A multicomponent pharmacophore fragment-decoration approach to identify selective LRRK2-targeting probes
Tassini, Sabrina, Castagnolo, Daniele, Scalacci, Nicolo, Kissova, Miroslava, Armijos-Rivera, Jorge I., Giagnorio, Federica, Maga, Giovanni, Costantino, Gabriele, Crespan, Emmanuele, Radi, Marco
Published in MedChemComm (16.03.2016)
Published in MedChemComm (16.03.2016)
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Journal Article
A multicomponent pharmacophore fragment-decoration approach to identify selective LRRK2-targeting probesThe authors declare no competing interest.Electronic supplementary information (ESI) available: Experimental procedures and analytical data for compounds 9 and 10, in vitro LRRK2 inhibition assays, inhibition mechanism and kinase panel data. See DOI: 10.1039/c5md00462d
Tassini, Sabrina, Castagnolo, Daniele, Scalacci, Nicolò, Kissova, Miroslava, Armijos-Rivera, Jorge I, Giagnorio, Federica, Maga, Giovanni, Costantino, Gabriele, Crespan, Emmanuele, Radi, Marco
Year of Publication 16.03.2016
Year of Publication 16.03.2016
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Journal Article