Hahne, Gernot, Rademacher, Christoph, Ottmann, Christian, Grossmann, Tom N.
Published in Angewandte Chemie (International ed.) (24.02.2014)
Published in Angewandte Chemie (International ed.) (24.02.2014)
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Journal Article
Makrocyclische Peptide mit dem Zielprotein angepassten Kohlenwasserstoffbrücken: Inhibitoren einer pathogenen Protein‐Protein‐Wechselwirkung
Glas, Adrian, Bier, David, Hahne, Gernot, Rademacher, Christoph, Ottmann, Christian, Grossmann, Tom N.
Published in Angewandte Chemie (24.02.2014)
Published in Angewandte Chemie (24.02.2014)
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Journal Article
Makrocyclische Peptide mit dem Zielprotein angepassten Kohlenwasserstoffbrücken: Inhibitoren einer pathogenen Protein-Protein-Wechselwirkung
Glas, Adrian, Bier, David, Hahne, Gernot, Rademacher, Christoph, Ottmann, Christian, Grossmann, Tom N.
Published in Angewandte Chemie (24.02.2014)
Published in Angewandte Chemie (24.02.2014)
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Journal Article
Rücktitelbild: Makrocyclische Peptide mit dem Zielprotein angepassten Kohlenwasserstoffbrücken: Inhibitoren einer pathogenen Protein-Protein-Wechselwirkung (Angew. Chem. 9/2014)
Glas, Adrian, Bier, David, Hahne, Gernot, Rademacher, Christoph, Ottmann, Christian, Grossmann, Tom N.
Published in Angewandte Chemie (24.02.2014)
Published in Angewandte Chemie (24.02.2014)
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Journal Article