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Gawalska, Alicja, Kołaczkowski, Marcin, Bucki, Adam
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Published in Molecules (Basel, Switzerland) (11.05.2022)
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Advances in Discovery of PDE10A Inhibitors for CNS-Related Disorders. Part 1: Overview of the Chemical and Biological Research
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Published in Current drug targets (01.01.2019)
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The selective 5-HT1A receptor biased agonists, F15599 and F13714, show antidepressant-like properties after a single administration in the mouse model of unpredictable chronic mild stress
Głuch-Lutwin, Monika, Sałaciak, Kinga, Gawalska, Alicja, Jamrozik, Marek, Sniecikowska, Joanna, Newman-Tancredi, Adrian, Kołaczkowski, Marcin, Pytka, Karolina
Published in Psychopharmacology (01.08.2021)
Published in Psychopharmacology (01.08.2021)
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The selective 5-HT.sub.1A receptor biased agonists, F15599 and F13714, show antidepressant-like properties after a single administration in the mouse model of unpredictable chronic mild stress
Gluch-Lutwin, Monika, Salaciak, Kinga, Gawalska, Alicja, Jamrozik, Marek, Sniecikowska, Joanna, Newman-Tancredi, Adrian, Kolaczkowski, Marcin
Published in Psychopharmacology (01.08.2021)
Published in Psychopharmacology (01.08.2021)
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Application of automated machine learning in the identification of multi‐target‐directed ligands blocking PDE4B, PDE8A, and TRPA1 with potential use in the treatment of asthma and COPD
Gawalska, Alicja, Czub, Natalia, Sapa, Michał, Kołaczkowski, Marcin, Bucki, Adam, Mendyk, Aleksander
Published in Molecular informatics (01.07.2023)
Published in Molecular informatics (01.07.2023)
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The 5-HT1A receptor biased agonist, NLX-204, shows rapid-acting antidepressant-like properties and neurochemical changes in two mouse models of depression
Głuch-Lutwin, Monika, Sałaciak, Kinga, Pytka, Karolina, Gawalska, Alicja, Jamrozik, Marek, Śniecikowska, Joanna, Kołaczkowski, Marcin, Depoortère, Ronan Y., Newman-Tancredi, Adrian
Published in Behavioural brain research (13.02.2023)
Published in Behavioural brain research (13.02.2023)
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Novel butanehydrazide derivatives of purine-2,6-dione as dual PDE4/7 inhibitors with potential anti-inflammatory activity: Design, synthesis and biological evaluation
Chłoń-Rzepa, Grażyna, Jankowska, Agnieszka, Ślusarczyk, Marietta, Świerczek, Artur, Pociecha, Krzysztof, Wyska, Elżbieta, Bucki, Adam, Gawalska, Alicja, Kołaczkowski, Marcin, Pawłowski, Maciej
Published in European journal of medicinal chemistry (25.02.2018)
Published in European journal of medicinal chemistry (25.02.2018)
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Hybrid molecules combining GABA-A and serotonin 5-HT6 receptors activity designed to tackle neuroinflammation associated with depression
Marcinkowska, Monika, Mordyl, Barbara, Fajkis-Zajaczkowska, Nikola, Siwek, Agata, Karcz, Tadeusz, Gawalska, Alicja, Bucki, Adam, Żmudzki, Paweł, Partyka, Anna, Jastrzębska-Więsek, Magdalena, Pomierny, Bartosz, Walczak, Maria, Smolik, Magdalena, Pytka, Karolina, Mika, Kamil, Kotańska, Magdalena, Kolaczkowski, Marcin
Published in European journal of medicinal chemistry (05.02.2023)
Published in European journal of medicinal chemistry (05.02.2023)
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Novel anilide and benzylamide derivatives of arylpiperazinylalkanoic acids as 5-HT1A/5-HT7 receptor antagonists and phosphodiesterase 4/7 inhibitors with procognitive and antidepressant activity
