Hindered dialkyl ether synthesis with electrogenerated carbocations
Xiang, Jinbao, Shang, Ming, Kawamata, Yu, Lundberg, Helena, Reisberg, Solomon H, Chen, Miao, Mykhailiuk, Pavel, Beutner, Gregory, Collins, Michael R, Davies, Alyn, Del Bel, Matthew, Gallego, Gary M, Spangler, Jillian E, Starr, Jeremy, Yang, Shouliang, Blackmond, Donna G, Baran, Phil S
Published in Nature (London) (01.09.2019)
Published in Nature (London) (01.09.2019)
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Strain-release amination
Gianatassio, Ryan, Lopchuk, Justin M., Wang, Jie, Pan, Chung-Mao, Malins, Lara R., Prieto, Liher, Brandt, Thomas A., Collins, Michael R., Gallego, Gary M., Sach, Neal W., Spangler, Jillian E., Zhu, Huichin, Zhu, Jinjiang, Baran, Phil S.
Published in Science (American Association for the Advancement of Science) (15.01.2016)
Published in Science (American Association for the Advancement of Science) (15.01.2016)
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A Radical Approach to Anionic Chemistry: Synthesis of Ketones, Alcohols, and Amines
Ni, Shengyang, Padial, Natalia M, Kingston, Cian, Vantourout, Julien C, Schmitt, Daniel C, Edwards, Jacob T, Kruszyk, Monika M, Merchant, Rohan R, Mykhailiuk, Pavel K, Sanchez, Brittany B, Yang, Shouliang, Perry, Matthew A, Gallego, Gary M, Mousseau, James J, Collins, Michael R, Cherney, Robert J, Lebed, Pavlo S, Chen, Jason S, Qin, Tian, Baran, Phil S
Published in Journal of the American Chemical Society (24.04.2019)
Published in Journal of the American Chemical Society (24.04.2019)
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Organic chemistry. Strain-release amination
Gianatassio, Ryan, Lopchuk, Justin M, Wang, Jie, Pan, Chung-Mao, Malins, Lara R, Prieto, Liher, Brandt, Thomas A, Collins, Michael R, Gallego, Gary M, Sach, Neal W, Spangler, Jillian E, Zhu, Huichin, Zhu, Jinjiang, Baran, Phil S
Published in Science (American Association for the Advancement of Science) (15.01.2016)
Published in Science (American Association for the Advancement of Science) (15.01.2016)
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Strain-Release Heteroatom Functionalization: Development, Scope, and Stereospecificity
Lopchuk, Justin M, Fjelbye, Kasper, Kawamata, Yu, Malins, Lara R, Pan, Chung-Mao, Gianatassio, Ryan, Wang, Jie, Prieto, Liher, Bradow, James, Brandt, Thomas A, Collins, Michael R, Elleraas, Jeff, Ewanicki, Jason, Farrell, William, Fadeyi, Olugbeminiyi O, Gallego, Gary M, Mousseau, James J, Oliver, Robert, Sach, Neal W, Smith, Jason K, Spangler, Jillian E, Zhu, Huichin, Zhu, Jinjiang, Baran, Phil S
Published in Journal of the American Chemical Society (01.03.2017)
Published in Journal of the American Chemical Society (01.03.2017)
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Modular radical cross-coupling with sulfones enables access to sp3-rich (fluoro)alkylated scaffolds
Merchant, Rohan R, Edwards, Jacob T, Tian, Qin, Kruszyk, Monika M, Bi, Cheng, Guanda, Che, Deng-Hui, Bao, Qiao Wenhua, Sun Lijie, Collins, Michael R, Fadeyi, Olugbeminiyi O, Gallego, Gary M, Mousseau, James J, Nuhant Philippe, Baran, Phil S
Published in Science (American Association for the Advancement of Science) (06.04.2018)
Published in Science (American Association for the Advancement of Science) (06.04.2018)
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A General Amino Acid Synthesis Enabled by Innate Radical Cross‐Coupling
Ni, Shengyang, Garrido‐Castro, Alberto F., Merchant, Rohan R., de Gruyter, Justine N., Schmitt, Daniel C., Mousseau, James J., Gallego, Gary M., Yang, Shouliang, Collins, Michael R., Qiao, Jennifer X., Yeung, Kap‐Sun, Langley, David R., Poss, Michael A., Scola, Paul M., Qin, Tian, Baran, Phil S.
