Benzothiazolyl and Benzoxazolyl Hydrazones Function as Zinc Metallochaperones to Reactivate Mutant p53
Gilleran, John A, Yu, Xin, Blayney, Alan J, Bencivenga, Anthony F, Na, Bing, Augeri, David J, Blanden, Adam R, Kimball, S. David, Loh, Stewart N, Roberge, Jacques Y, Carpizo, Darren R
Published in Journal of medicinal chemistry (25.02.2021)
Published in Journal of medicinal chemistry (25.02.2021)
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Correction to “Structure–Activity Relationship of a Pyrrole Based Series of PfPKG Inhibitors as Anti-Malarials”
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Published in Journal of medicinal chemistry (25.07.2024)
Published in Journal of medicinal chemistry (25.07.2024)
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Journal Article
Structure–Activity Relationship of a Pyrrole Based Series of PfPKG Inhibitors as Anti-Malarials
Gilleran, John A., Ashraf, Kutub, Delvillar, Melvin, Eck, Tyler, Fondekar, Raheel, Miller, Edward B., Hutchinson, Ashley, Dong, Aiping, Seitova, Alma, De Souza, Mariana Laureano, Augeri, David, Halabelian, Levon, Siekierka, John, Rotella, David P., Gordon, John, Childers, Wayne E., Grier, Mark C., Staker, Bart L., Roberge, Jacques Y., Bhanot, Purnima
Published in Journal of medicinal chemistry (14.03.2024)
Published in Journal of medicinal chemistry (14.03.2024)
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Synthetic metallochaperone ZMC1 rescues mutant p53 conformation by transporting zinc into cells as an ionophore
Blanden, Adam R, Yu, Xin, Wolfe, Aaron J, Gilleran, John A, Augeri, David J, O'Dell, Ryan S, Olson, Eric C, Kimball, S David, Emge, Thomas J, Movileanu, Liviu, Carpizo, Darren R, Loh, Stewart N
Published in Molecular pharmacology (01.05.2015)
Published in Molecular pharmacology (01.05.2015)
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Acylpyrazoline-Based Third-Generation Selective Antichlamydial Compounds with Enhanced Potency
Lu, Bin, Qiao, Qi, Park, Elizabeth R., Wang, Yuxuan, Gilleran, John A., Pan, Matthew, Pilch, Daniel S., Wu, Xiang, Roberge, Jacques Y., Fan, Huizhou
Published in ACS omega (21.02.2023)
Published in ACS omega (21.02.2023)
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Synthesis and Characterization of Novel BMI1 Inhibitors Targeting Cellular Self-Renewal in Hepatocellular Carcinoma
Bartucci, Monica, Hussein, Mohamed S., Huselid, Eric, Flaherty, Kathleen, Patrizii, Michele, Laddha, Saurabh V., Kui, Cindy, Bigos, Rachel A., Gilleran, John A., El Ansary, Mervat M. S., Awad, Mona A. M., Kimball, S. David, Augeri, David J., Sabaawy, Hatem E.
Published in Targeted oncology (01.08.2017)
Published in Targeted oncology (01.08.2017)
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CARBONIC ANHYDRASE ENZYME INHIBITORS AND METHODS OF USE THEREOF
SIRACUSA, Mark C, ROBERGE, Jacques Y, PIWINSKI, John, GILLERAN, John A
Year of Publication 18.07.2024
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Year of Publication 18.07.2024
Patent
CARBONIC ANHYDRASE ENZYME INHIBITORS AND METHODS OF USE THEREOF
SIRACUSA, Mark C, ROBERGE, Jacques Y, PIWINSKI, John, GILLERAN, John A
Year of Publication 13.06.2024
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Year of Publication 13.06.2024
Patent