Dynamic Combinatorial Selection of Molecules Capable of Inhibiting the (CUG) Repeat RNA−MBNL1 Interaction In Vitro: Discovery of Lead Compounds Targeting Myotonic Dystrophy (DM1)
Gareiss, Peter C, Sobczak, Krzysztof, McNaughton, Brian R, Palde, Prakash B, Thornton, Charles A, Miller, Benjamin L
Published in Journal of the American Chemical Society (03.12.2008)
Published in Journal of the American Chemical Society (03.12.2008)
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Journal Article
Selective Recognition of Alkyl Pyranosides in Protic and Aprotic Solvents
Palde, Prakash B, Gareiss, Peter C, Miller, Benjamin L
Published in Journal of the American Chemical Society (23.07.2008)
Published in Journal of the American Chemical Society (23.07.2008)
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Journal Article
Targeting the von Hippel–Lindau E3 Ubiquitin Ligase Using Small Molecules To Disrupt the VHL/HIF-1α Interaction
Buckley, Dennis L, Van Molle, Inge, Gareiss, Peter C, Tae, Hyun Seop, Michel, Julien, Noblin, Devin J, Jorgensen, William L, Ciulli, Alessio, Crews, Craig M
Published in Journal of the American Chemical Society (14.03.2012)
Published in Journal of the American Chemical Society (14.03.2012)
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Journal Article
Small-Molecule Inhibitors of the Interaction between the E3 Ligase VHL and HIF1α
Buckley, Dennis L., Gustafson, Jeffrey L., Van Molle, Inge, Roth, Anke G., Tae, Hyun Seop, Gareiss, Peter C., Jorgensen, William L., Ciulli, Alessio, Crews, Craig M.
Published in Angewandte Chemie (International ed.) (12.11.2012)
Published in Angewandte Chemie (International ed.) (12.11.2012)
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Journal Article
A Potent Activator of Melanogenesis Identified from Small‐Molecule Screening
McNaughton, Brian R., Gareiss, Peter C., Jacobs, Stacey E., Fricke, Alex F., Scott, Glynis A., Miller, Benjamin L.
Published in ChemMedChem (01.10.2009)
Published in ChemMedChem (01.10.2009)
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Journal Article
An analysis of original research contributions toward FDA-approved drugs
Patridge, Eric V., Gareiss, Peter C., Kinch, Michael S., Hoyer, Denton W.
Published in Drug discovery today (01.10.2015)
Published in Drug discovery today (01.10.2015)
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Journal Article
An allosteric site on MKP5 reveals a strategy for small-molecule inhibition
Gannam, Zira T K, Min, Kisuk, Shillingford, Shanelle R, Zhang, Lei, Herrington, James, Abriola, Laura, Gareiss, Peter C, Pantouris, Georgios, Tzouvelekis, Argyrios, Kaminski, Naftali, Zhang, Xinbo, Yu, Jun, Jamali, Haya, Ellman, Jonathan A, Lolis, Elias, Anderson, Karen S, Bennett, Anton M
Published in Science signaling (25.08.2020)
Published in Science signaling (25.08.2020)
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Journal Article
Identification of a Selective Small-Molecule Ligand for HIV-1 Frameshift-Inducing Stem-Loop RNA from an 11,325 Member Resin Bound Dynamic Combinatorial Library
McNaughton, Brian R, Gareiss, Peter C, Miller, Benjamin L
Published in Journal of the American Chemical Society (19.09.2007)
Published in Journal of the American Chemical Society (19.09.2007)
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Journal Article
Strategies for Recognition of Stem−Loop RNA Structures by Synthetic Ligands: Application to the HIV-1 Frameshift Stimulatory Sequence
Palde, Prakash B, Ofori, Leslie O, Gareiss, Peter C, Lerea, Jaclyn, Miller, Benjamin L
Published in Journal of medicinal chemistry (26.08.2010)
Published in Journal of medicinal chemistry (26.08.2010)
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Journal Article
Identification of a Novel Noncatalytic Bicarbonate Binding Site in Eubacterial β-Carbonic Anhydrase
