Mechanism-Based Target Identification and Drug Discovery in Cancer Research
Gibbs, Jackson B.
Published in Science (American Association for the Advancement of Science) (17.03.2000)
Published in Science (American Association for the Advancement of Science) (17.03.2000)
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Journal Article
Sequence dependence of protein isoprenylation
MOORES, S. L, SCHABER, M. D, MOSSER, S. D, RANDS, E, O'HARA, M. B, GARSKY, V. M, MARSHALL, M. S, POMPLIANO, D. L, GIBBS, J. B
Published in The Journal of biological chemistry (05.08.1991)
Published in The Journal of biological chemistry (05.08.1991)
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Journal Article
Kinase-deficient Pak1 mutants inhibit Ras transformation of Rat-1 fibroblasts
Tang, Yi, Chen, Zunxuan, Ambrose, Diane, Liu, Jianhua, Gibbs, Jackson B., Chernoff, Jonathan, Field, Jeffrey
Published in Molecular and Cellular Biology (01.08.1997)
Published in Molecular and Cellular Biology (01.08.1997)
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Journal Article
Selective Inhibition of ras-Dependent Transformation by a Farnesyltransferase Inhibitor
Kohl, Nancy E., Mosser, Scott D., deSolms, S. Jane, Giuliani, Elizabeth A., Pompliano, David L., Graham, Samuel L., Smith, Robert L., Scolnick, Edward M., Oliff, Allen, Gibbs, Jackson B.
Published in Science (American Association for the Advancement of Science) (25.06.1993)
Published in Science (American Association for the Advancement of Science) (25.06.1993)
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Journal Article
Antitumor effect of a farnesyl protein transferase inhibitor in mammary and lymphoid tumors overexpressing N-ras in transgenic mice
MANGUES, R, CORRAL, T, KOHL, N. E, SYMMANS, W. F, SUYING LU, MALUMBRES, M, GIBBS, J. B, OLIFF, A, PELLICER, A
Published in Cancer research (Chicago, Ill.) (15.03.1998)
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Published in Cancer research (Chicago, Ill.) (15.03.1998)
Journal Article
Selective inhibition of farnesyl-protein transferase blocks ras processing in vivo
GIBBS, J. B, POMPLIANO, D. L, MOSSER, S. D, RANDS, E, LINGHAM, R. B, SHEO BUX SINGH, SCOLNICK, E. M, KOHL, N. E, OLIFF, A
Published in The Journal of biological chemistry (15.04.1993)
Published in The Journal of biological chemistry (15.04.1993)
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Journal Article
In vitro and In vivo effects of a farnesyltransferase inhibitor on Nf1-deficient hematopoietic cells
MAHGOUB, N, TAYLOR, B. R, GRATIOT, M, KOHL, N. E, GIBBS, J. B, JACKS, T, SHANNON, K. M
Published in Blood (01.10.1999)
Published in Blood (01.10.1999)
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Journal Article
Farnesyltransferase inhibition causes morphological reversion of ras-transformed cells by a complex mechanism that involves regulation of the actin cytoskeleton
Prendergast, G C, Davide, J P, deSolms, S J, Giuliani, E A, Graham, S L, Gibbs, J B, Oliff, A, Kohl, N E
Published in Molecular and Cellular Biology (01.06.1994)
Published in Molecular and Cellular Biology (01.06.1994)
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Journal Article
cDNA cloning and expression of rat and human protein geranylgeranyltransferase type-I
ZHANG, F. L, DIEHL, R. E, KOHL, N. E, GIBBS, J. B, GIROS, B, CASEY, P. J, OMER, C. A
Published in The Journal of biological chemistry (04.02.1994)
Published in The Journal of biological chemistry (04.02.1994)
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Journal Article
Farnesyltransferase inhibitors potentiate the antitumor effect of radiation on a human tumor xenograft expressing activated HRAS
Cohen-Jonathan, E, Muschel, R J, Gillies McKenna, W, Evans, S M, Cerniglia, G, Mick, R, Kusewitt, D, Sebti, S M, Hamilton, A D, Oliff, A, Kohl, N, Gibbs, J B, Bernhard, E J
Published in Radiation research (01.08.2000)
Published in Radiation research (01.08.2000)
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Journal Article
PDGF induction of tyrosine phosphorylation of GTPase activating protein
Molloy, C J, Bottaro, D P, Fleming, T P, Marshall, M S, Gibbs, J B, Aaronson, S A
Published in Nature (London) (07.12.1989)
Published in Nature (London) (07.12.1989)
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Journal Article
Steady-state kinetic mechanism of ras farnesyl:protein transferase
Pompliano, David L, Rands, Elaine, Schaber, Michael D, Mosser, Scott D, Anthony, Neville J, Gibbs, Jackson B
Published in Biochemistry (Easton) (21.04.1992)
Published in Biochemistry (Easton) (21.04.1992)
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Journal Article
Imidazole-containing diarylether and diarylsulfone inhibitors of farnesyl-protein transferase
Dinsmore, Christopher J., Williams, Theresa M., O'Neill, Timothy J., Liu, Dongming, Rands, Elaine, Culberson, J.Christopher, Lobell, Robert B., Koblan, Kenneth S., Kohl, Nancy E., Gibbs, Jackson B., Oliff, Allen I., Graham, Samuel L., Hartman, George D.
Published in Bioorganic & medicinal chemistry letters (06.12.1999)
Published in Bioorganic & medicinal chemistry letters (06.12.1999)
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Journal Article
Purification of ras GTPase activating protein from bovine brain
Gibbs, J.B, Schaber, M.D, Allard, W.J, Sigal, I.S, Scolnick, E.M
Published in Proceedings of the National Academy of Sciences - PNAS (01.07.1988)
Published in Proceedings of the National Academy of Sciences - PNAS (01.07.1988)
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