Published in Angewandte Chemie International Edition (26.10.2018)
Published in Angewandte Chemie International Edition (26.10.2018)
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1,2-Difunctionalized bicyclo[1.1.1]pentanes: Long-sought-after mimetics for ortho / meta -substituted arenes
Zhao, Jin-Xin, Chang, Yu-Xuan, He, Chi, Burke, Benjamin J, Collins, Michael R, Del Bel, Matthew, Elleraas, Jeff, Gallego, Gary M, Montgomery, T Patrick, Mousseau, James J, Nair, Sajiv K, Perry, Matthew A, Spangler, Jillian E, Vantourout, Julien C, Baran, Phil S
Published in Proceedings of the National Academy of Sciences - PNAS (13.07.2021)
Published in Proceedings of the National Academy of Sciences - PNAS (13.07.2021)
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A Unifying Synthesis Approach to the C18-, C19-, and C20-Diterpenoid Alkaloids
Kou, Kevin G. M, Kulyk, Svitlana, Marth, Christopher J, Lee, Jack C, Doering, Nicolle A, Li, Beryl X, Gallego, Gary M, Lebold, Terry P, Sarpong, Richmond
Published in Journal of the American Chemical Society (04.10.2017)
Published in Journal of the American Chemical Society (04.10.2017)
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Palladium(ii)-catalyzed γ-selective hydroarylation of alkenyl carbonyl compounds with arylboronic acids
Matsuura, Rei, Jankins, Tanner C, Hill, David E, Yang, Kin S, Gallego, Gary M, Yang, Shouliang, He, Mingying, Wang, Fen, Marsters, Rohan P, McAlpine, Indrawan, Engle, Keary M
Published in Chemical science (Cambridge) (28.11.2018)
Published in Chemical science (Cambridge) (28.11.2018)
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Journal Article
A Unifying Synthesis Approach to the C-18-, C-19-, and C-20-Diterpenoid Alkaloids
Kou, Kevin G. M., Kulyk, Svitlana, Marth, Christopher J., Lee, Jack C., Doering, Nicolle A., Li, Beryl X., Gallego, Gary M., Lebold, Terry P., Sarpong, Richmond
Published in Journal of the American Chemical Society (04.10.2017)
Published in Journal of the American Chemical Society (04.10.2017)
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Multifaceted Substrate–Ligand Interactions Promote the Copper-Catalyzed Hydroboration of Benzylidenecyclobutanes and Related Compounds
Kang, Taeho, Erbay, Tuğçe G, Xu, Kane L, Gallego, Gary M, Burtea, Alexander, Nair, Sajiv K, Patman, Ryan L, Zhou, Ru, Sutton, Scott C, McAlpine, Indrawan J, Liu, Peng, Engle, Keary M
Published in ACS catalysis (06.11.2020)
Published in ACS catalysis (06.11.2020)
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Syntheses of Denudatine Diterpenoid Alkaloids: Cochlearenine, N‑Ethyl-1α-hydroxy-17-veratroyldictyzine, and Paniculamine
Kou, Kevin G. M, Li, Beryl X, Lee, Jack C, Gallego, Gary M, Lebold, Terry P, DiPasquale, Antonio G, Sarpong, Richmond
Published in Journal of the American Chemical Society (31.08.2016)
Published in Journal of the American Chemical Society (31.08.2016)
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Structure-Based Drug Design and Synthesis of PI3K alpha-Selective Inhibitor (PF-06843195)
Cheng, Hengmiao, Orr, Suvi T. M., Bailey, Simon, Brooun, Alexei, Chen, Ping, Deal, Judith G., Deng, Yali L., Edwards, Martin P., Gallego, Gary M., Grodsky, Neil, Huang, Buwen, Jalaie, Mehran, Kaiser, Stephen, Kania, Robert S., Kephart, Susan E., Lafontaine, Jennifer, Ornelas, Martha A., Pairish, Mason, Planken, Simon, Shen, Hong, Sutton, Scott, Zehnder, Luke, Almaden, Chau D., Bagrodia, Shubha, Falk, Matthew D., Gukasyan, Hovhannes J., Ho, Caroline, Kang, Xiaolin, Kosa, Rachel E., Liu, Ling, Spilker, Mary E., Timofeevski, Sergei, Visswanathan, Ravi, Wang, Zhenxiong, Meng, Fanxiu, Ren, Shijian, Shao, Li, Xu, Feng, Kath, John C.
