Candidate Selection and Preclinical Evaluation of N-tert-Butyl Isoquine (GSK369796), An Affordable and Effective 4-Aminoquinoline Antimalarial for the 21st Century
O’Neill, Paul M, Park, B. Kevin, Shone, Alison E, Maggs, James L, Roberts, Phillip, Stocks, Paul A, Biagini, Giancarlo A, Bray, Patrick G, Gibbons, Peter, Berry, Neil, Winstanley, Peter A, Mukhtar, Amira, Bonar-Law, Richard, Hindley, Stephen, Bambal, Ramesh B, Davis, Charles B, Bates, Martin, Hart, Timothy K, Gresham, Stephanie L, Lawrence, Ron M, Brigandi, Richard A, Gomez-delas-Heras, Federico M, Gargallo, Domingo V, Ward, Stephen A
Published in Journal of medicinal chemistry (12.03.2009)
Published in Journal of medicinal chemistry (12.03.2009)
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Uptake of Ozenoxacin and Other Quinolones in Gram-Positive Bacteria
López, Yuly, Muñoz, Laura, Gargallo-Viola, Domingo, Cantón, Rafael, Vila, Jordi, Zsolt, Ilonka
Published in International journal of molecular sciences (12.12.2021)
Published in International journal of molecular sciences (12.12.2021)
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Synthesis, Antimalarial Activity, and Preclinical Pharmacology of a Novel Series of 4′-Fluoro and 4′-Chloro Analogues of Amodiaquine. Identification of a Suitable “Back-Up” Compound for N-tert-Butyl Isoquine
O’Neill, Paul M, Shone, Alison E, Stanford, Deborah, Nixon, Gemma, Asadollahy, Eghbaleh, Park, B. Kevin, Maggs, James L, Roberts, Phil, Stocks, Paul A, Biagini, Giancarlo, Bray, Patrick G, Davies, Jill, Berry, Neil, Hall, Charlotte, Rimmer, Karen, Winstanley, Peter A, Hindley, Stephen, Bambal, Ramesh B, Davis, Charles B, Bates, Martin, Gresham, Stephanie L, Brigandi, Richard A, Gomez-de-las-Heras, Federico M, Gargallo, Domingo V, Parapini, Silvia, Vivas, Livia, Lander, Hollie, Taramelli, Donatella, Ward, Stephen A
Published in Journal of medicinal chemistry (09.04.2009)
Published in Journal of medicinal chemistry (09.04.2009)
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A murine model of falciparum-malaria by in vivo selection of competent strains in non-myelodepleted mice engrafted with human erythrocytes
Angulo-Barturen, Iñigo, Jiménez-Díaz, María Belén, Mulet, Teresa, Rullas, Joaquín, Herreros, Esperanza, Ferrer, Santiago, Jiménez, Elena, Mendoza, Alfonso, Regadera, Javier, Rosenthal, Philip J, Bathurst, Ian, Pompliano, David L, Gómez de las Heras, Federico, Gargallo-Viola, Domingo
Published in PloS one (21.05.2008)
Published in PloS one (21.05.2008)
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Improvement of detection specificity of Plasmodium‐infected murine erythrocytes by flow cytometry using autofluorescence and YOYO‐1
Jiménez‐Díaz, María Belén, Rullas, Joaquín, Mulet, Teresa, Fernández, Laura, Bravo, Carmen, Gargallo‐Viola, Domingo, Angulo‐Barturen, Iñigo
Published in Cytometry. Part A (01.09.2005)
Published in Cytometry. Part A (01.09.2005)
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Effect of the haematocrit layer geometry on Plasmodium falciparum static thin-layer in vitro cultures
Ferrer, Jordi, Rosal, Marina D, Vidal, Jaume M, Prats, Clara, Valls, Joaquim, Herreros, Esperanza A, López, Daniel, Gargallo, Domingo
Published in Malaria journal (08.10.2008)
Published in Malaria journal (08.10.2008)
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Microbiological profile of ozenoxacin
Morrissey, Ian, Cantón, Rafael, Vila, Jordi, Gargallo-Viola, Domingo, Zsolt, Ilonka, Garcia-Castillo, Maria, López, Yuly
Published in Future microbiology (01.06.2019)
Published in Future microbiology (01.06.2019)
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A novel class of fast‐acting antimalarial agents: Substituted 15‐membered azalides
Peric, Mihaela, Pešić, Dijana, Alihodžić, Sulejman, Fajdetić, Andrea, Herreros, Esperanza, Gamo, Francisco Javier, Angulo‐Barturen, Iñigo, Jiménez‐Díaz, María Belén, Ferrer‐Bazaga, Santiago, Martínez, María S., Gargallo‐Viola, Domingo, Mathis, Amanda, Kessler, Albane, Banjanac, Mihailo, Padovan, Jasna, Bencetić Mihaljević, Vlatka, Munic Kos, Vesna, Bukvić, Mirjana, Eraković Haber, Vesna, Spaventi, Radan
Published in British journal of pharmacology (01.01.2021)
Published in British journal of pharmacology (01.01.2021)
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Thermodynamic concepts in the study of microbial populations: age structure in Plasmodium falciparum infected red blood cells
Ferrer, Jordi, Prats, Clara, López, Daniel, Vidal-Mas, Jaume, Gargallo-Viola, Domingo, Guglietta, Antonio, Giró, Antoni
