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Published in Bioorganic & medicinal chemistry letters (01.05.2011)
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Pyrimido[4,5- d]azepines as potent and selective 5-HT 2C receptor agonists: Design, synthesis, and evaluation of PF-3246799 as a treatment for urinary incontinence
Andrews, Mark D., Fish, Paul V., Blagg, Julian, Brabham, Tiffini K., Brennan, Paul E., Bridgeland, Alison, Brown, Alan D., Bungay, Peter J., Conlon, Kelly M., Edmunds, Nicholas J., af Forselles, Kerry, Gibbons, Colleen P., Green, Martin P., Hanton, Giles, Holbrook, Mark, Jessiman, Alan S., McIntosh, Karin, McMurray, Gordon, Nichols, Carly L., Root, James A., Storer, R. Ian, Sutton, Michael R., Ward, Robin V., Westbrook, Dominique, Whitlock, Gavin A.
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