Jankowska, Agnieszka, Satała, Grzegorz, Kołaczkowski, Marcin, Bucki, Adam, Głuch-Lutwin, Monika, Świerczek, Artur, Pociecha, Krzysztof, Partyka, Anna, Jastrzębska-Więsek, Magdalena, Lubelska, Annamaria, Latacz, Gniewomir, Gawalska, Alicja, Bojarski, Andrzej J., Wyska, Elżbieta, Chłoń-Rzepa, Grażyna
Published in European journal of medicinal chemistry (01.09.2020)
Published in European journal of medicinal chemistry (01.09.2020)
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New imidazopyridines with phosphodiesterase 4 and 7 inhibitory activity and their efficacy in animal models of inflammatory and autoimmune diseases
Ručilová, Veronika, Świerczek, Artur, Vanda, David, Funk, Petr, Lemrová, Barbora, Gawalska, Alicja, Bucki, Adam, Nowak, Barbara, Zadrożna, Monika, Pociecha, Krzysztof, Soural, Miroslav, Wyska, Elżbieta, Pawłowski, Maciej, Chłoń-Rzepa, Grażyna, Zajdel, Paweł
Published in European journal of medicinal chemistry (01.01.2021)
Published in European journal of medicinal chemistry (01.01.2021)
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Novel amide derivatives of 1,3-dimethyl-2,6-dioxopurin-7-yl-alkylcarboxylic acids as multifunctional TRPA1 antagonists and PDE4/7 inhibitors: A new approach for the treatment of pain
Chłoń-Rzepa, Grażyna, Ślusarczyk, Marietta, Jankowska, Agnieszka, Gawalska, Alicja, Bucki, Adam, Kołaczkowski, Marcin, Świerczek, Artur, Pociecha, Krzysztof, Wyska, Elżbieta, Zygmunt, Małgorzata, Kazek, Grzegorz, Sałat, Kinga, Pawłowski, Maciej
Published in European journal of medicinal chemistry (05.10.2018)
Published in European journal of medicinal chemistry (05.10.2018)
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Dual Molecules Targeting 5-HT 6 and GABA-A Receptors as a New Approach to Combat Depression Associated with Neuroinflammation
Marcinkowska, Monika, Mordyl, Barbara, Siwek, Agata, Głuch-Lutwin, Monika, Karcz, Tadeusz, Gawalska, Alicja, Sapa, Michał, Bucki, Adam, Szafrańska, Katarzyna, Pomierny, Bartosz, Pytka, Karolina, Kotańska, Magdalena, Mika, Kamil, Kolaczkowski, Marcin
Published in ACS chemical neuroscience (04.04.2023)
Published in ACS chemical neuroscience (04.04.2023)
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Dual Molecules Targeting 5‑HT6 and GABA‑A Receptors as a New Approach to Combat Depression Associated with Neuroinflammation
Marcinkowska, Monika, Mordyl, Barbara, Siwek, Agata, Głuch-Lutwin, Monika, Karcz, Tadeusz, Gawalska, Alicja, Sapa, Michał, Bucki, Adam, Szafrańska, Katarzyna, Pomierny, Bartosz, Pytka, Karolina, Kotańska, Magdalena, Mika, Kamil, Kolaczkowski, Marcin
Published in ACS chemical neuroscience (19.04.2023)
Published in ACS chemical neuroscience (19.04.2023)
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Novel pyridine-2,4,6-tricarbohydrazide thiourea compounds as small key organic molecules for the potential treatment of type-2 diabetes mellitus: In vitro studies against yeast - and -glucosidase and in silico molecular modeling
Rehman, Tanzeel Ur, Riaz, Sadaf, Khan, Islam Ullah, Ashraf, Muhammad, Bajda, Marek, Gawalska, Alicja, Yar, Muhammad
Published in Archiv der Pharmazie (Weinheim) (01.01.2018)
Published in Archiv der Pharmazie (Weinheim) (01.01.2018)
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Novel pyridine‐2,4,6‐tricarbohydrazide thiourea compounds as small key organic molecules for the potential treatment of type‐2 diabetes mellitus: In vitro studies against yeast α‐ and β‐glucosidase and in silico molecular modeling
Rehman, Tanzeel Ur, Riaz, Sadaf, Khan, Islam Ullah, Ashraf, Muhammad, Bajda, Marek, Gawalska, Alicja, Yar, Muhammad
Published in Archiv der Pharmazie (Weinheim) (01.01.2018)
Published in Archiv der Pharmazie (Weinheim) (01.01.2018)
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