Published in PloS one (31.10.2011)
Published in PloS one (31.10.2011)
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Computer-assisted enhanced volumetric segmentation magnetic resonance imaging data using a mixture of artificial neural networks
Pérez de Alejo, Rigoberto, Ruiz-Cabello, Jesús, Cortijo, Manuel, Rodriguez, Ignacio, Echave, Imanol, Regadera, Javier, Arrazola, Juan, Avilés, Pablo, Barreiro, Pilar, Gargallo, Domingo, Graña, Manuel
Published in Magnetic resonance imaging (01.10.2003)
Published in Magnetic resonance imaging (01.10.2003)
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Quantitative measurement of Plasmodium‐infected erythrocytes in murine models of malaria by flow cytometry using bidimensional assessment of SYTO‐16 fluorescence
Jiménez‐Díaz, María Belén, Mulet, Teresa, Gómez, Vanesa, Viera, Sara, Alvarez, Angela, Garuti, Helena, Vázquez, Yolanda, Fernández, Alejandra, Ibáñez, Javier, Jiménez, Magdalena, Gargallo‐Viola, Domingo, Angulo‐Barturen, Iñigo
Published in Cytometry. Part A (01.03.2009)
Published in Cytometry. Part A (01.03.2009)
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Improved Murine Model of Malaria Using Plasmodium falciparum Competent Strains and Non-Myelodepleted NOD-scid IL2Rγnull Mice Engrafted with Human Erythrocytes
Jiménez-Díaz, María Belén, Mulet, Teresa, Viera, Sara, Gómez, Vanessa, Garuti, Helen, Ibáñez, Javier, Alvarez-Doval, Angela, Shultz, Leonard D., Martínez, Antonio, Gargallo-Viola, Domingo, Angulo-Barturen, Iñigo
Published in Antimicrobial Agents and Chemotherapy (01.10.2009)
Published in Antimicrobial Agents and Chemotherapy (01.10.2009)
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Antifungal Efficacy of GM237354, a Sordarin Derivative, in Experimental Oral Candidiasis in Immunosuppressed Rats
MARTINEZ, Antonio, REGADERA, Javier, JIMENEZ, Elena, SANTOS, Inmaculada, GARGALLO-VIOLA, Domingo
Published in Antimicrobial Agents and Chemotherapy (01.04.2001)
Published in Antimicrobial Agents and Chemotherapy (01.04.2001)
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Journal Article
In Vitro Pharmacodynamic Parameters of Sordarin Derivatives in Comparison with Those of Marketed Compounds against Pneumocystis carinii Isolated from Rats
AVILES, P, ALIOUAT, E.-M, MARTINEZ, A, DEI-CAS, E, HERREROS, E, DUJARDIN, L, GARGALLO-VIOLA, D
Published in Antimicrobial Agents and Chemotherapy (01.05.2000)
Published in Antimicrobial Agents and Chemotherapy (01.05.2000)
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Therapeutic Efficacies of GW471552 and GW471558, Two New Azasordarin Derivatives, against Pneumocystosis in Two Immunosuppressed-Rat Models
JIMENEZ, Elena, MARTINEZ, Antonio, ALIOUAT, El Moukhtar, CABALLERO, Jesus, DEI-CAS, Eduardo, GARGALLO-VIOLA, Domingo
Published in Antimicrobial Agents and Chemotherapy (01.08.2002)
Published in Antimicrobial Agents and Chemotherapy (01.08.2002)
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Journal Article
Antifungal Activities of Two New Azasordarins, GW471552 and GW471558, in Experimental Models of Oral and Vulvovaginal Candidiasis in Immunosuppressed Rats
MARTINEZ, Antonio, FERRER, Santiago, SANTOS, Inmaculada, JIMENEZ, Elena, SPARROWE, John, REGADERA, Javier, GOMEZ DE LAS HERAS, Federico, GARGALLO-VIOLA, Domingo
Published in Antimicrobial Agents and Chemotherapy (01.12.2001)
Published in Antimicrobial Agents and Chemotherapy (01.12.2001)
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Journal Article
Two-Step Synthesis of Achiral Dispiro-1,2,4,5-tetraoxanes with Outstanding Antimalarial Activity, Low Toxicity, and High-Stability Profiles
Ellis, Gemma L, Amewu, Richard, Sabbani, Sunil, Stocks, Paul A, Shone, Alison, Stanford, Deborah, Gibbons, Peter, Davies, Jill, Vivas, Livia, Charnaud, Sarah, Bongard, Emily, Hall, Charlotte, Rimmer, Karen, Lozanom, Sonia, Jesús, María, Gargallo, Domingo, Ward, Stephen A, O’Neill, Paul M
Published in Journal of medicinal chemistry (10.04.2008)
Published in Journal of medicinal chemistry (10.04.2008)
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Journal Article
Antibacterial Activities and Pharmacokinetics of E-4767 and E-5065, Two New 8-Chlorofluoroquinolones with a 7-Azetidin Ring Substituent
GARGALLO-VIOLA, Domingo, FERRER, Santiago, TUDELA, Encarna, ROBERT, Marta, COLL, Ramon, ROSER, Roberto, GUINEA, Jesus
Published in Antimicrobial Agents and Chemotherapy (01.11.2001)
Published in Antimicrobial Agents and Chemotherapy (01.11.2001)
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