Antagonists of the human adenosine A2A receptor. Part 3 Design and synthesis of pyrazolo[3,4-d]pyrimidines, pyrrolo[2,3-d]pyrimidines and 6-arylpurines
GILLESPIE, Roger J, CLIFFE, Ian A, ROLFEY, Jonathan, STRATTON, Gemma C, UPTON, Rebecca, WEISS, Scott M, WILLIAMSON, Douglas S, DAWSON, Claire E, DOURISH, Colin T, GAUR, Suneel, JORDAN, Allan M, KNIGHT, Antony R, LERPINIERE, Joanne, MISRA, Anil, PRATT, Robert M
Published in Bioorganic & medicinal chemistry letters (01.05.2008)
Published in Bioorganic & medicinal chemistry letters (01.05.2008)
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Antagonists of the Human A2A Adenosine Receptor. 4. Design, Synthesis, and Preclinical Evaluation of 7-Aryltriazolo[4,5-d]pyrimidines
Gillespie, Roger J, Bamford, Samantha J, Botting, Ruth, Comer, Mike, Denny, Sarah, Gaur, Suneel, Griffin, Michael, Jordan, Allan M, Knight, Anthony R, Lerpiniere, Joanne, Leonardi, Stefania, Lightowler, Sean, McAteer, Steven, Merrett, Angela, Misra, Anil, Padfield, Antony, Reece, Mark, Saadi, Mona, Selwood, Daniel L, Stratton, Gemma C, Surry, Dominic, Todd, Richard, Tong, Xin, Ruston, Vicki, Upton, Rebecca, Weiss, Scott M
Published in Journal of medicinal chemistry (08.01.2009)
Published in Journal of medicinal chemistry (08.01.2009)
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Antagonists of the Human A(2A) Adenosine Receptor. 4. Design, Synthesis, and Preclinical Evaluation of 7-Aryltriazolo[4,5-d]pyrimidines
Gillespie, Roger J., Bamford, Samantha J., Botting, Ruth, Comer, Mike, Denny, Sarah, Gaur, Suneel, Griffin, Michael, Jordan, Allan M., Knight, Anthony R., Lerpiniere, Joanne, Leonardi, Stefania, Lightowler, Sean, McAteer, Steven, Merrett, Angela, Misra, Anil, Padfield, Antony, Reece, Mark, Saadi, Mona, Selwood, Daniel L., Stratton, Gemma C., Surry, Dominic, Todd, Richard, Tong, Xin, Ruston, Vicki, Upton, Rebecca, Weiss, Scott M.
Published in Journal of medicinal chemistry (08.01.2009)
Published in Journal of medicinal chemistry (08.01.2009)
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Antagonists of the human A2A receptor. Part 5: Highly bio-available pyrimidine-4-carboxamides
GILLESPIE, Roger J, BAMFORD, Samantha J, GAUR, Suneel, JORDAN, Allan M, LERPINIERE, Joanne, MANSELL, Howard L, STRATTON, Gemma C
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
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Journal Article
Antagonists of the human A(2A) receptor. Part 5: Highly bio-available pyrimidine-4-carboxamides
Gillespie, Roger J, Bamford, Samantha J, Gaur, Suneel, Jordan, Allan M, Lerpiniere, Joanne, Mansell, Howard L, Stratton, Gemma C
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
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Antagonists of the human A2A receptor. Part 6: Further optimization of pyrimidine-4-carboxamides
GILLESPIE, Roger J, BAMFORD, Samantha J, MANSELL, Howard L, NG, Sean, SAADI, Mona, SIMMONITE, Heather, STRATTON, Gemma C, TODD, Richard S, WILLIAMSON, Douglas S, YULE, Ian A, CLAY, Alex, GAUR, Suneel, HAYMES, Tim, JACKSON, Philip S, JORDAN, Allan M, KLENKE, Burlchard, LEONARDI, Stefania, LIU, Jeanette
Published in Bioorganic & medicinal chemistry (15.09.2009)
Published in Bioorganic & medicinal chemistry (15.09.2009)
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Antagonists of the human A(2A) receptor. Part 6: Further optimization of pyrimidine-4-carboxamides
Gillespie, Roger J, Bamford, Samantha J, Clay, Alex, Gaur, Suneel, Haymes, Tim, Jackson, Philip S, Jordan, Allan M, Klenke, Burkhard, Leonardi, Stefania, Liu, Jeanette, Mansell, Howard L, Ng, Sean, Saadi, Mona, Simmonite, Heather, Stratton, Gemma C, Todd, Richard S, Williamson, Douglas S, Yule, Ian A
Published in Bioorganic & medicinal chemistry (15.09.2009)
Published in Bioorganic & medicinal chemistry (15.09.2009)
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Antagonists of the human adenosine A2A receptor. Part 1 Discovery and synthesis of thieno[3,2-d]pyrimidine-4-methanone derivatives
GILLESPIE, Roger J, ADAMS, David R, JORDAN, Allan M, KNIGHT, Antony R, KNUTSEN, Lars J. S, LAWRENCE, Anthony, LERPINIERE, Joanne, MISRA, Anil, PORTER, Richard H. P, PRATT, Robert M, SHEPHERD, Robin, UPTON, Rebecca, BEBBINGTON, David, WARD, Simon E, WEISS, Scott M, WILLIAMSON, Douglas S, BENWELL, Karen, CLIFFE, Ian A, DAWSON, Claire E, DOURISH, Colin T, FLETCHER, Allan, GAUR, Suneel, GILES, Paul R
Published in Bioorganic & medicinal chemistry letters (01.05.2008)
Published in Bioorganic & medicinal chemistry letters (01.05.2008)
