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Roymans, Dirk, Alnajjar, Sarhad S, Battles, Michael B, Sitthicharoenchai, Panchan, Furmanova-Hollenstein, Polina, Rigaux, Peter, Berg, Joke Van den, Kwanten, Leen, Ginderen, Marcia Van, Verheyen, Nick, Vranckx, Luc, Jaensch, Steffen, Arnoult, Eric, Voorzaat, Richard, Gallup, Jack M., Larios-Mora, Alejandro, Crabbe, Marjolein, Huntjens, Dymphy, Raboisson, Pierre, Langedijk, Johannes P., Ackermann, Mark R., McLellan, Jason S, Vendeville, Sandrine, Koul, Anil
Published in Nature communications (01.08.2017)
Published in Nature communications (01.08.2017)
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Resistance Mutations in Human Immunodeficiency Virus Type 1 Integrase Selected with Elvitegravir Confer Reduced Susceptibility to a Wide Range of Integrase Inhibitors
GOETHALS, Olivia, CLAYTON, Reginald, MEERSSEMAN, Geert, JOCHMANS, Dirk, VERMEIRE, Kurt, SCHOLS, Dominique, HALLENBERGER, Sabine, HERTOGS, Kurt, VAN GINDEREN, Marcia, VEREYCKEN, Inge, WAGEMANS, Elisabeth, GELUYKENS, Peggy, DOCKX, Koen, STRIJBOS, Rudy, SMITS, Veerle, VOS, Ann
Published in Journal of Virology (01.11.2008)
Published in Journal of Virology (01.11.2008)
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Binding of a potent small-molecule inhibitor of six-helix bundle formation requires interactions with both heptad-repeats of the RSV fusion protein
Roymans, Dirk, De Bondt, Hendrik L, Arnoult, Eric, Geluykens, Peggy, Gevers, Tom, Van Ginderen, Marcia, Verheyen, Nick, Kim, Hidong, Willebrords, Rudy, Bonfanti, Jean-François, Bruinzeel, Wouter, Cummings, Maxwell D, van Vlijmen, Herman, Andries, Koen
Published in Proceedings of the National Academy of Sciences - PNAS (05.01.2010)
Published in Proceedings of the National Academy of Sciences - PNAS (05.01.2010)
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TMC310911, a Novel Human Immunodeficiency Virus Type 1 Protease Inhibitor, Shows In Vitro an Improved Resistance Profile and Higher Genetic Barrier to Resistance Compared with Current Protease Inhibitors
DIERYNCK, Inge, VAN MARCK, Herwig, VAN GINDEREN, Marcia, JONCKERS, Tim H. M, NALAM, Madhavi N. L, SCHIFFER, Celia A, RAOOF, Araz, KRAUS, Guenter, PICCHIO, Gaston
Published in Antimicrobial Agents and Chemotherapy (01.12.2011)
Published in Antimicrobial Agents and Chemotherapy (01.12.2011)
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Indolopyridones Inhibit Human Immunodeficiency Virus Reverse Transcriptase with a Novel Mechanism of Action
JOCHMANS, Dirk, DEVAL, Jérome, EHTESHAMI, Maryam, WIGERINCK, Piet, GÖTTE, Matthias, HERTOGS, Kurt, KESTELEYN, Bart, VAN MARCK, Herwig, BETTENS, Eva, DE BAERE, Inky, DEHERTOGH, Pascale, IVENS, Tania, VAN GINDEREN, Marcia, VAN SCHOUBROECK, Bertrand
Published in Journal of Virology (01.12.2006)
Published in Journal of Virology (01.12.2006)
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JNJ-7184, a respiratory syncytial virus inhibitor targeting the connector domain of the viral polymerase
Bonneux, Brecht, Shareef, Afzaal, Tcherniuk, Sergey, Anson, Brandon, de Bruyn, Suzanne, Verheyen, Nick, Thys, Kim, Conceição-Neto, Nádia, van Ginderen, Marcia, Kwanten, Leen, Ysebaert, Nina, Vranckx, Luc, Peeters, Elien, Lanckacker, Ellen, Gallup, Jack, Sitthicharoenchai, Panchan, Alnajjar, Sarhad, Ackermann, Mark, Adhikary, Suraj, Bhaumik, Anusarka, Patrick, Aaron, Fung, Amy, Sutto-Ortiz, Priscila, Decroly, Etienne, Mason, Stephen, Lançois, David, Deval, Jerome, Jin, Zhinan, Eléouët, Jean-François, Fearns, Rachel, Koul, Anil, Roymans, Dirk, Rigaux, Peter, Herschke, Florence
Published in Antiviral research (01.07.2024)
Published in Antiviral research (01.07.2024)
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Journal Article
JNJ-7184, a respiratory syncytial virus inhibitor targeting the connector domain of the viral polymerase
Bonneux, Brecht, Shareef, Afzaal, Tcherniuk, Sergey, Anson, Brandon, de Bruyn, Suzanne, Verheyen, Nick, Thys, Kim, Conceição-Neto, Nádia, Van Ginderen, Marcia, Kwanten, Leen, Ysebaert, Nina, Vranckx, Luc, Peeters, Elien, Lanckacker, Ellen, Gallup, Jack M., Sitthicharoenchai, Panchan, Alnajjar, Sarhad, Ackermann, Mark R., Adhikary, Suraj, Bhaumik, Anusarka, Patrick, Aaron, Fung, Amy, Sutto-Ortiz, Priscila, Decroly, Etienne, Mason, Stephen W., Lançois, David, Deval, Jerome, Jin, Zhinan, Eléouët, Jean-François, Fearns, Rachel, Koul, Anil, Roymans, Dirk, Rigaux, Peter, Herschke, Florence
Published in Antiviral research (01.07.2024)
Published in Antiviral research (01.07.2024)
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Primary mutations selected in vitro with raltegravir confer large fold changes in susceptibility to first-generation integrase inhibitors, but minor fold changes to inhibitors with second-generation resistance profiles
Goethals, Olivia, Vos, Ann, Van Ginderen, Marcia, Geluykens, Peggy, Smits, Veerle, Schols, Dominique, Hertogs, Kurt, Clayton, Reginald
Published in Virology (New York, N.Y.) (05.07.2010)
Published in Virology (New York, N.Y.) (05.07.2010)
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Resistance to raltegravir highlights integrase mutations at codon 148 in conferring cross-resistance to a second-generation HIV-1 integrase inhibitor
Goethals, Olivia, Van Ginderen, Marcia, Vos, Ann, Cummings, Maxwell D., Van Der Borght, Koen, Van Wesenbeeck, Liesbeth, Feyaerts, Maxim, Verheyen, Ann, Smits, Veerle, Van Loock, Marnix, Hertogs, Kurt, Schols, Dominique, Clayton, Reginald F.
Published in Antiviral research (01.08.2011)
Published in Antiviral research (01.08.2011)
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