Platensimycin is a selective FabF inhibitor with potent antibiotic properties
Colwell, Lawrence, Becker, Joseph W, Parthasarathy, Gopalakrishnan, Tang, Yui S, Basilio, Ángela, Cummings, Richard, Hermes, Jeffery D, Lee, Sang Ho, Dorso, Karen, Motyl, Mary, Soisson, Stephen M, Shoop, Wesley, Genilloud, Olga, Vicente, Francisca, Silver, Lynn L, Singh, Sheo B, Kodali, Srinivas, Jayasuriya, Hiranthi, Bartizal, Ken, Cully, Doris, Barrett, John, Allocco, John, Pelaez, Fernando, Wang, Jun, Young, Katherine, Painter, Ronald, Michael, Bruce, Hernandez, Lorraine, Felcetto, Thomas, Galgoci, Andrew, Gill, Charles, Tormo, José R, Schmatz, Dennis, Zhang, Chaowei, Ondeyka, John, Herath, Kithsiri, Ha, Sookhee
Published in Nature (18.05.2006)
Published in Nature (18.05.2006)
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Journal Article
High-throughput screening platform for natural product-based drug discovery against 3 neglected tropical diseases: human African trypanosomiasis, leishmaniasis, and Chagas disease
Annang, F, Pérez-Moreno, G, García-Hernández, R, Cordon-Obras, C, Martín, J, Tormo, J R, Rodríguez, L, de Pedro, N, Gómez-Pérez, V, Valente, M, Reyes, F, Genilloud, O, Vicente, F, Castanys, S, Ruiz-Pérez, L M, Navarro, M, Gamarro, F, González-Pacanowska, D
Published in Journal of biomolecular screening (01.01.2015)
Published in Journal of biomolecular screening (01.01.2015)
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Journal Article
Novel Biomarkers to Distinguish between Type 3c versus Type 2 Diabetes Mellitus by Untargeted Metabolomics
Caba, O., Jiménez-Luna, C., Martín-Blázquez, A., Diéguez-Castillo, C., Del Palacio J., Pérez, Díaz-Navarro, C., Melguizo, C., Genilloud, O., Vicente-Pérez, F., Prados, J.
Published in Pancreatology : official journal of the International Association of Pancreatology (IAP) ... [et al.] (01.11.2020)
Published in Pancreatology : official journal of the International Association of Pancreatology (IAP) ... [et al.] (01.11.2020)
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Journal Article
Patterns of antimicrobial activities from soil actinomycetes isolated under different conditions of pH and salinity
Basilio, A., González, I., Vicente, M.F., Gorrochategui, J., Cabello, A., González, A., Genilloud, O.
Published in Journal of applied microbiology (01.01.2003)
Published in Journal of applied microbiology (01.01.2003)
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Journal Article
Search for novel cosmeuceutical agents from the Actinobacteria Micromonospora sp
Peyrat, LA, Georgousaki, K, Tsafantakis, N, Gumeni, S, Oves-Costales, D, González, I, Almeida, C, Genilloud, O, Trougakos, IP, Fokialakis, N
Published in Planta Medica International Open (01.10.2017)
Published in Planta Medica International Open (01.10.2017)
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Conference Proceeding
The Complestatins as HIV-1 Integrase Inhibitors. Efficient Isolation, Structure Elucidation, and Inhibitory Activities of Isocomplestatin, Chloropeptin I, New Complestatins, A and B, and Acid-Hydrolysis Products of Chloropeptin I
Singh, Sheo B, Jayasuriya, Hiranthi, Salituro, Gino M, Zink, Deborah L, Shafiee, Ali, Heimbuch, Brian, Silverman, Keith C, Lingham, Russell B, Genilloud, Olga, Teran, Ana, Vilella, Dolores, Felock, Peter, Hazuda, Daria
Published in Journal of natural products (Washington, D.C.) (01.07.2001)
Published in Journal of natural products (Washington, D.C.) (01.07.2001)
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Journal Article
