Rapid hit to lead evaluation of pyrazolo[3,4- d]pyrimidin-4-one as selective and orally bioavailable mGluR1 antagonists
Wang, Xueqing, Kolasa, Teodozyi, El Kouhen, Odile F., Chovan, Linda E., Black-Shaefer, Candace L., Wagenaar, Frank L., Garton, Jennifer A., Moreland, Robert B., Honore, Prisca, Lau, Yau Yi, Dandliker, Peter J., Brioni, Jorge D., Stewart, Andrew O.
Published in Bioorganic & medicinal chemistry letters (01.08.2007)
Published in Bioorganic & medicinal chemistry letters (01.08.2007)
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