Two Approaches to a Trifluoromethyl Triazole: A Fit-for-Purpose Trifluoromethylation in Flow-Mode and a Long-Term Decarboxylative Click Approach
Ayothiraman, Rajaram, Gangu, Aravind S, Bandaru, Durgarao, Guturi, Siva Krishna, Lakshminarasimhan, Thirumalai, Jaleel, Mohamed, Kanagavel, Kishorekumar, Rangaswamy, Sundaramurthy, Cuniere, Nicolas L, Zaretsky, Serge, Camacho, Kathryn, Eastgate, Martin D, Vaidyanathan, Rajappa
Published in Organic process research & development (21.02.2020)
Published in Organic process research & development (21.02.2020)
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Development of a Scalable Synthetic Route to BMS-986251. Part 1: Synthesis of the Cyclohexane Dicarboxylate Fragment
Kuppusamy, Sankar, Gangu, Aravind S, Kalidindi, Srinivas, Ponnusamy, Muthukrishnan, Tendulkar, Shankar, Venu, Alla, Palani, Senthil, Nagappan, Vedhachalam, Vinodini, Arun, Mudryk, Boguslaw, Rupasinghe, Sanjeewa, Joe, Candice L, Coombs, John R, Gallagher, William P, Kopp, Nathaniel, Gonzalez-Bobes, Francisco, Eastgate, Martin D, Vaidyanathan, Rajappa
Published in Organic process research & development (16.07.2021)
Published in Organic process research & development (16.07.2021)
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Development of a Scalable Synthetic Route to BMS-986251, Part 2: Synthesis of the Tricyclic Core and the API
Kalidindi, Srinivas, Gangu, Aravind S, Kuppusamy, Sankar, Sathasivam, Shunmugaraj, Shekarappa, Vijaykumar, Murugan, Saravanan, Bondigela, Sivasankar, Kandasamy, Moorthy, Ghanta, Kishore, Vinodini, Arun, Shrikant, Abhishek, Ramachandran, Ravikumar, Gallagher, William P, Kopp, Nathaniel, González-Bobes, Francisco, Eastgate, Martin D, Vaidyanathan, Rajappa
Published in Organic process research & development (16.07.2021)
Published in Organic process research & development (16.07.2021)
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Development of Continuous Flow Processes to Access Pyrrolo[2,1‑f][1,2,4]triazin-4-amine: An RSM for the Synthesis of Antiviral Drugs
Vasilev, Maksim, Gangu, Aravind S., Gajula, Praveen, Kaetzel, Nathaniel D., Natarajan, Vasudevan, Desai, Bimbisar, Sirasani, Gopal, Qu, Bo, Senanayake, Chris H.
Published in Organic process research & development (17.05.2024)
Published in Organic process research & development (17.05.2024)
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Development and Execution of an Ni(II)-Catalyzed Reductive Cross-Coupling of Substituted 2-Chloropyridine and Ethyl 3-Chloropropanoate
Nimmagadda, Sri Krishna, Korapati, Satish, Dasgupta, Debottam, Malik, Noormohamed Abdul, Vinodini, Arun, Gangu, Aravind S., Kalidindi, Srinivas, Maity, Prantik, Bondigela, Siva Sankar, Venu, Alla, Gallagher, William P., Aytar, Selin, González-Bobes, Francisco, Vaidyanathan, Rajappa
Published in Organic process research & development (19.06.2020)
Published in Organic process research & development (19.06.2020)
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Development of a Safer Continuous Flow Process for B 2 (OH) 4 -Mediated Chemoselective Reduction of Nitroarenes to Anilines
Revu, Omkar, Vasilev, Maksim, Gajula, Praveen, Kalikinidi, Nageswara Rao, Gadi, Madhusudhan Reddy, Zhao, Huiping, Gamage, Shanika M. P., Hibbert, Graham, Ravikumar, Ongolu, Gummidi, Lalitha, Nasipireddy, Venkatarathnam, Vinodini, Arun, Bietsch, Jonathan, Wang, Zhirui, Brown, Jack D., Sirasani, Gopal, Armstrong, Joseph D., Gangu, Aravind S., Qu, Bo, Senanayake, Chris H.
Published in Organic process research & development (12.09.2024)
Published in Organic process research & development (12.09.2024)
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Synthesis of Chiral 1,2-Amino Alcohol-Containing Compounds Utilizing Ruthenium-Catalyzed Asymmetric Transfer Hydrogenation of Unprotected α‑Ketoamines
Mangunuru, Hari P. R., Terrab, Leila, Janganati, Venumadhav, Kalikinidi, Nageswara Rao, Tenneti, Srinivasarao, Natarajan, Vasudevan, Shada, Arun D. R., Naini, Santhosh Reddy, Gajula, Praveen, Lee, Daniel, Samankumara, Lalith P., Mamunooru, Manasa, Jayaraman, Aravindan, Sahani, Rajkumar Lalji, Yin, Jinya, Hewa-Rahinduwage, Chathuranga C., Gangu, Aravind, Chen, Anji, Wang, Zhirui, Desai, Bimbisar, Yue, Tai Y., Wannere, Chaitanya S., Armstrong, Joseph D., Donsbach, Kai O., Sirasani, Gopal, Gupton, B. Frank, Qu, Bo, Senanayake, Chris H.
Published in Journal of organic chemistry (03.05.2024)
Published in Journal of organic chemistry (03.05.2024)
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Alternative Approach to the Large-Scale Synthesis of the Densely Functionalized Pyrrolidone BMT-415200
Rakshit, Souvik, Sathasivam, Shunmugaraj, Reddy, Raghurami, Rao, Saladi V., Shekarappa, Vijaykumar, Kandasamy, Moorthy, Jaleel, Mohamed, Murugan, Saravanan, Bhat, Anuradha, Subramani, Tamilarasan, Lakshminarasimhan, Thirumalai, Gangu, Aravind, Wisniewski, Steven R., Kopp, Nathaniel, Hale, Ian, Stevens, Jason M., Rosso, Victor W., Eastgate, Martin D., Vaidyanathan, Rajappa
Published in Organic process research & development (21.04.2023)
Published in Organic process research & development (21.04.2023)
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Facile and Scalable Methodology for the Pyrrolo[2,1‑f][1,2,4]triazine of Remdesivir
Roy, Sarabindu, Yadaw, Ajay, Roy, Subho, Sirasani, Gopal, Gangu, Aravind, Brown, Jack D, Armstrong, Joseph D, Stringham, Rodger W, Gupton, B. Frank, Senanayake, Chris H, Snead, David R
Published in Organic process research & development (21.01.2022)
Published in Organic process research & development (21.01.2022)
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