Published in Journal of medicinal chemistry (14.01.2021)
Published in Journal of medicinal chemistry (14.01.2021)
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Correction to “Automated Nanomole-Scale Reaction Screening toward Benzoate Bioisosteres: A Photocatalyzed Approach to Highly Elaborated Bicyclo[1.1.1]Pentanes”
Mousseau, James J, Perry, Matthew A, Bundesmann, Mark W, Chinigo, Gary M, Choi, Chulho, Gallego, Gary M, Hicklin, Robert W, Hoy, Susan, Limburg, David C, Sach, Neal W, Zhang, Yuan
Published in ACS catalysis (18.02.2022)
Published in ACS catalysis (18.02.2022)
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A Copper-Mediated Conjugate Addition Approach to Analogues of Aconitine-Type Diterpenoid Alkaloids
Doering, Nicolle A, Kou, Kevin G. M, Norseeda, Krissada, Lee, Jack C, Marth, Christopher J, Gallego, Gary M, Sarpong, Richmond
Published in Journal of organic chemistry (19.10.2018)
Published in Journal of organic chemistry (19.10.2018)
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Cu-Catalyzed Hydroboration of Benzylidenecyclopropanes: Reaction Optimization, (Hetero)Aryl Scope, and Origins of Pathway Selectivity
Medina, Jose M, Kang, Taeho, Erbay, Tuğçe G, Shao, Huiling, Gallego, Gary M, Yang, Shouliang, Tran-Dubé, Michelle, Richardson, Paul F, Derosa, Joseph, Helsel, Ryan T, Patman, Ryan L, Wang, Fen, Ashcroft, Christopher P, Braganza, John F, McAlpine, Indrawan, Liu, Peng, Engle, Keary M
Published in ACS catalysis (06.12.2019)
Published in ACS catalysis (06.12.2019)
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Characterization of Specific N-alpha-Acetyltransferase 50 (Naa50) Inhibitors Identified Using a DNA Encoded Library
Kung, Pei-Pei, Bingham, Patrick, Burke, Benjamin J., Chen, Qiuxia, Cheng, Xuemin, Deng, Ya-Li, Dou, Dengfeng, Feng, Junli, Gallego, Gary M., Gehring, Michael R., Grant, Stephan K., Greasley, Samantha, Harris, Anthony R., Maegley, Karen A., Meier, Jordan, Meng, Xiaoyun, Montano, Jose L., Morgan, Barry A., Naughton, Brigitte S., Palde, Prakash B., Paul, Thomas A., Richardson, Paul, Sakata, Sylvie, Shaginian, Alex, Sonnenburg, William K., Subramanyam, Chakrapani, Timofeevski, Sergei, Wan, Jinqiao, Yan, Wen, Stewart, Albert E.
Published in ACS medicinal chemistry letters (11.06.2020)
Published in ACS medicinal chemistry letters (11.06.2020)
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