Mapping the Melatonin Receptor. 6. Melatonin Agonists and Antagonists Derived from 6H-Isoindolo[2,1-a]indoles, 5,6-Dihydroindolo[2,1-a]isoquinolines, and 6,7-Dihydro-5H-benzo[c]azepino[2,1-a]indoles
Faust, Rüdiger, Garratt, Peter J, Jones, Rob, Yeh, Li-Kuan, Tsotinis, Andrew, Panoussopoulou, Maria, Calogeropoulou, Theodora, Teh, Muy-Teck, Sugden, David
Published in Journal of medicinal chemistry (23.03.2000)
Published in Journal of medicinal chemistry (23.03.2000)
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Mapping the Melatonin Receptor. 8. Selective MT2 Agonists Derived from 5,6‐Dihydroindolo[2,1‐a]isoquinolines and Related Systems
Tsotinis, Andrew, Afroudakis, Pandelis A., Papanastasiou, Ioannis P., Sakellaropoulou, Aikaterini, Boniakou, Marina, Komiotis, Dimitri, Garratt, Peter J., Delagrange, Philippe, Bocianowska‐Zbrog, Alina, Sugden, David
Published in ChemMedChem (20.06.2022)
Published in ChemMedChem (20.06.2022)
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Mapping the Melatonin Receptor. 5. Melatonin Agonists and Antagonists Derived from Tetrahydrocyclopent[b]indoles, Tetrahydrocarbazoles and Hexahydrocyclohept[b]indoles
Davies, David J, Garratt, Peter J, Tocher, Derek A, Vonhoff, Stefan, Davies, John, Teh, Muy-Teck, Sugden, David
Published in Journal of medicinal chemistry (12.02.1998)
Published in Journal of medicinal chemistry (12.02.1998)
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Evidence of the Indirect Formation of the Catecholic Intermediate Substrate Responsible for the Autoactivation Kinetics of Tyrosinase
Cooksey, Christopher J., Garratt, Peter J., Land, Edward J., Pavel, Stan, Ramsden, Christopher A., Riley, Patrick A., Smit, Nico P.M.
Published in The Journal of biological chemistry (17.10.1997)
Published in The Journal of biological chemistry (17.10.1997)
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Mapping the Melatonin Receptor. 7. Subtype Selective Ligands Based on β-Substituted N-Acyl-5-methoxytryptamines and β-Substituted N-Acyl-5-methoxy-1-methyltryptamines
Tsotinis, Andrew, Vlachou, Margarita, Papahatjis, Demetris P, Calogeropoulou, Theodora, Nikas, Spyros P, Garratt, Peter J, Piccio, Vincent, Vonhoff, Stefan, Davidson, Kathryn, Teh, Muy-Teck, Sugden, David
Published in Journal of medicinal chemistry (15.06.2006)
Published in Journal of medicinal chemistry (15.06.2006)
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7-Substituted-melatonin and 7-substituted-1-methylmelatonin analogues: Effect of substituents on potency and binding affinity
Faust, Rüdiger, Garratt, Peter J., Trujillo Pérez, Maria Angeles, Piccio, Vincent J.-D., Madsen, Christian, Stenstrøm, Ane, Frølund, Bente, Davidson, Kathryn, Teh, Muy-Teck, Sugden, David
Published in Bioorganic & medicinal chemistry (01.07.2007)
Published in Bioorganic & medicinal chemistry (01.07.2007)
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Binding affinity and biological activity of oxygen and sulfur isosteres at melatonin receptors as a function of their hydrogen bonding capability
Davies, David J, Faust, Rüdiger, Garratt, Peter J, Marivingt-Mounir, Cécile, Kathryn Davidson, Teh, Muy-Teck, Sugden, David
Published in Bioorganic chemistry (01.02.2004)
Published in Bioorganic chemistry (01.02.2004)
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Molecular design using electrostatic interactions. Part 4: Synthesis and properties of flexible tetrapodand tetracations derived from naphthalene. Role of structured water in the electrostatic binding of polyanion guests: a model for interactions in biological systems
Maria Christofi, A, Garratt, Peter J, Hogarth, Graeme, Ibbett, Ashley J, Ng, Yiu-Fai, Steed, Jonathan W
Published in Tetrahedron (27.05.2002)
Published in Tetrahedron (27.05.2002)
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Melatonin receptor pharmacology: toward subtype specificity
Sugden, David, Pickering, Hannah, Teh, Mui-Teck, Garratt, Peter J
Published in Biology of the cell (01.11.1997)
Published in Biology of the cell (01.11.1997)
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Mapping the Melatonin Receptor. 8. Selective MT2 Agonists Derived from 5,6‐Dihydroindoloisoquinolines and Related Systems
Tsotinis, Andrew, Afroudakis, Pandelis A, Papanastasiou, Ioannis P, Sakellaropoulou, Aikaterini, Boniakou, Marina, Komiotis, Dimitri, Garratt, Peter J, Delagrange, Philippe, Alina Bocianowska‐Zbrog, Sugden, David
Published in ChemMedChem (01.06.2022)
Published in ChemMedChem (01.06.2022)
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Intramolecular anionic cyclization route to capped [3]peristylanes
Garratt, Peter J, Doecke, Christopher W, Weber, Jeffrey C, Paquette, Leo A
Published in Journal of organic chemistry (01.02.1986)
Published in Journal of organic chemistry (01.02.1986)
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