Combination of Docetaxel Plus Savolitinib in Refractory Cancer Patients: A Report on Phase I Trial
Kim, Seung Tae, Lee, Sujin, Park, Minhwa, Park, Se Hoon, Park, Joon Oh, Lim, Ho Yeong, Park, Young Suk, Kang, Won Ki, Gangolli, Esha A., Shin, Hyeongchan, Kim, Kyoung-Mee, Hollingsworth, Simon J., Mortimer, Peter G.S., Lee, Jeeyun
Published in Translational oncology (01.04.2019)
Published in Translational oncology (01.04.2019)
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1340 NDI-101150 is a potent and highly selective hematopoietic progenitor kinase 1 (HPK1) inhibitor that promotes a robust and broad anti-tumor immune response
Ciccone, David, Kuo, Fu-Shan, Boiko, Scott, Daigle, Scott, Carreiro, Samantha, Kaila, Neelu, Yau, Gene, Gangolli, Esha A, Levasseur, Denise, Srivastava, Bhaskar, Basile, Frank G, Loh, Christine
Published in Journal for immunotherapy of cancer (01.11.2023)
Published in Journal for immunotherapy of cancer (01.11.2023)
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751 Monotherapy results from an ongoing phase 1a dose escalation study of NDI-101150, a highly selective oral hematopoietic progenitor kinase 1 (HPK1) inhibitor
Sommerhalder, David, Noel, Marcus, Boiko, Scott, Daigle, Scott, Zhang, Xinyan, Fraser, Patricia, Hoerres, Amanda, Rana, Nawaid, Gangolli, Esha A, Basile, Frank G, Srivastava, Bhaskar, Sharma, Sunil, Balaraman, Rama, Gutierrez, Martin
Published in Journal for immunotherapy of cancer (01.11.2023)
Published in Journal for immunotherapy of cancer (01.11.2023)
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Journal Article
Reproductive Function in Protein Kinase Inhibitor-Deficient Mice
Belyamani, Mouna, Gangolli, Esha A., Idzerda, Rejean L.
Published in Molecular and Cellular Biology (01.06.2001)
Published in Molecular and Cellular Biology (01.06.2001)
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Phase 1/2 trial of the HPK1 inhibitor NDI-101150 as monotherapy and in combination with pembrolizumab: Clinical update
Noel, Marcus Smith, Demel, Kurt C., Srivastava, Bhaskar, Daigle, Scott R., Boiko, Scott, Hoerres, Amanda, Basile, Frank G., Zhang, Xinyan, Fraser, Patricia, Dasen, Sue, Chabas, Daria, Gangolli, Esha A., Balaraman, Rama, Sharma, Sunil, Gutierrez, Martin, Sommerhalder, David
Published in Journal of clinical oncology (01.06.2024)
Published in Journal of clinical oncology (01.06.2024)
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Abstract 445: Genomic characteristics and response to rucaparib and enzalutamide in the phase 1b RAMP study of metastatic castration-resistant prostate cancer (mCRPC) patients
Rao, Arpit, Ryan, Charles J., Morris, David, Assikis, Vasileios, Jha, Gautam, Ablaza, Adriel-John, Habeck, Jenn, Loehr, Andrea, Xiao, Jim, Gangolli, Esha A.
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Rucaparib plus enzalutamide in patients (pts) with metastatic castration-resistant prostate cancer (mCRPC): Pharmacokinetics (PK) and safety data from the phase Ib RAMP study
Rao, Arpit, Morris, David, Assikis, Vasily J., Jha, Gautam Gopalji, Ryan, Charles J., Ablaza, Adriel-John, Habeck, Jenn, Loehr, Andrea, Xiao, Jim, Gangolli, Esha A.
Published in Journal of clinical oncology (20.02.2021)
Published in Journal of clinical oncology (20.02.2021)
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Journal Article
Deficient Gene Expression in Protein Kinase Inhibitor α Null Mutant Mice
Gangolli, Esha A., Belyamani, Mouna, Muchinsky, Sara, Narula, Anita, Burton, Kimberly A., McKnight, G. Stanley, Uhler, Michael D., Idzerda, Rejean L.
Published in Molecular and Cellular Biology (01.05.2000)
Published in Molecular and Cellular Biology (01.05.2000)
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Phase 1 trial of the adenosine A 2A receptor antagonist inupadenant (EOS-850): Update on tolerability, and antitumor activity potentially associated with the expression of the A 2A receptor within the tumor
Buisseret, Laurence, Rottey, Sylvie, De Bono, Johann S., Migeotte, Ariane, Delafontaine, Brant, Manickavasagar, Thubeena, Martinoli, Chiara, Wald, Noémie, Rossetti, Maura, Gangolli, Esha A., Wiegert, Erol, McIntyre, Nicola, Lager, Joanne J., Machiels, Jean-Pascal H.
