Selectivity of Kinase Inhibitor Fragments
Bamborough, Paul, Brown, Murray J, Christopher, John A, Chung, Chun-wa, Mellor, Geoff W
Published in Journal of medicinal chemistry (28.07.2011)
Published in Journal of medicinal chemistry (28.07.2011)
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4-Phenyl-7-azaindoles as potent and selective IKK2 inhibitors
Liddle, John, Bamborough, Paul, Barker, Michael D., Campos, Sebastien, Cousins, Rick P.C., Cutler, Geoffrey J., Hobbs, Heather, Holmes, Duncan S., Ioannou, Chris, Mellor, Geoff W., Morse, Mary A., Payne, Jeremy J., Pritchard, John M., Smith, Kathryn J., Tape, Daniel T., Whitworth, Caroline, Williamson, Richard A.
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
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Site Distribution in Resin Beads as Determined by Confocal Raman Spectroscopy
Kress, Jürgen, Rose, Abigail, Frey, Jeremy G., Brocklesby, William S., Ladlow, Mark, Mellor, Geoff W., Bradley, Mark
Published in Chemistry : a European journal (17.09.2001)
Published in Chemistry : a European journal (17.09.2001)
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Attenuation of Murine Collagen-Induced Arthritis by a Novel, Potent, Selective Small Molecule Inhibitor of IκB Kinase 2, TPCA-1 (2-[(Aminocarbonyl)amino]-5-(4-fluorophenyl)-3-thiophenecarboxamide), Occurs via Reduction of Proinflammatory Cytokines and Antigen-Induced T Cell Proliferation
Podolin, Patricia L., Callahan, James F., Bolognese, Brian J., Li, Yue H., Carlson, Karey, Davis, T. Gregg, Mellor, Geoff W., Evans, Christopher, Roshak, Amy K.
Published in The Journal of pharmacology and experimental therapeutics (01.01.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.01.2005)
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Attenuation of murine collagen-induced arthritis by a novel, potent, selective small molecule inhibitor of IkappaB Kinase 2, TPCA-1 (2-[(aminocarbonyl)amino]-5-(4-fluorophenyl)-3-thiophenecarboxamide), occurs via reduction of proinflammatory cytokines and antigen-induced T cell Proliferation
Podolin, Patricia L, Callahan, James F, Bolognese, Brian J, Li, Yue H, Carlson, Karey, Davis, T Gregg, Mellor, Geoff W, Evans, Christopher, Roshak, Amy K
Published in The Journal of pharmacology and experimental therapeutics (01.01.2005)
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Published in The Journal of pharmacology and experimental therapeutics (01.01.2005)
Journal Article
Attenuation of Murine Collagen-Induced Arthritis by a Novel, Potent, Selective Small Molecule Inhibitor of IκB Kinase 2, TPCA-1 (2-[(Aminocarbonyl)amino]-5-(4-fluorophenyl)-3-thiophenecarboxamide), Occurs via Reduction of Proinflammatory Cytokines and Antigen-Induced T Cell Proliferation
Patricia L. Podolin, James F. Callahan, Brian J. Bolognese, Yue H. Li, Karey Carlson, T. Gregg Davis, Geoff W. Mellor, Christopher Evans, Amy K. Roshak
Published in The Journal of pharmacology and experimental therapeutics (01.01.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.01.2005)
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Journal Article