Cronk, Jeff D, Rowlett, Roger S, Zhang, Kam Y. J, Tu, Chingkuang, Endrizzi, James A, Lee, Joseph, Gareiss, Peter C, Preiss, Jeffrey R
Published in Biochemistry (Easton) (11.04.2006)
Published in Biochemistry (Easton) (11.04.2006)
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Journal Article
A HaloTag-Based Small Molecule Microarray Screening Methodology with Increased Sensitivity and Multiplex Capabilities
Noblin, Devin J, Page, Charlotte M, Tae, Hyun Seop, Gareiss, Peter C, Schneekloth, John S, Crews, Craig M
Published in ACS chemical biology (21.12.2012)
Published in ACS chemical biology (21.12.2012)
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Journal Article
Allosteric Site Variants of Haemophilus influenzae β-Carbonic Anhydrase
Rowlett, Roger S, Tu, Chingkuang, Lee, Joseph, Herman, Ariel G, Chapnick, Douglas A, Shah, Shalini H, Gareiss, Peter C
Published in Biochemistry (Easton) (07.07.2009)
Published in Biochemistry (Easton) (07.07.2009)
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Journal Article
E3 Compounds and Methods for the Enhanced Degradation of Targeted Proteins and Other Polypeptides by an E3 Ubiquitin Ligase
SMITH IAN EDWARD DAVID, MOLLE INGE VAN, BUCKLEY DENNIS, CAMPOS SEBASTIEN ANDRE, ROTH ANKE G, TAE HYUN SEOP, GAREISS PETER C, MIAH AFJAL HUSSAIN, MICHEL JULIEN, HARLING JOHN DAVID, LE JOELLE, JORGENSEN WILLIAM, HOYER DENTIN WADE, CREWS CRAIG M, GUSTAFSON JEFFREY, CIULLI ALESSIO
Year of Publication 26.06.2024
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Year of Publication 26.06.2024
Patent
Ribosomal frameshifting: an emerging drug target for HIV
Gareiss, Peter C, Miller, Benjamin L
Published in Current opinion in investigational drugs (London, England : 2000) (01.02.2009)
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Published in Current opinion in investigational drugs (London, England : 2000) (01.02.2009)
Journal Article
E3 Compounds and Methods for the Enhanced Degradation of Targeted Proteins and Other Polypeptides by an E3 Ubiquitin Ligase
SMITH IAN EDWARD DAVID, MOLLE INGE VAN, BUCKLEY DENNIS, CAMPOS SEBASTIEN ANDRE, ROTH ANKE G, TAE HYUN SEOP, GAREISS PETER C, MIAH AFJAL HUSSAIN, MICHEL JULIEN, HARLING JOHN DAVID, LE JOELLE, JORGENSEN WILLIAM, HOYER DENTIN WADE, CREWS CRAIG M, GUSTAFSON JEFFREY, CIULLI ALESSIO
Year of Publication 14.09.2022
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Year of Publication 14.09.2022
Patent
Small-Molecule Inhibitors of the Interaction between the E3 Ligase VHL and HIF1a
Buckley, Dennis L., Gustafson, Jeffrey L., Van Molle, Inge, Roth, Anke G., Tae, Hyun Seop, Gareiss, Peter C., Jorgensen, William L., Ciulli, Alessio, Crews, Craig M.
Published in Angewandte Chemie International Edition (01.01.2012)
Published in Angewandte Chemie International Edition (01.01.2012)
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Journal Article
E3 Compounds and Methods for the Enhanced Degradation of Targeted Proteins and Other Polypeptides by an E3 Ubiquitin Ligase
SMITH IAN EDWARD DAVID, MOLLE INGE VAN, BUCKLEY DENNIS, CAMPOS SEBASTIEN ANDRE, ROTH ANKE G, TAE HYUN SEOP, GAREISS PETER C, MIAH AFJAL HUSSAIN, MICHEL JULIEN, HARLING JOHN DAVID, LE JOELLE, JORGENSEN WILLIAM, HOYER DENTIN WADE, CREWS CRAIG M, GUSTAFSON JEFFREY, CIULLI ALESSIO
Year of Publication 04.06.2020
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Year of Publication 04.06.2020
Patent
COMPOUNDS AND METHODS FOR THE ENHANCED DEGRADATION OF TARGETED PROTEINS AND OTHER POLYPEPTIDES BY AN E3 UBIQUITIN LIGASE
SMITH IAN EDWARD DAVID, MOLLE INGE VAN, BUCKLEY DENNIS, CAMPOS SEBASTIEN ANDRE, ROTH ANKE G, TAE HYUN SEOP, GAREISS PETER C, MIAH AFJAL HUSSAIN, MICHEL JULIEN, HARLING JOHN DAVID, LE JOELLE, JORGENSEN WILLIAM, HOYER DENTIN WADE, CREWS CRAIG M, GUSTAFSON JEFFREY, CIULLI ALESSIO
Year of Publication 29.01.2015
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Year of Publication 29.01.2015
Patent