New genus-specific primers for the PCR identification of members of the genus Saccharomonospora and evaluation of the microbial diversity of wild-type isolates of Saccharomonospora detected from soil DNAs
Salazar, O, Moron, R, Genilloud, O
Published in International journal of systematic and evolutionary microbiology (01.11.2000)
Published in International journal of systematic and evolutionary microbiology (01.11.2000)
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Journal Article
Inhibitors of farnesylation of Ras from a microbial natural products screening program
VILELLA, D, SANCHEZ, M, LINGHAM, R. B, SINGH, S. B, JAYASURIYA, H, PELAEZ, F, PLATAS, G, SALAZAR, O, GENILLOUD, O, ROYO, I, CASCALES, C, MARTIN, I, DIEZ, T, SILVERMAN, K. C
Published in Journal of industrial microbiology & biotechnology (01.12.2000)
Published in Journal of industrial microbiology & biotechnology (01.12.2000)
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Journal Article
1542P Untargeted metabolomics to identify novel biomarkers of pancreatic cancer
Caba, O., Jimenez-Luna, C., Martin-Blazquez, A., Martinez-Galan, J., Perez Del Palacio, J., Melguizo, C., Diaz, C., Dieguez, C., Vicente, F., Genilloud, O., Martin-Ruiz, J.L., Prados, J.
Published in Annals of oncology (01.09.2020)
Published in Annals of oncology (01.09.2020)
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Journal Article
Differential induction of secondary metabolite profiles in endophyte fungi by the addition of epigenetic modifiers
González-Menéndez, V, Serrano, R, Muñoz, F, Reyes, F, Genilloud, O, Tormo, JR
Published in Planta Medica (25.06.2015)
Published in Planta Medica (25.06.2015)
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Conference Proceeding
Isolation, Structure, and Absolute Stereochemistry of Platensimycin, A Broad Spectrum Antibiotic Discovered Using an Antisense Differential Sensitivity Strategy
Singh, Sheo B, Jayasuriya, Hiranthi, Ondeyka, John G, Herath, Kithsiri B, Zhang, Chaowei, Zink, Deborah L, Tsou, Nancy N, Ball, Richard G, Basilio, Angela, Genilloud, Olga, Diez, Maria Teresa, Vicente, Francisca, Pelaez, Fernando, Young, Katherine, Wang, Jun
Published in Journal of the American Chemical Society (13.09.2006)
Published in Journal of the American Chemical Society (13.09.2006)
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Journal Article
Kocurin, the true structure of PM181104, an anti-methicillin-resistant Staphylococcus aureus (MRSA) thiazolyl peptide from the marine-derived bacterium Kocuria palustris
Martín, Jesús, da S Sousa, Thiciana, Crespo, Gloria, Palomo, Sara, González, Ignacio, Tormo, José R, de la Cruz, Mercedes, Anderson, Matthew, Hill, Russell T, Vicente, Francisca, Genilloud, Olga, Reyes, Fernando
Published in Marine drugs (04.02.2013)
Published in Marine drugs (04.02.2013)
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Journal Article
Exploitation of global microbial biodiversity for the discovery of novel cosmeceuticals using LC-HRMS based metabolomics
Almeida, C, González-Menéndez, V, González, I, del Palacio, JP, Reyes, F, Lemonakis, N, Tsafantakis, N, Gikas, E, Fokialakis, N, Genilloud, O
Published in Planta Medica (25.11.2015)
Published in Planta Medica (25.11.2015)
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Conference Proceeding
High throughput screening of microbial biodiversity for the discovery of novel cosmeceutical agents
Georgousaki, K, DePedro, N, Chinchilla, AM, Aliagiannis, N, Vicente, F, de Castro, P, Fotinos, S, Genilloud, O, Fokialakis, N
Published in Planta Medica (25.11.2015)
Published in Planta Medica (25.11.2015)
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Conference Proceeding