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Antagonists of the human adenosine A2A receptor. Part 2 Design and synthesis of 4-arylthieno[3,2-d]pyrimidine derivatives
GILLESPIE, Roger J, CLIFFE, Ian A, MISRA, Anil, PRATT, Robert M, TODD, Richard S, UPTON, Rebecca, WEISS, Scott M, WILLIAMSON, Douglas S, DAWSON, Claire E, DOURISH, Colin T, GAUR, Suneel, GILES, Paul R, JORDAN, Allan M, KNIGHT, Antony R, LAWRENCE, Anthony, LERPINIERE, Joanne
Published in Bioorganic & medicinal chemistry letters (01.05.2008)
Published in Bioorganic & medicinal chemistry letters (01.05.2008)
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Journal Article
Identification of non-furan containing A2A antagonists using database mining and molecular similarity approaches
RICHARDSON, Christine M, GILLESPIE, Roger J, WILLIAMSON, Douglas S, JORDAN, Allan M, FINK, Alexandra, KNIGHT, Antony R, SELLWOOD, Daniel M, MISRA, Anil
Published in Bioorganic & medicinal chemistry letters (01.12.2006)
Published in Bioorganic & medicinal chemistry letters (01.12.2006)
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Total syntheses of close analogues of the immunosuppressant FK506
Batchelor, Mark J, Gillespie, Roger J, Golec, Julian MC, Hedgecock, Charles JR, Jones, Stuart D, Murdoch, Robert
Published in Tetrahedron (17.01.1994)
Published in Tetrahedron (17.01.1994)
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PROCESS FOR THE PREPARATION OF BENZOTHIO PYRANO-PYRIDINONES
AGER IAN R, ROWLANDS DAVID A, GILLESPIE ROGER J, JEWERY STEPHEN C, GARDENER COLIN R
Year of Publication 20.09.1990
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Year of Publication 20.09.1990
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Antagonists of the human A 2A receptor. Part 5: Highly bio-available pyrimidine-4-carboxamides
Gillespie, Roger J., Bamford, Samantha J., Gaur, Suneel, Jordan, Allan M., Lerpiniere, Joanne, Mansell, Howard L., Stratton, Gemma C.
Published in Bioorganic & medicinal chemistry letters (2009)
Published in Bioorganic & medicinal chemistry letters (2009)
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Antagonists of the human A sub(2A) receptor. Part 6: Further optimization of pyrimidine-4-carboxamides
Gillespie, Roger J, Bamford, Samantha J, Clay, Alex, Gaur, Suneel, Haymes, Tim, Jackson, Philip S, Jordan, Allan M, Klenke, Burkhard, Leonardi, Stefania, Liu, Jeanette, Mansell, Howard L, Ng, Sean, Saadi, Mona, Simmonite, Heather, Stratton, Gemma C, Todd, Richard S, Williamson, Douglas S, Yule, Ian A
Published in Bioorganic & medicinal chemistry (01.09.2009)
Published in Bioorganic & medicinal chemistry (01.09.2009)
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Journal Article
Antagonists of the Human A 2A Adenosine Receptor. 4. Design, Synthesis, and Preclinical Evaluation of 7-Aryltriazolo[4,5- d ]pyrimidines
Gillespie, Roger J., Bamford, Samantha J., Botting, Ruth, Comer, Mike, Denny, Sarah, Gaur, Suneel, Griffin, Michael, Jordan, Allan M., Knight, Anthony R., Lerpiniere, Joanne, Leonardi, Stefania, Lightowler, Sean, McAteer, Steven, Merrett, Angela, Misra, Anil, Padfield, Antony, Reece, Mark, Saadi, Mona, Selwood, Daniel L., Stratton, Gemma C., Surry, Dominic, Todd, Richard, Tong, Xin, Ruston, Vicki, Upton, Rebecca, Weiss, Scott M.
Published in Journal of medicinal chemistry (08.01.2009)
Published in Journal of medicinal chemistry (08.01.2009)
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Journal Article
Antagonists of the human A 2A receptor. Part 6: Further optimization of pyrimidine-4-carboxamides
Gillespie, Roger J., Bamford, Samantha J., Clay, Alex, Gaur, Suneel, Haymes, Tim, Jackson, Philip S., Jordan, Allan M., Klenke, Burkhard, Leonardi, Stefania, Liu, Jeanette, Mansell, Howard L., Ng, Sean, Saadi, Mona, Simmonite, Heather, Stratton, Gemma C., Todd, Richard S., Williamson, Douglas S., Yule, Ian A.
Published in Bioorganic & medicinal chemistry (2009)
Published in Bioorganic & medicinal chemistry (2009)
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Journal Article
Antagonists of the human adenosine A 2A receptor. Part 3: Design and synthesis of pyrazolo[3,4- d]pyrimidines, pyrrolo[2,3- d]pyrimidines and 6-arylpurines
Gillespie, Roger J., Cliffe, Ian A., Dawson, Claire E., Dourish, Colin T., Gaur, Suneel, Jordan, Allan M., Knight, Antony R., Lerpiniere, Joanne, Misra, Anil, Pratt, Robert M., Roffey, Jonathan, Stratton, Gemma C., Upton, Rebecca, Weiss, Scott M., Williamson, Douglas S.
Published in Bioorganic & medicinal chemistry letters (2008)
Published in Bioorganic & medicinal chemistry letters (2008)
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