Deactivation of Akt and STAT3 signaling promotes apoptosis, inhibits proliferation, and enhances the sensitivity of hepatocellular carcinoma cells to an anticancer agent, Atiprimod
Choudhari, Sweeta R, Khan, Muhammad A, Harris, Genesis, Picker, Donald, Jacob, Gary S, Block, Timothy, Shailubhai, Kunwar
Published in Molecular cancer therapeutics (01.01.2007)
Published in Molecular cancer therapeutics (01.01.2007)
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A clinically relevant SCID-hu in vivo model of human multiple myeloma
Tassone, Pierfrancesco, Neri, Paola, Carrasco, Daniel R., Burger, Renate, Goldmacher, Victor S., Fram, Robert, Munshi, Vidit, Shammas, Masood A., Catley, Laurence, Jacob, Gary S., Venuta, Salvatore, Anderson, Kenneth C., Munshi, Nikhil C.
Published in Blood (15.07.2005)
Published in Blood (15.07.2005)
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Plecanatide, an Oral Guanylate Cyclase C Agonist Acting Locally in the Gastrointestinal Tract, Is Safe and Well-Tolerated in Single Doses
Shailubhai, Kunwar, Comiskey, Stephen, Foss, John A., Feng, Rong, Barrow, Laura, Comer, Gail M., Jacob, Gary S.
Published in Digestive diseases and sciences (01.09.2013)
Published in Digestive diseases and sciences (01.09.2013)
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Mo1316 Structural and Dynamic Features of Plecanatide: Insights From Molecular Dynamics Simulations
Brancale, Andrea, Shailubhai, Kunwar, Ferla, Salvatore, Ricci, Antonio, Bassetto, Marcella, Jacob, Gary S
Published in Gastroenterology (New York, N.Y. 1943) (01.04.2016)
Published in Gastroenterology (New York, N.Y. 1943) (01.04.2016)
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Therapeutically targeting guanylate cyclase‐C: computational modeling of plecanatide, a uroguanylin analog
Brancale, Andrea, Shailubhai, Kunwar, Ferla, Salvatore, Ricci, Antonio, Bassetto, Marcella, Jacob, Gary S
Published in Pharmacology research & perspectives (01.04.2017)
Published in Pharmacology research & perspectives (01.04.2017)
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967 Plecanatide, Like Uroguanylin, Activates Guanylate Cyclase-C Signaling in a pH-Dependent Manner in T84 Cells, and in Murine Intestinal Epithelial Cells and Tissues
Patwa, Viren, Joshi, Apoorva, Thadi, Anusha, Eddy, E. Priya, Palejwala, Vaseem A, Jacob, Gary S, Shailubhai, Kunwar
Published in Gastroenterology (New York, N.Y. 1943) (01.04.2016)
Published in Gastroenterology (New York, N.Y. 1943) (01.04.2016)
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925g Plecanatide, a Novel Guanylate Cyclase-C (GC-C) Receptor Agonist, is Efficacious and Safe in Patients with Chronic Idiopathic Constipation (CIC): Results from a 951 Patient, 12 Week, Multi-Center Trial
Miner, Philip B, Surowitz, Ron, Fogel, Ron, Koltun, William, Drossman, Douglas A, Camilleri, Michael, Mangel, Allen, Barrow, Laura, Jacob, Gary S, Shailubhai, Kunwar
Published in Gastroenterology (New York, N.Y. 1943) (01.05.2013)
Published in Gastroenterology (New York, N.Y. 1943) (01.05.2013)
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Azaspirane (N-N-diethyl-8,8-dipropyl-2-azaspiro [4.5] decane-2-propanamine) inhibits human multiple myeloma cell growth in the bone marrow milieu in vitro and in vivo
Hamasaki, Makoto, Hideshima, Teru, Tassone, Pierfrancesco, Neri, Paola, Ishitsuka, Kenji, Yasui, Hiroshi, Shiraishi, Norihiko, Raje, Noopur, Kumar, Shaji, Picker, Donald H., Jacob, Gary S., Richardson, Paul G., Munshi, Nikhil C., Anderson, Kenneth C.
Published in Blood (01.06.2005)
Published in Blood (01.06.2005)
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Plecanatide and dolcanatide, novel guanylate cyclase-C agonists, ameliorate gastrointestinal inflammation in experimental models of murine colitis
Shailubhai, Kunwar, Palejwala, Vaseem, Arjunan, Krishna Priya, Saykhedkar, Sayali, Nefsky, Bradley, Foss, John A, Comiskey, Stephen, Jacob, Gary S, Plevy, Scott E
Published in World journal of gastrointestinal pharmacology and therapeutics (06.11.2015)
Published in World journal of gastrointestinal pharmacology and therapeutics (06.11.2015)
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Treatment of chronic hepadnavirus infection in a woodchuck animal model with an inhibitor of protein folding and trafficking
Block, T M, Lu, X, Mehta, A S, Blumberg, B S, Tennant, B, Ebling, M, Korba, B, Lansky, D M, Jacob, G S, Dwek, R A
Published in Nature medicine (01.05.1998)
Published in Nature medicine (01.05.1998)
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Virulence of a phosphoribosylaminoimidazole carboxylase-deficient Candida albicans strain in an immunosuppressed murine model of systemic candidiasis
DONOVAN, Matthew, SCHUMUKE, Jon J, FONZI, William A, BONAR, Sheri L, GHEESLING-MULLIS, Karen, JACOB, Gary S, DAVISSON, Vincent Jo, DOTSON, Stanton B
Published in Infection and immunity (01.04.2001)
Published in Infection and immunity (01.04.2001)
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Inhibition of HIV replication by amino-sugar derivatives
Fleet, George W.J., Karpas, Abraham, Dwek, Raymond A., Fellows, Linda E., Tyms, A.S., Petursson, Sigthor, Namgoong, Sung K., Ramsden, Nigel G., Smith, Paul W., Son, Jong Chan, Wilson, Francis, Witty, David R., Jacob, Gary S., Rademacher, Thomas W.
Published in FEBS letters (12.09.1988)
Published in FEBS letters (12.09.1988)
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Aromatic Cross-Links in Insect Cuticle: Detection by Solid-State $^{13}$C and $^{15}$N NMR
Schaefer, Jacob, Kramer, Karl J., Garbow, Joel R., Jacob, Gary S., Stejskal, Edward O., Hopkins, Theodore L., Speirs, Roy D.
Published in Science (American Association for the Advancement of Science) (06.03.1987)
Published in Science (American Association for the Advancement of Science) (06.03.1987)
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Multivalent sialyl-LeX: potent inhibitors of E-selectin-mediated cell adhesion; reagent for staining activated endothelial cells
Welply, J K, Abbas, S Z, Scudder, P, Keene, J L, Broschat, K, Casnocha, S, Gorka, C, Steininger, C, Howard, S C, Schmuke, J J
Published in Glycobiology (Oxford) (01.06.1994)
Published in Glycobiology (Oxford) (01.06.1994)
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