Search Results - "Genadiy KALAYANOV" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Design and synthesis of HIV-1 protease inhibitors for a long-acting injectable drug application

Design and synthesis of HIV-1 protease inhibitors for a long-acting injectable drug application

by Kesteleyn, Bart, Amssoms, Katie, Schepens, Wim, Hache, Geerwin, Verschueren, Wim, Van De Vreken, Wim, Rombauts, Klara, Meurs, Greet, Sterkens, Patrick, Stoops, Bart, Baert, Lieven, Austin, Nigel, Wegner, Jörg, Masungi, Chantal, Dierynck, Inge, Lundgren, Stina, Jönsson, Daniel, Parkes, Kevin, Kalayanov, Genadiy, Wallberg, Hans, Rosenquist, Åsa, Samuelsson, Bertil, Van Emelen, Kristof, Thuring, Jan Willem
Published in Bioorganic & medicinal chemistry letters (01.01.2013)

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Journal Article

Discovery of β-d-2′-deoxy-2′-dichlorouridine nucleotide prodrugs as potent inhibitors of hepatitis C virus replication

Discovery of β-d-2′-deoxy-2′-dichlorouridine nucleotide prodrugs as potent inhibitors of hepatitis C virus replication

by Pinho, Pedro, Kalayanov, Genadiy, Westerlind, Hans, Rosenquist, Åsa, Wähling, Horst, Sund, Christian, Almeida, Maria, Ayesa, Susana, Tejbrant, Jan, Targett-Adams, Paul, Eneroth, Anders, Lindqvist, Annelie
Published in Bioorganic & medicinal chemistry letters (01.08.2017)

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The Design, Synthesis, and Antiviral Activity of Monofluoro and Difluoro Analogues of 4′-Azidocytidine against Hepatitis C Virus Replication: The Discovery of 4′-Azido-2′-deoxy-2′-fluorocytidine and 4′-Azido-2′-dideoxy-2′,2′-difluorocytidine

The Design, Synthesis, and Antiviral Activity of Monofluoro and Difluoro Analogues of 4′-Azidocytidine against Hepatitis C Virus Replication: The Discovery of 4′-Azido-2′-deoxy-2′-fluorocytidine and 4′-Azido-2′-dideoxy-2′,2′-difluorocytidine

by Smith, David B, Kalayanov, Genadiy, Sund, Christian, Winqvist, Anna, Maltseva, Tatiana, Leveque, Vincent J.-P, Rajyaguru, Sonal, Pogam, Sophie Le, Najera, Isabel, Benkestock, Kurt, Zhou, Xiao-Xiong, Kaiser, Ann C, Maag, Hans, Cammack, Nick, Martin, Joseph A, Swallow, Steven, Johansson, Nils Gunnar, Klumpp, Klaus, Smith, Mark
Published in Journal of medicinal chemistry (14.05.2009)

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Synthesis of pyrazolo[4,3-c]quinoline-5-oxide by reductive cyclization of 4-acetyl-5-(2-nitrophenyl)pyrazole: Revision of the reported structures

Synthesis of pyrazolo[4,3-c]quinoline-5-oxide by reductive cyclization of 4-acetyl-5-(2-nitrophenyl)pyrazole: Revision of the reported structures

by Kalayanov, GD, Choi, JK
Published in Heterocycles (1998)

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2′-Deoxy-4′-azido Nucleoside Analogs Are Highly Potent Inhibitors of Hepatitis C Virus Replication Despite the Lack of 2′-α-Hydroxyl Groups

2′-Deoxy-4′-azido Nucleoside Analogs Are Highly Potent Inhibitors of Hepatitis C Virus Replication Despite the Lack of 2′-α-Hydroxyl Groups

by Klumpp, Klaus, Kalayanov, Genadiy, Ma, Han, Le Pogam, Sophie, Leveque, Vincent, Jiang, Wen-Rong, Inocencio, Nicole, De Witte, Anniek, Rajyaguru, Sonal, Tai, Ezra, Chanda, Sushmita, Irwin, Michael R., Sund, Christian, Winqist, Anna, Maltseva, Tatiana, Eriksson, Staffan, Usova, Elena, Smith, Mark, Alker, Andre, Najera, Isabel, Cammack, Nick, Martin, Joseph A., Johansson, Nils Gunnar, Smith, David B.
Published in The Journal of biological chemistry (25.01.2008)

