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1,4-Dihydroindeno[1,2-c]pyrazoles with Acetylenic Side Chains as Novel and Potent Multitargeted Receptor Tyrosine Kinase Inhibitors with Low Affinity for the hERG Ion Channel
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Discovery of + (2 -{4 -[2 -(5,6,7,8 -tetrahydro -1,8 -naphthyridin -2-yl )ethoxy ]phenyl} -cyclopropyl )acetic acid as potent and selective αvβ3 inhibitor : Design, synthesis, and optimization
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Published in Bioorganic & medicinal chemistry (15.05.2007)
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Synthesis of imidazopyridines and purines as potent inhibitors of leukotriene A4 hydrolase
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Published in Bioorganic & medicinal chemistry letters (24.03.2003)
Published in Bioorganic & medicinal chemistry letters (24.03.2003)
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Pyrrolidine and piperidine analogues of SC-57461A as potent, orally active inhibitors of leukotriene A4 hydrolase
PENNING, Thomas D, CHANDRAKUMAR, Nizal S, HARDING, Elizabeth I, HIGHKIN, Maureen K, KACHUR, James F, KIM, Suzanne H, VILLANI-PRICE, Doreen, PYLA, E. Yvonne, GHOREISHI-HAACK, Nayereh S, SMITH, Walter G, DESAI, Bipin N, DJURIC, Stevan W, GASIECKI, Alan F, LIANG, Chi-Dean, MIYASHIRO, Julie M, RUSSELL, Mark A, ASKONAS, Leslie J, GIERSE, James K
Published in Bioorganic & medicinal chemistry letters (01.12.2002)
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5 MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF
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Year of Publication 02.09.2013
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Year of Publication 02.09.2013
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MODULATORS OF 5-HT RECEPTORS AND METHODS OF USE THEREOF
WELCH DENNIE S, ZHAO HONGYU, WILSON NOEL S, BRAJE WILFRIED, RELO ANA LUCIA, THOMPSON CHRISTINA M, TURNER SEAN C, KRUGER ALBERT W, SHEKHAR SHASHANK, LI HUANQIU, ZHANG MIN, GASIECKI ALAN F, AKRITOPOULOU ZANZE IRINI, DJURIC STEVAN W, GANDARILLA JORGE
Year of Publication 12.06.2012
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Year of Publication 12.06.2012
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Synthesis of fused imidazole rings by sequential van Leusen/C–H bond activation
Gracias, Vijaya, Gasiecki, Alan F., Pagano, Thomas G., Djuric, Stevan W.
Published in Tetrahedron letters (11.12.2006)
Published in Tetrahedron letters (11.12.2006)
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Year of Publication 26.03.2010
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Year of Publication 26.03.2010
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An expedient route to diaza-spirocycles utilizing a sequential multicomponent α-aminoallylation/ring-closing metathesis strategy
Gracias, Vijaya, Gasiecki, Alan F., Moore, Joel D., Akritopoulou-Zanze, Irini, Djuric, Stevan W.
Published in Tetrahedron letters (11.12.2006)
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Catalytic functionalization of polymers: a novel approach to site-specific delivery of misoprostol to the stomach
Tremont, Samuel J, Collins, Paul W, Perkins, William E, Fenton, Rick L, Forster, Denis, McGrath, Martin P, Wagner, Grace M, Gasiecki, Alan F, Bianchi, Robert G
Published in Journal of medicinal chemistry (15.10.1993)
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Redox glycosidation: a new strategy for disaccharide synthesis
Barrett, Anthony G. M, Bezuidenhoudt, Barend C. B, Gasiecki, Alan F, Howell, Amy R, Russell, Mark A
Published in Journal of the American Chemical Society (01.02.1989)
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Application of (chloromethyl)aluminum 2-(2-propenyl)anilide in the conversion of .gamma.- and .delta.-lactones into protected hydroxy acids
Barrett, Anthony G. M, Bezuidenhoudt, Barend C. B, Dhanak, Dashyant, Gasiecki, Alan F, Howell, Amy R, Lee, Albert C, Russell, Mark A
Published in Journal of organic chemistry (01.07.1989)
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18-Cycloalkyl analogs of enisoprost
Collins, Paul W, Gasiecki, Alan F, Perkins, William E, Gullikson, Gary W, Jones, Peter H, Bauer, Raymond F
Published in Journal of medicinal chemistry (01.05.1989)
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Conference Proceeding
Synthesis and gastrointestinal pharmacology of a 3E,5Z diene analog of misoprostol
Collins, Paul W, Kramer, Steven W, Gasiecki, Alan F, Weier, Richard M, Jones, Peter H, Gullikson, Gary W, Bianchi, Robert G, Bauer, Raymond F
Published in Journal of medicinal chemistry (01.01.1987)
Published in Journal of medicinal chemistry (01.01.1987)
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