Published in Journal of clinical oncology (20.05.2021)
Published in Journal of clinical oncology (20.05.2021)
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MLN2480, an investigational oral pan-RAF kinase inhibitor, in patients (pts) with relapsed or refractory solid tumors: Phase I study
Rasco, Drew Warren, Olszanski, Anthony J., Patnaik, Amita, Espino, Guillermo, Neuwirth, Rachel, Faucette, Stephanie, Bargfrede, Michael, Gangolli, Esha A., Walker, Russell M, Kneissl, Michelle, Bozon, Viviana
Published in Journal of clinical oncology (20.05.2013)
Published in Journal of clinical oncology (20.05.2013)
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Abstract 3532: Preclinical-to-clinical translation of optimal schedule for MLN0128, an investigational novel small-molecule selective mTOR1/2 inhibitor, based on exposure-efficacy modeling
Patel, Mayankbhai, Staunton, Jocelyn, Mettetal, Jerome, Palani, Santhosh, Ecsedy, Jeffrey, Lu, Chuang, Barry, Elly, Westin, Eric, Manfredi, Mark, Shyu, Wej Chyi, Jessen, Katayoun, Gangolli, Esha A., Chakravarty, Arijit
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
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Clinical pharmacokinetics (PK) and translational PK-pharmacodynamic (PD) modeling and simulation to predict antitumor response of various dosing schedules to guide the selection of a recommended phase II dose (RP2D) and schedule for the investigational agent MLN0128
Patel, Chirag G., Patel, Mayank, Chakravarty, Arijit, Gangolli, Esha A., Barry, Elly, Westin, Eric H., Jessen, Katti, Chitnis, Shripad D., Infante, Jeffrey R., Gordon, Michael S., Macarulla, Teresa, Cervantes-Ruiperez, Andres, Jalal, Shadia Ibrahim, Venkatakrishnan, Karthik
Published in Journal of clinical oncology (20.05.2013)
Published in Journal of clinical oncology (20.05.2013)
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Phase I, dose-escalation study of the investigational drug TAK-733, an oral MEK inhibitor, in patients (pts) with advanced solid tumors
Adjei, Alex A., LoRusso, Patricia, Ribas, Antoni, Sosman, Jeffrey Alan, Pavlick, Anna C., Dy, Grace K., Zhou, Xiaofei, Gangolli, Esha A., Walker, Russell M, Kneissl, Michelle, Faucette, Stephanie, Neuwirth, Rachel, Bozon, Viviana
Published in Journal of clinical oncology (20.05.2013)
Published in Journal of clinical oncology (20.05.2013)
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Journal Article
GPCR-PROTEINS AND NUCLEIC ACIDS ENCODING SAME
SZEKERES, EDWARD, S, RASTELLI, LUCA, BURGESS, CATHERINE, E, GANGOLLI, ESHA, A., GANGOLLI, SMITHSON, GLENNDA, TCHERNEV, VELIZAR, T, VERNET, CORINE, A., M, GORSSE, WILLIAM, WOLENC, ADAM, R, ALSOBROOK, JOHN, P, CASMAN, STACIE, J, SHENOY, SURESH, PADIGARU, MURALIDHARA
Year of Publication 15.08.2002
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Year of Publication 15.08.2002
Patent
NOVEL GPCR-PROTEINS AND NUCLEIC ACIDS ENCODING SAME
SZEKERES, EDWARD, S, RASTELLI, LUCA, BURGESS, CATHERINE, E, GANGOLLI, ESHA, A., GANGOLLI, SMITHSON, GLENNDA, TCHERNEV, VELIZAR, T, VERNET, CORINE, A., M, GORSSE, WILLIAM, WOLENC, ADAM, R, ALSOBROOK, JOHN, P, CASMAN, STACIE, J, SHENOY, SURESH, PADIGARU, MURALIDHARA
Year of Publication 18.04.2002
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Year of Publication 18.04.2002
Patent
NOVEL GPCR-PROTEINS AND NUCLEIC ACIDS ENCODING SAME
SZEKERES, EDWARD, S, RASTELLI, LUCA, BURGESS, CATHERINE, E, GANGOLLI, ESHA, A., GANGOLLI, SMITHSON, GLENNDA, TCHERNEV, VELIZAR, T, VERNET, CORINE, A., M, GORSSE, WILLIAM, WOLENC, ADAM, R, ALSOBROOK, JOHN, P, CASMAN, STACIE, J, SHENOY, SURESH, PADIGARU, MURALIDHARA
Year of Publication 18.10.2001
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Year of Publication 18.10.2001
Patent
GPCR-PROTEINS AND NUCLEIC ACIDS ENCODING SAME
TCHERNEV, VELIZAR T, CASMAN, STACIE J, WOLENC, ADAM R, GANGOLLI, ESHA A., GANGOLLI, RASTELLI, LUCA, VERNET, CORINE A. M, SMITHSON, GLENNDA, GORSSE, WILLIAM, ALSOBROOK, JOHN P, BURGESS, CATHERINE E, SHENOY, SURESH, PADIGARU, MURALIDHARA, SZEKERES, EDWARD S
Year of Publication 18.10.2001
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Year of Publication 18.10.2001
Patent
Deficient Gene Expression in Protein Kinase Inhibitor α Null Mutant Mice
Gangolli, Esha A., Belyamani, Mouna, Muchinsky, Sara, Narula, Anita, Burton, Kimberly A., McKnight, G. Stanley, Uhler, Michael D., Idzerda, Rejean L.
Published in Molecular and cellular biology (2000)
Published in Molecular and cellular biology (2000)
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