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The Design, Synthesis, and Antiviral Activity of 4′-Azidocytidine Analogues against Hepatitis C Virus Replication: The Discovery of 4′-Azidoarabinocytidine

The Design, Synthesis, and Antiviral Activity of 4′-Azidocytidine Analogues against Hepatitis C Virus Replication: The Discovery of 4′-Azidoarabinocytidine

by Smith, David B, Kalayanov, Genadiy, Sund, Christian, Winqvist, Anna, Pinho, Pedro, Maltseva, Tatiana, Morisson, Veronique, Leveque, Vincent, Rajyaguru, Sonal, Pogam, Sophie Le, Najera, Isabel, Benkestock, Kurt, Zhou, Xiao-Xiong, Maag, Hans, Cammack, Nick, Martin, Joseph A, Swallow, Steven, Johansson, Nils Gunnar, Klumpp, Klaus, Smith, Mark
Published in Journal of medicinal chemistry (08.01.2009)

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Nicotine hapten structure, antibody selectivity and effect relationships: Results from a nicotine vaccine screening procedure

Nicotine hapten structure, antibody selectivity and effect relationships: Results from a nicotine vaccine screening procedure

by de Villiers, Sabina H.L, Lindblom, Nina, Kalayanov, Genadiy, Gordon, Sandra, Baraznenok, Ivan, Malmerfelt, Anna, Marcus, Monica M, Johansson, Anette M, Svensson, Torgny H
Published in Vaccine (02.03.2010)

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Design and synthesis of potent hydroxyethylamine (HEA) BACE-1 inhibitors carrying prime side 4,5,6,7-tetrahydrobenzazole and 4,5,6,7-tetrahydropyridinoazole templates

Design and synthesis of potent hydroxyethylamine (HEA) BACE-1 inhibitors carrying prime side 4,5,6,7-tetrahydrobenzazole and 4,5,6,7-tetrahydropyridinoazole templates

by Sund, Christian, Belda, Oscar, Borkakoti, Neera, Lindberg, Jimmy, Derbyshire, Dean, Vrang, Lotta, Hamelink, Elizabeth, Åhgren, Cathrine, Woestenenk, Esmeralda, Wikström, Kristina, Eneroth, Anders, Lindström, Erik, Kalayanov, Genadiy
Published in Bioorganic & medicinal chemistry letters (01.11.2012)

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Discovery of 4′-azido-2′-deoxy-2′-C-methyl cytidine and prodrugs thereof: A potent inhibitor of Hepatitis C virus replication

Discovery of 4′-azido-2′-deoxy-2′-C-methyl cytidine and prodrugs thereof: A potent inhibitor of Hepatitis C virus replication

by Nilsson, Magnus, Kalayanov, Genadiy, Winqvist, Anna, Pinho, Pedro, Sund, Christian, Zhou, Xiao-Xiong, Wähling, Horst, Belfrage, Anna-Karin, Pelcman, Michael, Agback, Tatiana, Benckestock, Kurt, Wikström, Kristina, Boothee, Mirva, Lindqvist, Anneli, Rydegård, Christina, Jonckers, Tim H.M., Vandyck, Koen, Raboisson, Pierre, Lin, Tse-I, Lachau-Durand, Sophie, de Kock, Herman, Smith, David B., Martin, Joseph A., Klumpp, Klaus, Simmen, Kenneth, Vrang, Lotta, Terelius, Ylva, Samuelsson, Bertil, Rosenquist, Åsa, Johansson, Nils Gunnar
Published in Bioorganic & medicinal chemistry letters (01.05.2012)

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Regioselective functionalization of guanine: Simple and practical synthesis of 7-and 9-alkylated guanines starting from guanosine

Regioselective functionalization of guanine: Simple and practical synthesis of 7-and 9-alkylated guanines starting from guanosine

by Kalayanov, G, Jaksa, S, Scarcia, T, Kobe, J
Published in Synthesis (Stuttgart) (19.08.2004)

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2â€²-Deoxy-4â€²-azido Nucleoside Analogs Are Highly Potent Inhibitors of Hepatitis C Virus Replication Despite the Lack of 2â€²-Î±-Hydroxyl Groups

