8-Fluoroimidazo[1,2-a]pyridine: Synthesis, physicochemical properties and evaluation as a bioisosteric replacement for imidazo[1,2-a]pyrimidine in an allosteric modulator ligand of the GABAA receptor
Humphries, Alexander C., Gancia, Emanuela, Gilligan, Myra T., Goodacre, Simon, Hallett, David, Merchant, Kevin J., Thomas, Steve R.
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
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Journal Article
4-Fluorosulfonylpiperidines: selective 5-HT2A ligands for the treatment of insomnia
Fish, L Rebecca, Gilligan, Myra T, Humphries, Alexander C, Ivarsson, Magnus, Ladduwahetty, Tammy, Merchant, Kevin J, O'Connor, Desmond, Patel, Smita, Philipps, Elisabeth, Vargas, Hugo M, Hutson, Peter H, MacLeod, Angus M
Published in Bioorganic & medicinal chemistry letters (15.08.2005)
Published in Bioorganic & medicinal chemistry letters (15.08.2005)
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Journal Article
8-Fluoroimidazo[1,2-a]pyridine: synthesis, physicochemical properties and evaluation as a bioisosteric replacement for imidazo[1,2-a]pyrimidine in an allosteric modulator ligand of the GABA A receptor
Humphries, Alexander C, Gancia, Emanuela, Gilligan, Myra T, Goodacre, Simon, Hallett, David, Merchant, Kevin J, Thomas, Steve R
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
Get full text
Journal Article
8-Fluoroimidazo[1,2-a]pyridine: Synthesis, physicochemical properties and evaluation as a bioisosteric replacement for imidazo[1,2-a]pyrimidine in an allosteric modulator ligand of the GABA sub(A) receptor
Humphries, Alexander C, Gancia, Emanuela, Gilligan, Myra T, Goodacre, Simon, Hallett, David, Merchant, Kevin J, Thomas, Steve R
Published in Bioorganic & medicinal chemistry letters (01.01.2006)
Published in Bioorganic & medicinal chemistry letters (01.01.2006)
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Journal Article
4-Fluorosulfonylpiperidines: Selective 5-HT 2A ligands for the treatment of insomnia
Fish, L. Rebecca, Gilligan, Myra T., Humphries, Alexander C., Ivarsson, Magnus, Ladduwahetty, Tammy, Merchant, Kevin J., O’Connor, Desmond, Patel, Smita, Philipps, Elisabeth, Vargas, Hugo M., Hutson, Peter H., MacLeod, Angus M.
Published in Bioorganic & medicinal chemistry letters (2005)
Published in Bioorganic & medicinal chemistry letters (2005)
Get full text
Journal Article
4-Fluorosulfonylpiperidines : Selective 5-HT2A ligands for the treatment of insomnia: G-protein-coupled receptors in drug discovery
FISH, L. Rebecca, GILLIGAN, Myra T, HUTSON, Peter H, MACLEOD, Angus M, HUMPHRIES, Alexander C, IVARSSON, Magnus, LADDUWAHETTY, Tammy, MERCHANT, Kevin J, O'CONNOR, Desmond, PATEL, Smita, PHILIPPS, Elisabeth, VARGAS, Hugo M
Published in Bioorganic & medicinal chemistry letters (2005)
Get full text
Published in Bioorganic & medicinal chemistry letters (2005)
Journal Article