2â²-Deoxy-4â²-azido Nucleoside Analogs Are Highly Potent Inhibitors of Hepatitis C Virus Replication Despite the Lack of 2â²-Î±-Hydroxyl Groups

by Klaus Klumpp, Genadiy Kalayanov, Han Ma, Sophie Le Pogam, Vincent Leveque, Wen-Rong Jiang, Nicole Inocencio, Anniek De Witte, Sonal Rajyaguru, Ezra Tai, Sushmita Chanda, Michael R. Irwin, Christian Sund, Anna Winqist, Tatiana Maltseva, Staffan Eriksson, Elena Usova, Mark Smith, Andre Alker, Isabel Najera, Nick Cammack, Joseph A. Martin, Nils Gunnar Johansson, David B. Smith
Published in The Journal of biological chemistry (25.01.2008)

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Different Incorporation Efficiencies for Nucleotide Analogs During HCV Polymerase RNA Synthesis Initiation and Elongation Phases

Different Incorporation Efficiencies for Nucleotide Analogs During HCV Polymerase RNA Synthesis Initiation and Elongation Phases

by Ma, Han, Inocencio, Nicole, Leveque, Vincent, Kalayanov, Genadiy, Smith, David, Cammack, Nick, Johansson, Nils Gunnar, Klumpp, Klaus
Published in Antiviral research (01.05.2008)

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Journal Article

Active immunisation against nicotine blocks the reward facilitating effects of nicotine and partially prevents nicotine withdrawal in the rat as measured by dopamine output in the nucleus accumbens, brain reward thresholds and somatic signs

Active immunisation against nicotine blocks the reward facilitating effects of nicotine and partially prevents nicotine withdrawal in the rat as measured by dopamine output in the nucleus accumbens, brain reward thresholds and somatic signs

by Lindblom, Nina, de Villiers, Sabina H L, Semenova, Svetlana, Kalayanov, Genadiy, Gordon, Sandra, Schilström, Björn, Johansson, Anette M, Markou, Athina, Svensson, Torgny H
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.11.2005)

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2′-Deoxy-nucleoside Analogs can be Potent Dual Inhibitors of HCV and HIV Replication with Selectivity against Human Polymerases

2′-Deoxy-nucleoside Analogs can be Potent Dual Inhibitors of HCV and HIV Replication with Selectivity against Human Polymerases

by Klumpp, Klaus, Su, Guoping, Leveque, Vincent, Deval, Jerome, Heilek, Gabrielle, Rajyaguru, Sonal, Li, Yu, Hang, Julie Q., Ma, Han, Inocencio, Nicole, Kalayanov, Genadiy, Winqvist, Anna, Smith, David B., Cammack, Nick, Johansson, Nils Gunnar, Najera, Isabel
Published in Antiviral research (01.05.2009)

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Journal Article

HCV POLYMERASE INHIBITORS

HCV POLYMERASE INHIBITORS

by WAHLING, HORST, TORSSELL, STAFFAN, KALAYANOV, GENADIY
Year of Publication 23.09.2020

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Patent

Active immunization against nicotine alters the distribution of nicotine but not the metabolism to cotinine in the rat

Active immunization against nicotine alters the distribution of nicotine but not the metabolism to cotinine in the rat

by de Villiers, Sabina H L, Lindblom, Nina, Kalayanov, Genadiy, Gordon, Sandra, Johansson, Anette M, Svensson, Torgny H
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.10.2004)

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Journal Article

SYNTHESIS OF FLG

SYNTHESIS OF FLG

by KALAYANOV, GENADIY
Year of Publication 30.08.2012

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Patent

HCV POLYMERASE INHIBITORS

HCV POLYMERASE INHIBITORS

by KALAYANOV, Genadiy, WÄHLING, Horst, TORSSELL, Staffan
Year of Publication 22.05.2019

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Patent

HCV polymerase inhibitors

HCV polymerase inhibitors

by Wahling, Horst, Kalayanov, Genadiy, Torssell, Staffan
Year of Publication 09.05.2019

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Patent

HCV POLYMERASE INHIBITORS

HCV POLYMERASE INHIBITORS

by KALAYANOV, Genadiy, WAHLING, Horst, TORSSELL, Staffan
Year of Publication 21.03.2019

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Patent

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